Receptor de estrógeno / progestágeno
Los receptores de estrógenos y progestágenos son receptores hormonales nucleares que median los efectos del estrógeno y la progesterona, respectivamente. Estos receptores regulan varios procesos fisiológicos, incluyendo la función reproductiva, la densidad ósea y la salud cardiovascular. Los moduladores de los receptores de estrógenos y progestágenos se estudian extensamente por sus roles en la terapia de reemplazo hormonal, la anticoncepción y el tratamiento de cánceres hormonoresponsivos. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores de estrógenos y progestágenos de alta calidad para apoyar su investigación en endocrinología, salud reproductiva y biología del cáncer.
Se han encontrado 71 productos para "Receptor de estrógeno / progestágeno".
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Propyl pyrazole triol
CAS:PPT is a selective ERα agonist with 410x higher affinity than for ERβ.Fórmula:C24H22N2O3Pureza:97.86%Forma y color:SolidPeso molecular:386.44Ref: TM-T16566
1mg43,00€1mL*10mM (DMSO)90,00€5mg93,00€10mg133,00€25mg250,00€50mg378,00€100mg570,00€200mg800,00€Bazedoxifene acetate
CAS:Bazedoxifene acetate (WAY-TES 424) is a novel selective estrogen receptor modulator (SERM).Fórmula:C32H38N2O5Pureza:99.24% - 99.97%Forma y color:White SolidPeso molecular:530.67Ref: TM-T2544
1200mgA consultar5mg44,00€1mL*10mM (DMSO)50,00€10mg57,00€25mg86,00€50mg105,00€100mg152,00€200mg219,00€500mg358,00€AZD9496
CAS:AZD9496 is an orally available selective estrogen receptor(ERα) antagonist, with potential antineoplastic activity.Fórmula:C25H25F3N2O2Pureza:97.28% - 98.47%Forma y color:Yellow SolidPeso molecular:442.47Ref: TM-T3975
1mg52,00€2mg73,00€1mL*10mM (DMSO)105,00€5mg110,00€10mg178,00€25mg334,00€50mg494,00€100mg712,00€H3B-5942
CAS:H3B-5942 belongs to a class of ERα antagonists referred to as selective estrogen receptor covalent antagonists (SERCA).Fórmula:C31H34N4O2Pureza:98.06% - ≥95%Forma y color:SolidPeso molecular:494.63Ref: TM-T5633
1mg49,00€5mg105,00€1mL*10mM (DMSO)110,00€10mg164,00€25mg306,00€50mg439,00€100mg583,00€200mg785,00€Ulipristal
CAS:Ulipristal is a selective SPRM for emergency contraception after an unprotected intercourse or contraceptive failure.Fórmula:C28H35NO3Pureza:99.82%Forma y color:SolidPeso molecular:433.58PHTPP
CAS:PHTPP is a selective ERβ antagonist.Fórmula:C20H11F6N3OPureza:98.81% - 99.57%Forma y color:Red SolidPeso molecular:423.314-Hydroxytamoxifen
CAS:4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.Fórmula:C26H29NO2Pureza:99.37% - 99.93%Forma y color:SolidPeso molecular:387.51Nestoron
CAS:Nestoron (Segesterone Acetate), a synthetic progestin, is a high-affinity agonist of the progesterone receptor (EC50: 10.3 nM).Fórmula:C23H30O4Pureza:99.83% - 99.92%Forma y color:SolidPeso molecular:370.48Elacestrant dihydrochloride
CAS:Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM forFórmula:C30H40Cl2N2O2Pureza:99.59% - 99.99%Forma y color:SolidPeso molecular:531.56Ref: TM-T13675
1mg113,00€5mg225,00€1mL*10mM (DMSO)264,00€10mg356,00€25mg598,00€50mg852,00€100mg1.153,00€Medroxyprogesterone
CAS:Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.Fórmula:C22H32O3Pureza:99.18% - 99.51%Forma y color:SolidPeso molecular:344.49Fulvestrant-D3
Fulvestrant-d3 is a isotope labeled compound of Fulvestrant.an estrogen receptor (ER) antagonist and GPR30 agonist thatinduces apoptosis and autophagy.Fórmula:C32H47F5O3SForma y color:White SolidPeso molecular:609.79Endoxifen E-isomer hydrochloride
CAS:Endoxifen E-isomer hydrochloride (E-Endoxifen hydrochloride) , a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).Fórmula:C25H28ClNO2Pureza:98%Forma y color:SolidPeso molecular:409.95NXT629
CAS:NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.Fórmula:C35H39N5O3SPureza:99.07% - 99.07%Forma y color:SolidPeso molecular:609.78OP-1074
CAS:OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.Fórmula:C29H31NO4Pureza:98%Forma y color:SolidPeso molecular:457.56Bisphenol Z
CAS:Bisphenol Z is a bisphenol compound and high-performance monomer used in advanced engineering plastics, having antagonistic activity towards ERα.Fórmula:C18H20O2Pureza:99.88%Forma y color:White SolidPeso molecular:268.35Norethisterone enanthate
CAS:Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.Fórmula:C27H38O3Pureza:99.23%Forma y color:SolidPeso molecular:410.59SIM-688
CAS:SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).Fórmula:C34H31F3N2O2Pureza:99.56%Forma y color:SolidPeso molecular:556.62Erteberel
CAS:Erteberel (LY500307) is a potent, selective estrogen receptor β agonist with EC50 of 0.66 nM, 32-fold selectivity against estrogen receptor α. Phase 2.Fórmula:C18H18O3Pureza:99.46%Forma y color:SolidPeso molecular:282.33BHPI
CAS:BHPI is a potent ERα inhibitor, activating UPR and blocking protein synthesis with an IC50 value. It depletes EnR Ca(2+) via PLCγ in ERα(+) cancer cells.Fórmula:C21H17NO3Pureza:99.85%Forma y color:White SolidPeso molecular:331.36ERRγ Inverse Agonist 1
CAS:ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].Fórmula:C30H38Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:529.54
