Somatostatina
La somatostatina es una hormona peptídica que inhibe la liberación de varias otras hormonas, incluyendo la hormona de crecimiento, insulina y glucagón. Actúa al unirse a los receptores de somatostatina, que son receptores acoplados a proteínas G expresados en varios tejidos. Los análogos de la somatostatina se utilizan en el tratamiento de la acromegalia, tumores neuroendocrinos y trastornos gastrointestinales. Estos análogos también son herramientas valiosas para estudiar la secreción y señalización hormonal. En CymitQuimica, ofrecemos una gama completa de análogos de somatostatina de alta calidad para apoyar su investigación en endocrinología, regulación hormonal y desarrollo terapéutico.
Se han encontrado 61 productos para "Somatostatina".
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L-796,778 acetate
L-796,778 acetate is a slective somatostatin receptor agonist with IC50 of 24nM for sst3, for sst1, sst2, sst4 and sst5, IC50 is >1000nM.Fórmula:C31H44N6O9Pureza:98%Forma y color:SoildPeso molecular:644.72Tau conotoxin CnVA
CAS:Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Fórmula:C72H116N24O17S4Forma y color:SolidPeso molecular:1718.1L-797,591 hydrochloride
L-797,591 HCl activates SSTR1, boosts p-ERK5 with AG1478, and enhances p38 phosphorylation, reversible by AG1478.Fórmula:C38H50ClN5O2Pureza:98.65% - >99.99%Forma y color:White SolidPeso molecular:644.30Anti-Somatostatin Antibody (9L93)
Anti-Somatostatin Antibody (9L93) is a Rabbit antibody targeting Somatostatin. Anti-Somatostatin Antibody (9L93) can be used in ELISA.Forma y color:Odour LiquidLanreotide
CAS:Lanreotide, a somatostatin analogue, suppresses GH/IGF-I hypersecretion in acromegaly patients. It also used to manage neuroendocrine tumours.Fórmula:C54H69N11O10S2Forma y color:SolidPeso molecular:1096.32CYN 154806 TFA
CAS:CYN 154806 TFA: cyclic octapeptide, selective somatostatin sst2 antagonist; pIC50: sst2 - 8.58, sst1 - 5.41, sst3 - 6.07, sst4 - 5.76, sst5 - 6.48.Fórmula:C58H69F3N12O16S2Pureza:99.7%Forma y color:SolidPeso molecular:1311.36Edotreotide
CAS:Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.Fórmula:C65H92N14O18S2Pureza:96.95%Forma y color:White SolidPeso molecular:1421.64Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Fórmula:C51H70N10O12S2Pureza:99.03% - 99.87%Forma y color:White SolidPeso molecular:1079.30Paltusotine
CAS:Paltusotine: nonpeptide SST2 agonist, orally bioavailable, regulates GH/IGF-1 in acromegaly.Fórmula:C27H22F2N4OPureza:99.91%Forma y color:SolidPeso molecular:456.49Pasireotide Acetate
CAS:The pKi of Pasireotide (SOM230) acetate for sst1, 2, 3, 4, and 5 were 8.2, 9.0, 9.1, less than 7.0, and 9.9, respectively.Cost-effective and quality-assured.Fórmula:C60H70N10O11Pureza:98.64% - 99.92%Forma y color:SolidPeso molecular:1107.26Ref: TM-TP2207
1mg90,00€2mg138,00€5mg236,00€10mg409,00€25mg745,00€50mg1.189,00€100mg1.684,00€200mg2.268,00€Somatostatin Impurity 2 (13-Dha) Trifluoroacetate
Fórmula:C76H102N18O18S2·C2HF3O2Peso molecular:1619.88 114.02BIM-23190 aceate
BIM-23190 aceate, a somatostatin analog, a selective agonist of SSTR2 and SSTR5. BIM-23190 can be used in cancer and acromegaly studies.Fórmula:C59H83N13O14S2Pureza:99.31%Forma y color:White SolidPeso molecular:1262.5FK962
CAS:FK962 is an somatostatin release enhancer , exerts cognitive-enhancing actions.Fórmula:C14H17FN2O2Pureza:99.89%Forma y color:SolidPeso molecular:264.3Ref: TM-T7829
2mg34,00€5mg52,00€1mL*10mM (DMSO)57,00€10mg82,00€25mg144,00€50mg200,00€100mg278,00€200mg389,00€L-803087
CAS:L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Fórmula:C25H29F2N5O3Pureza:99.37%Forma y color:White SolidPeso molecular:485.53Ref: TM-T11800
1mg50,00€5mg112,00€1mL*10mM (DMSO)126,00€10mg175,00€25mg366,00€50mg585,00€100mg928,00€200mg1.234,00€SSTR4 agonist 5
CAS:SSTR4 agonist5 (Compound 5) is an orally active agonist of the somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. It demonstrates good stability in human/rat liver microsomes and can inhibit mechanical hyperalgesia in rat models.Fórmula:C20H26N4OPeso molecular:338.447SST1 receptor antagonist-1
CAS:SST1 receptor antagonist-1 (Compound 23) is a selective antagonist of the somatostatin receptor 1 (SST1), showing a pKd of 9.11 for rSST1 and 8.79 for hSST1. This compound is applicable in research related to retinal and endocrine dysfunction, cancer, and neuropsychiatric disorders.Fórmula:C29H31F2N3O2Forma y color:SolidPeso molecular:491.57L-796778 acetate
CAS:L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.Fórmula:C31H44N6O9Forma y color:SolidPeso molecular:644.716SSTR5 antagonist 6
CAS:SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].Fórmula:C22H28ClN3O4Forma y color:SolidPeso molecular:433.93
