Receptor de estrógeno / progestágeno
Los receptores de estrógenos y progestágenos son receptores hormonales nucleares que median los efectos del estrógeno y la progesterona, respectivamente. Estos receptores regulan varios procesos fisiológicos, incluyendo la función reproductiva, la densidad ósea y la salud cardiovascular. Los moduladores de los receptores de estrógenos y progestágenos se estudian extensamente por sus roles en la terapia de reemplazo hormonal, la anticoncepción y el tratamiento de cánceres hormonoresponsivos. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores de estrógenos y progestágenos de alta calidad para apoyar su investigación en endocrinología, salud reproductiva y biología del cáncer.
Se han encontrado 64 productos de "Receptor de estrógeno / progestágeno"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
(R)-Equol
CAS:(R)-Equol ((+)-Equol) is an ERα and ERβ agonist with Kis of 27.4 and 15.4 nM, respectively.Fórmula:C15H14O3Pureza:99.59%Forma y color:SolidPeso molecular:242.274,4'-Iminodiphenol
CAS:4,4'-Iminodiphenol (Leucoindophenol) is an inactive estrogen receptor ligand with a diphenylamine backbone.Fórmula:C12H11NO2Pureza:98.68%Forma y color:SolidPeso molecular:201.22Promestriene
CAS:Promestriene (3-propyl ethyl) (INN) is a synthetic estrogen and glucocorticoid used topically in a 1% cream formulation.Fórmula:C22H32O2Pureza:99.35%Forma y color:White SolidPeso molecular:328.49Ethynodiol diacetate
CAS:Ethynodiol diacetate (Ethynodiol acetate) is a synthetic progestational hormone used alone or in combination with estrogens as an oral contraceptive.Fórmula:C24H32O4Pureza:99.48% - 99.54%Forma y color:SolidPeso molecular:384.51Toremifene
CAS:Toremifene (GTx 006) is a selective estrogen-receptor modulator (SERM).Fórmula:C26H28ClNOPureza:99.77% - >99.99%Forma y color:White-To-Off-White SolidPeso molecular:405.96Gestrinone
CAS:Gestrinone (R 2323) 是一种合成类固醇激素，能够抑制平滑肌瘤(IC50:43.67 μM)，有用于子宫内膜异位症的研究潜力。Fórmula:C21H24O2Pureza:99.21%Forma y color:Light Yellow SolidPeso molecular:308.41SLU-PP-332
CAS:SLU-PP-332 is a pan-estrogen receptor-related receptor (ERR) agonist with high affinity for ERRα, ERRβ, and ERRγ with EC50 values of 98, 230, and 430 nM,Fórmula:C18H14N2O2Pureza:97.53% - 98.60%Forma y color:SoildPeso molecular:290.32Clomiphene citrate
CAS:Clomiphene citrate (NSC 35770) is a selective estrogen receptor modulator.Fórmula:C32H36ClNO8Pureza:98.67% - >99.99%Forma y color:White Crystalline PowderPeso molecular:598.1Dienestrol
CAS:Dienestrol (Restrol) is a synthetic and nonsteroidal estrogen, which is an estrogen receptor agonist.Fórmula:C18H18O2Pureza:96.73% - 98%Forma y color:Minute Needles From Dilute Alc SolidPeso molecular:266.33Giredestrant
CAS:Giredestrant (GDC-9545) is a potent oral anti-tumor ER antagonist competing with estradiol.Fórmula:C27H31F5N4OPureza:98.96% - 99.56%Forma y color:SolidPeso molecular:522.55Ref: TM-T11399
1mg105,00€5mg212,00€10mg334,00€25mg643,00€50mg1.018,00€100mg1.611,00€1mL*10mM (DMSO)245,00€Quinestrol
CAS:Quinestrol (Ethinylestradiol 3-cyclopentyl ether) is a synthetic estrogen, applied in hormone replacement therapy, and occasionally to use in cancer andFórmula:C25H32O2Pureza:99.36% - 99.72%Forma y color:SolidPeso molecular:364.52Elacestrant
CAS:Elacestrant (RAD1901) with IC50s of 48 and 870 nM for ERα and ERβ, respectively.Elacestrant is an orally available selective estrogen receptor degrader .Fórmula:C30H38N2O2Pureza:98.31%Forma y color:SolidPeso molecular:458.63Ref: TM-T13674
