Receptor de vasopresina
Los receptores de vasopresina son una familia de receptores acoplados a proteínas G que median los efectos de la vasopresina, una hormona involucrada en la regulación del equilibrio hídrico, la presión arterial y la función renal. Los agonistas y antagonistas de los receptores de vasopresina se estudian por su papel en el tratamiento de afecciones como la diabetes insípida, la hiponatremia y la insuficiencia cardíaca. Estos receptores también son objetivos importantes en la investigación sobre el equilibrio de líquidos y la salud cardiovascular. En CymitQuimica, ofrecemos una selección de moduladores de receptores de vasopresina de alta calidad para apoyar su investigación en endocrinología, nefrología y biología cardiovascular.
Se han encontrado 44 productos de "Receptor de vasopresina"
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Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Fórmula:C110H161N31O27S2Pureza:98%Forma y color:SolidPeso molecular:2413.78[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Fórmula:C48H69N13O11S2Pureza:98%Forma y color:SolidPeso molecular:1068.27Val9-Oxytocin
CAS:<p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>Fórmula:C46H72N12O12S2Pureza:98%Forma y color:SolidPeso molecular:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:<p>(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].</p>Fórmula:C52H76N14O11S2Pureza:98%Forma y color:SolidPeso molecular:1137.38V1a/V2 antagonist 1
<p>V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.</p>Fórmula:C25H26ClN5O3Forma y color:SolidPeso molecular:479.96Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Fórmula:C27H34N4O3Pureza:99.33%Forma y color:SolidPeso molecular:462.58Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Fórmula:C46H65N15O12S2Pureza:98%Forma y color:White PowderPeso molecular:1084.23Atosiban
CAS:<p>Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.</p>Fórmula:C43H67N11O12S2Pureza:98%Forma y color:SolidPeso molecular:994.19Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Fórmula:C26H31N3O4Pureza:98.13% - 99.66%Forma y color:SolidPeso molecular:449.54d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Fórmula:C52H75N13O13S2Pureza:99.86%Forma y color:SolidPeso molecular:1154.37Atosiban acetate
CAS:<p>Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.</p>Fórmula:C45H71N11O14S2Pureza:99.84% - 99.92%Forma y color:SolidPeso molecular:1054.24Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Fórmula:C43H77N17O12S2Pureza:99.79%Forma y color:SolidPeso molecular:1088.32LIXIVAPTAN
CAS:<p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>Fórmula:C27H21ClFN3O2Pureza:98.36%Forma y color:SolidPeso molecular:473.93Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Fórmula:C48H68N14O14S2Pureza:98.84% - >99.99%Forma y color:SolidPeso molecular:1129.26Tolvaptan
CAS:<p>Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.</p>Fórmula:C26H25ClN2O3Pureza:99.78% - >99.99%Forma y color:SolidPeso molecular:448.94Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Fórmula:C32H26N4O2·HClPureza:98.33% - 99.86%Forma y color:SolidPeso molecular:535.04RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Fórmula:C25H28ClN3O2Pureza:99.74%Forma y color:SolidPeso molecular:437.96Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Fórmula:C27H29N3O2Pureza:98.98% - 99.12%Forma y color:SolidPeso molecular:427.54Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Fórmula:C46H65N13O11S2Pureza:99.65%Forma y color:SolidPeso molecular:1040.22Felypressin acetate
CAS:<p>Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.</p>Fórmula:C48H69N13O13S2Pureza:97.06%Forma y color:SolidPeso molecular:1100.27
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