
Receptor de vasopresina
Los receptores de vasopresina son una familia de receptores acoplados a proteínas G que median los efectos de la vasopresina, una hormona involucrada en la regulación del equilibrio hídrico, la presión arterial y la función renal. Los agonistas y antagonistas de los receptores de vasopresina se estudian por su papel en el tratamiento de afecciones como la diabetes insípida, la hiponatremia y la insuficiencia cardíaca. Estos receptores también son objetivos importantes en la investigación sobre el equilibrio de líquidos y la salud cardiovascular. En CymitQuimica, ofrecemos una selección de moduladores de receptores de vasopresina de alta calidad para apoyar su investigación en endocrinología, nefrología y biología cardiovascular.
Se han encontrado 44 productos de "Receptor de vasopresina"
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Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Forma y color:SolidPeso molecular:1347.5Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Fórmula:C30H32ClN3O8SPureza:98.46% - 99.89%Forma y color:SolidPeso molecular:630.11Balovaptan
CAS:<p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>Fórmula:C22H24ClN5OPureza:99.88%Forma y color:SolidPeso molecular:409.91Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Fórmula:C110H161N31O27S2Pureza:98%Forma y color:SolidPeso molecular:2413.78(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:<p>V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.</p>Fórmula:C52H74N14O12S2Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:1151.38Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:<p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>Fórmula:C49H70N14O12S2Pureza:98%Forma y color:SolidPeso molecular:1111.3d[Cha4]-AVP
CAS:<p>Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.</p>Fórmula:C50H71N13O11S2Pureza:98%Forma y color:SolidPeso molecular:1094.31d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Fórmula:C47H67N11O11S2Pureza:98%Forma y color:SolidPeso molecular:1026.2d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Fórmula:C52H72F3N13O13S2Forma y color:SolidPeso molecular:1208.33Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:<p>Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent</p>Fórmula:C45H63N15O11S2Forma y color:SolidPeso molecular:1054.21[Asu1,6-Arg8]Vasopressin
CAS:<p>[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.</p>Fórmula:C48H68N14O12Forma y color:SolidPeso molecular:1033.14(Phe2,Orn8)-Oxytocin acetate
<p>(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.</p>Fórmula:C44H69N13O13S2Forma y color:SolidPeso molecular:1052.23Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Fórmula:C48H77N13O13S2Forma y color:SolidPeso molecular:1108.33Endolide F
<p>Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.</p>Fórmula:C25H32N4O6Peso molecular:484.23218D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Fórmula:C49H68F3N11O13S2Forma y color:SolidPeso molecular:1140.25(Phe2,Orn8)-Oxytocin
CAS:<p>(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.</p>Fórmula:C42H65N13O11S2Forma y color:SolidPeso molecular:992.18(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:<p>Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.</p>Fórmula:C54H76N14O11Forma y color:SolidPeso molecular:1097.27[8-L-arginine] deaminovasopressin
CAS:<p>[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .</p>Fórmula:C46H64N14O13S2Forma y color:SolidPeso molecular:1085.22Velmupressin acetate
CAS:<p>Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).</p>Fórmula:C44H64ClN11O10S2Pureza:98%Forma y color:SolidPeso molecular:1006.63d[Leu4,Lys8]-VP acetate
<p>d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.</p>Fórmula:C49H71N11O13S2Pureza:98.86%Forma y color:SolidPeso molecular:1086.28