1mg124,00€5mg235,00€10mg376,00€25mg645,00€50mg913,00€100mg1.216,00€1mL*10mM (DMSO)235,00€Gestodene
CAS:Gestodene (WL 70) is a progestogen hormonal contraceptive.Fórmula:C21H26O2Pureza:98% - 99.68%Forma y color:White Crystalline SolidPeso molecular:310.43Mestranol
CAS:Mestranol (Devocin), a semisynthetic estrogen, is used as an estrogen receptor agonist and must be demethylated to be biologically active.Fórmula:C21H26O2Pureza:99.16%Forma y color:Crystals From Methanol Or Acetone SolidPeso molecular:310.43Ethisterone
CAS:Ethisterone (17α-Ethynyltestosterone) is a progestogen hormone.Fórmula:C21H28O2Pureza:97.96% - 99.50%Forma y color:Off-White PowderPeso molecular:312.45Panomifene TFA
Panomifene TFA（GYKl13504 TFA） is a antagonist of ERs with anticancer activity that can be used to study breast cancer and musculoskeletal diseases.Fórmula:C27H25F6NO4Pureza:99.74%Forma y color:SoildPeso molecular:541.48Altrenogest
CAS:Altrenogest (Allyltrenbolone)(A35957; RU2267), a progestogen, has structural relation with veterinary steroid trenbolone.Fórmula:C21H26O2Pureza:98.98% - 99.66%Forma y color:Slightly Yellow PowderPeso molecular:310.43Methylpiperidino pyrazole
CAS:Methylpiperidino pyrazole is an ERα inhibitor and can prevent the BPS-induced Rb phosphorylation and cell cycle progression.Fórmula:C29H31N3O3Pureza:98.84%Forma y color:SolidPeso molecular:469.57AC-186
CAS:AC-186 is an ERβ agonist with neuroprotective activity for the study of Parkinson's disease.
Fórmula:C18H17F3OPureza:99.53%Forma y color:SolidPeso molecular:306.32Endoxifen Z-isomer hydrochloride
CAS:Endoxifen Z-isomer hydrochloride (Endoxifen HCl) is the active metabolite of Tamoxifen, which is an effective and selective estrogen receptor antagonist.Fórmula:C25H28ClNO2Forma y color:SolidPeso molecular:409.95Bazedoxifene
CAS:Bazedoxifene is an orally active SERM against ERα and ERβ and inhibits IL-6/GP130, applied in postmenopausal osteoporosis and pancreatic cancer research.Fórmula:C30H34N2O3Pureza:98.79%Forma y color:SolidPeso molecular:470.61Nestoron
CAS:Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).Fórmula:C23H30O4Pureza:99.83% - 99.92%Forma y color:SolidPeso molecular:370.48Ulipristal
CAS:Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.Fórmula:C28H35NO3Pureza:99.82%Forma y color:SolidPeso molecular:433.584-Hydroxytamoxifen
CAS:4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.Fórmula:C26H29NO2Pureza:99.37% - 99.93%Forma y color:SolidPeso molecular:387.51Elacestrant dihydrochloride
CAS:Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM forFórmula:C30H40Cl2N2O2Pureza:99.59% - 99.99%Forma y color:SolidPeso molecular:531.56Ref: TM-T13675
1mg113,00€5mg225,00€10mg356,00€25mg598,00€50mg852,00€100mg1.153,00€1mL*10mM (DMSO)264,00€Medroxyprogesterone
CAS:Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.Fórmula:C22H32O3Pureza:99.18% - 99.51%Forma y color:Crystals From Chloroform SolidPeso molecular:344.49Desogestrel
CAS:Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.Fórmula:C22H30OPureza:99.8%Forma y color:Crystals SolidPeso molecular:310.47Ferrous Bisglycinate
CAS:Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.Fórmula:C4H8FeN2O4Pureza:≥95%Forma y color:SolidPeso molecular:203.96Norgestrel
CAS:Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.
