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Receptor de la hormona tiroidea (THR)

Receptor de la hormona tiroidea (THR)

Los receptores de hormonas tiroideas (THR) son receptores nucleares que median los efectos de las hormonas tiroideas, que son fundamentales para regular el metabolismo, el crecimiento y el desarrollo. La modulación de la actividad de los THR es importante en el tratamiento de trastornos tiroideos, síndromes metabólicos y ciertos tipos de cáncer. Los agonistas y antagonistas de THR se utilizan en la investigación para estudiar los roles fisiológicos y patológicos de las hormonas tiroideas. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de hormonas tiroideas de alta calidad para apoyar su investigación en endocrinología, metabolismo y regulación hormonal.

Se han encontrado 26 productos de "Receptor de la hormona tiroidea (THR)"

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  • PCO371

    CAS:
    <p>PCO371 (2,4-Imidazolidinedione, 1-(3,5-dimethyl-4-(2-((4-oxo-2-(4-(trifluoromethoxy)phenyl)-1,3,8-triazaspiro(4.5)dec-1-en-8-yl)sulfonyl)ethyl)phenyl)-5,5-</p>
    Fórmula:C29H32F3N5O6S
    Pureza:97.17% - 99.25%
    Forma y color:Solid
    Peso molecular:635.65
  • 3,5-Diiodothyropropionic acid

    CAS:
    <p>3,5-Diiodothyropropionic acid: thyroid hormone analog, boosts α-myosin mRNA, binds TRα1 &amp; TRβ1 (Ka: 2.40/M, 4.06/M).</p>
    Fórmula:C15H12I2O4
    Pureza:98.42%
    Forma y color:Solid
    Peso molecular:510.06
  • Osteostatin

    CAS:
    <p>Osteostatin, derived from parathyroid hormone-related protein (PTHrP) 107-111, has demonstrated properties conducive to bone repair in animal models presenting</p>
    Fórmula:C27H41N9O8
    Forma y color:Solid
    Peso molecular:619.67
  • NH-3

    CAS:
    <p>NH-3, an orally active THR antagonist with a 55 nM IC50, blocks thyroid hormone binding and cofactor recruitment.</p>
    Fórmula:C28H27NO6
    Pureza:97.79% - 99.40%
    Forma y color:Solid
    Peso molecular:473.52
  • Parathyroid hormone (1-34) (rat)

    CAS:
    <p>Parathyroid hormone (PTH) receptor agonist. Increases serum PTH levels and bone mass in rats.</p>
    Fórmula:C180H291N55O48S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:4057.74
  • DPC-AJ1951

    CAS:
    <p>Potent 14 amino acid peptide agonist of the parathyroid hormone (PTH) receptor (EC50 = 26 nM).</p>
    Fórmula:C76H127N23O19
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1666.98
  • THR-β agonist 2 diacetate


    <p>THR-β agonist 2 diacetate (Compound 3) is a potent THR-β agonist with potential applications in researching metabolic disorders such as obesity, hyperlipidemia, hypercholesterolemia, and diabetes, as well as other conditions like steatosis and non-alcoholic steatohepatitis (NASH), atherosclerosis, and other related diseases and conditions.</p>
    Forma y color:Odour Solid
  • DPC-AJ1951 TFA


    <p>DPC-AJ1951 TFA is a 14 amino acid peptide, potent PTH/PPR agonist, tested in bone resorption assays.</p>
    Fórmula:C78H128F3N23O21
    Forma y color:Solid
    Peso molecular:1781.02
  • Calcitonin, eel

    CAS:
    <p>Calcitonin from eel regulates calcium and is key in studying postmenopausal osteoporosis.</p>
    Fórmula:C146H241N43O47S2
    Pureza:98%
    Forma y color:White Powder
    Peso molecular:3414.91
  • Prepro-TRH-(160-169)

    CAS:
    <p>Prepro-TRH-(160-169), a pro-TRH peptide, enhances TRH-stimulated TSH secretion.</p>
    Fórmula:C54H75N11O18S
    Forma y color:Solid
    Peso molecular:1198.3
  • Taltirelin

    CAS:
    <p>Taltirelin (TA-0910) is at thyrotropin-releasing hormone receptor (TRH-R) superagonist (IC50 of 910 nM and EC50 of 36 nM for stimulating an increase in</p>
    Fórmula:C17H23N7O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:405.41
  • Eprotirome

    CAS:
    <p>Eprotirome (KB2115), a synthetic thyroid hormone mimetic, is a thyroid hormone receptor agonist.</p>
    Fórmula:C18H17Br2NO5
    Pureza:98.42% - 98.56%
    Forma y color:Solid
    Peso molecular:487.14
  • REVERSE T3

    CAS:
    <p>Reverse T3 (3,3',5'-triiodo-L-thyronine) inhibits the increase of sodium current generated by other thyroid hormone analogs in neonatal rat myocytes.</p>
    Fórmula:C15H12I3NO4
    Pureza:95.99% - 97.89%
    Forma y color:Powder
    Peso molecular:650.97
  • Resmetirom

    CAS:
    <p>Resmetirom (MGL-3196) is a THR-β agonist (EC50=0.21 μM), with high selectivity and oral activity. High-Quality, Low-Cost!</p>
    Fórmula:C17H12Cl2N6O4
    Pureza:99.05% - >99.99%
    Forma y color:Solid
    Peso molecular:435.22
  • Sobetirome

    CAS:
    <p>Sobetirome (IACS-010759) is a selective agonist of thyroid hormone receptor β (TRβ) and binds selectively to TRβ-1 (EC50: 0.16 μM).</p>
    Fórmula:C20H24O4
    Pureza:98.08% - 98.25%
    Forma y color:Solid
    Peso molecular:328.4
  • (D-Trp12,Tyr34)-pTH (7-34) amide (bovine) acetate


    <p>D-Trp12,Tyr34-pTH(7-34) (bovine) is a PTH antagonist with a Ki of 69 nM in bovine kidneys.</p>
    Pureza:96.84%
    Forma y color:Liquid
    Peso molecular:N/A
  • 3,3',5-Triiodothyronine-(tyrosine ring-13C6)

    CAS:
    <p>3,3',5-Triiodothyronine-(tyrosine ring-13C6) is the 13C labeled compound of 3,3',5-Triiodothyronine. 3,3',5-Triiodothyronine has a CAS number of 5817-39-0.</p>
    Fórmula:C4C11H12I3NO4
    Forma y color:Solid
    Peso molecular:656.93
  • Azetirelin

    CAS:
    <p>Azetirelin, as a TRH analog, has a more potent effect than TRH on the central nervous system.</p>
    Fórmula:C15H20N6O4
    Pureza:99.72%
    Forma y color:Solid
    Peso molecular:348.36
  • KAT681

    CAS:
    <p>KAT681 is a liver selective thyromimetic.</p>
    Fórmula:C24H22FNNaO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:462.429
  • Glutaurine aceate


    <p>Glutaurine aceate containing glutamine and taurine residues is an orally active hormone of the parathyroid.</p>
    Fórmula:C9H18N2O8S
    Pureza:98%
    Forma y color:Soild
    Peso molecular:314.31