
Receptor de estrógeno / progestágeno
Los receptores de estrógenos y progestágenos son receptores hormonales nucleares que median los efectos del estrógeno y la progesterona, respectivamente. Estos receptores regulan varios procesos fisiológicos, incluyendo la función reproductiva, la densidad ósea y la salud cardiovascular. Los moduladores de los receptores de estrógenos y progestágenos se estudian extensamente por sus roles en la terapia de reemplazo hormonal, la anticoncepción y el tratamiento de cánceres hormonoresponsivos. En CymitQuimica, ofrecemos una gama completa de moduladores de receptores de estrógenos y progestágenos de alta calidad para apoyar su investigación en endocrinología, salud reproductiva y biología del cáncer.
Se han encontrado 49 productos de "Receptor de estrógeno / progestágeno"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Serba-2
CAS:<p>Serba-2 is an agonist of benzopyran selective estrogen receptor beta.</p>Fórmula:C18H18O3Pureza:>99.99%Forma y color:SolidPeso molecular:282.334-Hydroxytamoxifen
CAS:<p>4-Hydroxytamoxifen (ICI 79280) is the active metabolite of Tamoxifen, an estrogen receptor modulator (SERM) with selective and oral potency.</p>Fórmula:C26H29NO2Pureza:99.37% - 99.93%Forma y color:SolidPeso molecular:387.51Ulipristal acetate
CAS:<p>Ulipristal acetate (CDB-2914) is an oral selective progesterone modulator used for emergency contraception and suppressing uterine growths.</p>Fórmula:C30H37NO4Pureza:98.83% - 99.94%Forma y color:SolidPeso molecular:475.62Elacestrant dihydrochloride
CAS:<p>Elacestrant dihydrochloride (DA-DKRAD1901 dihydrochloride) is an orally available selective estrogen receptor degrader with IC50s of 48 for ERα and 870 nM for</p>Fórmula:C30H40Cl2N2O2Pureza:99.59% - >99.99%Forma y color:SolidPeso molecular:531.56Medroxyprogesterone
CAS:<p>Medroxyprogesterone is used in the treatment of renal carcinoma. It is a synthetic progestational hormone used in veterinary practice as an estrus regulator.</p>Fórmula:C22H32O3Pureza:99.18% - 99.51%Forma y color:Crystals From Chloroform SolidPeso molecular:344.49Desogestrel
CAS:<p>Desogestrel (Cerazette) is a synthetic progestational hormone used often as the progestogenic component of combined oral contraceptive agents.</p>Fórmula:C22H30OPureza:99.8%Forma y color:Crystals SolidPeso molecular:310.47Ferrous Bisglycinate
CAS:<p>Ferrous Bisglycinate (Bisglycine iron(II) salt) is used in the fortification of infant formulations and foods.</p>Fórmula:C4H8FeN2O4Pureza:≥95%Forma y color:SolidPeso molecular:203.96Norgestrel
CAS:<p>Norgestrel (WY-3707), a synthetic progestin, is used for contraception and hinders LH/FSH, thickens mucus, and slows ova transit.</p>Fórmula:C21H28O2Pureza:99.71% - 99.72%Forma y color:Crystals From Methanol White Crystalline PowderPeso molecular:312.45GSK5182
CAS:<p>GSK5182 is a highly selective inverse estrogen-related receptor γ agonist (IC50 : 79 nM)</p>Fórmula:C27H31NO3Pureza:97.63% - 99.42%Forma y color:SolidPeso molecular:417.54SNG-1153
CAS:<p>SNG-1153 is a estrogen receptor ER-alpha36 modulator.</p>Fórmula:C21H17F3O5Pureza:99.74%Forma y color:SolidPeso molecular:406.35Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel-
CAS:<p>Cyclopenta[c][1]benzopyran-8-ol, 1,2,3,3a,4,9b-hexahydro-4-(4-hydroxyphenyl)-, (3aR,4S,9bS)-rel- is an estrogen receptor beta (ERβ) agonist.</p>Fórmula:C18H18O3Pureza:99.85% - 99.96%Forma y color:SolidPeso molecular:282.33Fulvestrant-d3
<p>Fulvestrant-d3 is a isotope labeled compound of Fulvestrant.an estrogen receptor (ER) antagonist and GPR30 agonist thatinduces apoptosis and autophagy.</p>Fórmula:C32H47F5O3SForma y color:SolidPeso molecular:609.79NXT629
CAS:<p>NXT629 is a PPAR-α antagonist with anticancer activity, inhibiting PPARδ, and can be used in ovarian cancer and melanoma research.</p>Fórmula:C35H39N5O3SPureza:99.07% - 99.07%Forma y color:SolidPeso molecular:609.78OP-1074
CAS:<p>OP-1074 is a pure antiestrogen and a selective degrader of ER, shows specific antiestrogenic activity for ERα and ERβ.</p>Fórmula:C29H31NO4Pureza:98%Forma y color:SolidPeso molecular:457.56ERRγ Inverse Agonist 1
CAS:<p>ERRγ Inverse Agonist 1 (Compound 12) is a potent, selective and orally bioavailable Estrogen-related Receptor grammar (ERRγ) inverse agonist (IC 50=40 nM) [1].</p>Fórmula:C30H38Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:529.54SIM-688
CAS:<p>SIM-688 is a selective and orally active estrogen receptor inhibitor of NF-κB transcriptional activity (IC50 = 122 nM in HAECT-1 cells).</p>Fórmula:C34H31F3N2O2Pureza:99.56%Forma y color:SolidPeso molecular:556.62Bisphenol Z
CAS:<p>Bisphenol Z is a bisphenol compound and high-performance monomer used in advanced engineering plastics, having antagonistic activity towards ERα.</p>Fórmula:C18H20O2Pureza:99.88%Forma y color:SolidPeso molecular:268.35ERRα antagonist-1
CAS:<p>ERRα antagonist-1 (ERR+/- antagonist-1) is a high-affinity, selective antagonist of the estrogen-related receptor α (ERRα).</p>Fórmula:C21H19N3S2Pureza:99.66%Forma y color:SolidPeso molecular:377.53Capesaris
CAS:<p>Capesaris (GTX-758) is an oral estrogen receptor α agonist, used in prostate cancer research.</p>Fórmula:C19H13F2NO3Pureza:99.65%Forma y color:SolidPeso molecular:341.31Norethisterone enanthate
CAS:<p>Norethisterone enanthate (NSC-9564) is a long-acting parenteral progestogen with antigonadotropic effects.</p>Fórmula:C27H38O3Pureza:99.23%Forma y color:SolidPeso molecular:410.59