Fórmula:C21H28O2Pureza:99.71% - 99.72%Forma y color:Crystals From Methanol White Crystalline PowderPeso molecular:312.45GSK5182
CAS:GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)Fórmula:C27H31NO3Pureza:97.63% - 99.42%Forma y color:SolidPeso molecular:417.54Ref: TM-T8370
1mg50,00€2mg71,00€5mg90,00€10mg144,00€25mg260,00€50mg394,00€100mg582,00€1mL*10mM (DMSO)108,00€SNG-1153
CAS:SNG-1153 is a estrogen receptor ER-alpha36 modulator.Fórmula:C21H17F3O5Pureza:99.74%Forma y color:SolidPeso molecular:406.35Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS:Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.Fórmula:C18H18O3Pureza:99.85% - 99.96%Forma y color:SolidPeso molecular:282.33Ref: TM-T9800
1mg93,00€5mg182,00€10mg269,00€25mg429,00€50mg610,00€100mg820,00€200mg1.099,00€1mL*10mM (DMSO)172,00€Estradiol dipropionate
CAS:Estradiol dipropionate (17-Beta-Estradiol-3,17-Dipropionate) is a synthetic ester, specifically the 3, 17-dipropanoyl ester, of the natural estrogen, estradiol.Fórmula:C24H32O4Pureza:99.68%Forma y color:SolidPeso molecular:384.51WAY-200070
CAS:WAY-200070 is a specific agonist of estrogen receptor β (ERRβ, IC50: 2.3 nM).Fórmula:C13H8BrNO3Pureza:99.45% - 99.75%Forma y color:SolidPeso molecular:306.11Ref: TM-T3958
2mg42,00€5mg62,00€10mg96,00€25mg188,00€50mg311,00€100mg502,00€200mg715,00€1mL*10mM (DMSO)67,00€PROTAC ERRα ligand 2
CAS:PROTAC ERRα ligand 2 is an estrogen-related receptor α (ERRα) inverse agonist( IC50 : 5.67 nM)Fórmula:C20H13F6NO4Pureza:≥95%Forma y color:SolidPeso molecular:445.31Ref: TM-T5835
1mg43,00€5mg96,00€10mg116,00€25mg198,00€50mg299,00€100mg449,00€200mg627,00€1mL*10mM (DMSO)96,00€DY131
CAS:DY131 (DY-131) is a novel selective agonist of ERRβ and ERRγ.Fórmula:C18H21N3O2Pureza:98.65% - 99.66%Forma y color:SolidPeso molecular:311.38Brilanestrant
CAS:Brilanestrant (GDC-0810) is a selective estrogen receptor degrader (IC50: 0.7 nM).Fórmula:C26H20ClFN2O2Pureza:99.07% - 99.17%Forma y color:Solid PowderPeso molecular:446.9Ref: TM-T5118
1mg50,00€2mg73,00€5mg101,00€10mg142,00€25mg245,00€50mg405,00€100mg582,00€1mL*10mM (DMSO)120,00€FLTX1
CAS:FLTX1, a Tamoxifen derivative, fluoresces to mark estrogen receptors and acts as a strong antiestrogen in breast cancer without affecting the uterus.Fórmula:C31H28N4O4Pureza:98.42%Forma y color:SolidPeso molecular:520.58Ref: TM-T8984
1mg55,00€5mg119,00€10mg182,00€25mg313,00€50mg442,00€100mg627,00€200mg845,00€1mL*10mM (DMSO)137,00€Hexestrol
CAS:Hexestrol (Hexanoestrol) binds to ERα and ERβ with EC50 of 0.07 nM and 0.175 nM, respectively.Fórmula:C18H22O2Pureza:98.93% - 99.2%Forma y color:Needles From Benzene Thin Plates From Dil Alc Crystalline SolidPeso molecular:270.37Propyl pyrazole triol
CAS:PPT is a selective ERα agonist with 410x higher affinity than for ERβ.Fórmula:C24H22N2O3Pureza:97.86%Forma y color:SolidPeso molecular:386.44Ref: TM-T16566
1mg43,00€5mg93,00€10mg133,00€25mg250,00€50mg378,00€100mg570,00€200mg800,00€1mL*10mM (DMSO)90,00€Bazedoxifene acetate
CAS:Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).Fórmula:C32H38N2O5Pureza:99.24% - 99.97%Forma y color:SolidPeso molecular:530.67Ref: TM-T2544
5mg44,00€10mg57,00€25mg86,00€50mg105,00€100mg152,00€200mg219,00€500mg358,00€1200mg618,00€1mL*10mM (DMSO)50,00€AZD9496
CAS:AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.Fórmula:C25H25F3N2O2Pureza:97.28% - 98.47%Forma y color:SolidPeso molecular:442.47Ref: TM-T3975
1mg52,00€2mg73,00€5mg110,00€10mg178,00€25mg334,00€50mg494,00€100mg712,00€1mL*10mM (DMSO)105,00€SR 19881
CAS:SR 19881 is a full agonist of ERRγ(EC50 value of 0.39 μM in a binding assay and an EC50 value of 4.7 μM in a cell-based assay).Fórmula:C19H24N2O2Pureza:98.54%Forma y color:SolidPeso molecular:312.41Ref: TM-T7904
1mg97,00€2mg149,00€5mg202,00€10mg324,00€25mg548,00€50mg785,00€100mg1.074,00€1mL*10mM (DMSO)220,00€Serba-2
CAS:Serba-2 is an agonist of benzopyran selective estrogen receptor beta.Fórmula:C18H18O3Pureza:>99.99%Forma y color:SolidPeso molecular:282.33Fulvestrant-d3
Fulvestrant-d3 is a isotope labeled compound of Fulvestrant.an estrogen receptor (ER) antagonist and GPR30 agonist thatinduces apoptosis and autophagy.
Fórmula:C32H47F5O3SForma y color:SolidPeso molecular:609.79Endoxifen E-isomer hydrochloride
CAS:Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).Fórmula:C25H28ClNO2Pureza:98%Forma y color:SolidPeso molecular:409.95Erteberel
CAS:Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.Fórmula:C18H18O3Pureza:99.46%Forma y color:SolidPeso molecular:282.33OP-1074
CAS:OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.Fórmula:C29H31NO4Pureza:98%Forma y color:SolidPeso molecular:457.56DS20362725
CAS:DS20362725 is a selective estrogen-related receptor alpha (ERRα) agonist, commonly used in the study of metabolic disorders.Fórmula:C19H22N2O2Pureza:99.34%Forma y color:SolidPeso molecular:310.39Capesaris
CAS:Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.Fórmula:C19H13F2NO3Pureza:99.65%Forma y color:SolidPeso molecular:341.31ERRγ Inverse Agonist 1
CAS:ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].Fórmula:C30H38Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:529.54Bisphenol Z
CAS:Bisphenol Z is a bisphenol compound and high-performance monomer used in advanced engineering plastics, having antagonistic activity towards ERα.Fórmula:C18H20O2Pureza:99.88%Forma y color:SolidPeso molecular:268.35Norethisterone enanthate
CAS:Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.Fórmula:C27H38O3Pureza:99.23%Forma y color:SolidPeso molecular:410.59ERRα antagonist-1
CAS:ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα).Fórmula:C21H19N3S2Pureza:99.66%Forma y color:SolidPeso molecular:377.53SIM-688
CAS:SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).Fórmula:C34H31F3N2O2Pureza:99.56%Forma y color:SolidPeso molecular:556.62NXT629
CAS:NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.Fórmula:C35H39N5O3SPureza:99.07% - 99.07%Forma y color:SolidPeso molecular:609.78Estrogen receptor antagonist 8
CAS:Estrogen Receptor Antagonist 8 is an ER antagonist with anti-uterine activity and may be used in the study of ovarian dysfunction.CASNETIN SODIUM (CasN)Fórmula:C25H21N3O4Pureza:98.48%Forma y color:SolidPeso molecular:427.45Zindoxifene
CAS:Zindoxifene (D 16726) is an anti-estrogenic compound with antitumor activity that can be used in studies of breast and prostate cancer.Fórmula:C21H21NO4Pureza:98.99%Forma y color:SolidPeso molecular:351.4Palazestrant
CAS:Palazestrant, an antiestrogen and antineoplastic agent, effectively targets ER+/HER2+ cancer when used in conjunction with a HER2 inhibitor.Fórmula:C28H36FN3OPureza:97.55%Forma y color:SolidPeso molecular:449.6Ref: TM-T72945
1mg93,00€5mg150,00€10mg215,00€25mg358,00€50mg517,00€100mg707,00€1mL*10mM (DMSO)166,00€LY88074
CAS:LY88074, a raloxifene analog sans basic side chain, is an ERβ agonist (EC50 = 232 nM) that promotes uterine cell growth.
Fórmula:C21H14O4SPureza:98.31%Forma y color:SolidPeso molecular:362.4H3B-6545
CAS:H3B-6545 is a selective and oral estrogen receptor covalent antagonist (SERCA) used in the research of metastatic ER-positive, HER2-negative breast cancer.Fórmula:C30H29F4N5O2Forma y color:SolidPeso molecular:567.58ERRα antagonist-2
CAS:ERRα antagonist-2 is an estrogen-related receptor α inverse agonist, inhibiting migration and invasion in ER-negative MDA-MB-231,breast cancer.Fórmula:C19H16N2O6SPureza:99.26%Forma y color:SolidPeso molecular:400.41(E/Z)-GSK5182
CAS:GSK5182 is a racemic mix of (E/Z) isomers, a selective ERRγ inverse agonist (IC50: 79 nM), and induces ROS in liver cancer.Fórmula:C27H31NO3Pureza:97.58%Forma y color:SolidPeso molecular:417.54Ref: TM-T7709
1mg77,00€5mg167,00€10mg260,00€25mg477,00€50mg707,00€100mg1.063,00€1mL*10mM (DMSO)177,00€ERB-196
CAS:Erb-196 is an estrogen receptor-receptor agonist with non-steroidal selectivity.Fórmula:C17H10FNO2Pureza:98%Forma y color:SolidPeso molecular:279.27
![Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT9800.webp&w=3840&q=75)
