Receptor de vasopresina
Los receptores de vasopresina son una familia de receptores acoplados a proteínas G que median los efectos de la vasopresina, una hormona involucrada en la regulación del equilibrio hídrico, la presión arterial y la función renal. Los agonistas y antagonistas de los receptores de vasopresina se estudian por su papel en el tratamiento de afecciones como la diabetes insípida, la hiponatremia y la insuficiencia cardíaca. Estos receptores también son objetivos importantes en la investigación sobre el equilibrio de líquidos y la salud cardiovascular. En CymitQuimica, ofrecemos una selección de moduladores de receptores de vasopresina de alta calidad para apoyar su investigación en endocrinología, nefrología y biología cardiovascular.
Se han encontrado 44 productos de "Receptor de vasopresina"
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Terlipressin Acetate
CAS:<p>Terlipressin Acetate, a highly selective vasopressin V1 receptor agonist, on OGD/R-induced damage in intestinal epithelial cells (IEC-6).</p>Fórmula:C56H82N16O19S2Pureza:98.50% - 99.69%Forma y color:SolidPeso molecular:1347.5Nelivaptan
CAS:<p>Nelivaptan (SR 149415) is a vasopressin V1b receptor antagonist that can eliminate CHS-induced GE damage.Cost-effective and quality-assured.</p>Fórmula:C30H32ClN3O8SPureza:98.46% - 99.89%Forma y color:SolidPeso molecular:630.11Balovaptan
CAS:<p>Balovaptan (RG7314), a potent brain-penetrant hV1a receptor antagonist, Ki: 1 nM for hV1a, aids autism research.</p>Fórmula:C22H24ClN5OPureza:99.88%Forma y color:SolidPeso molecular:409.91(D-Arg8)-Inotocin
CAS:<p>'(D-Arg8)-Inotocin is a potent, selective, and competitive antagonist of the vasopressin receptor (V 1a R), exhibiting a binding affinity (K i) of 1.3 nM.</p>Fórmula:C39H68N14O11S2Pureza:98%Forma y color:SolidPeso molecular:973.17d[Cha4]-AVP
CAS:<p>Potent human V1B vasopressin receptor agonist; Ki: V1B=1.2 nM; increases ACTH, corticosterone; low vasopressor effect.</p>Fórmula:C50H71N13O11S2Pureza:98%Forma y color:SolidPeso molecular:1094.31(d(CH2)51,Tyr(Me)2,Arg8)-Vasopressin
CAS:<p>V1A receptor antagonist; blocks vasopressin & oxytocin, lowers Ca²⁺ levels (IC50: 5/30 nM); long-acting antivasopressor; anxiolytic in dorsal hippocampus.</p>Fórmula:C52H74N14O12S2Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:1151.38d[Leu4,Lys8]-VP
CAS:<p>Vasopressin V1B agonist; Ki: 0.16nM V1B, 64nM oxytocin; weak antidiuretic/vasopressor; minimal oxytocic action.</p>Fórmula:C47H67N11O11S2Pureza:98%Forma y color:SolidPeso molecular:1026.2d[Cha4]-AVP TFA
<p>d[Cha4]-AVP TFA: potent, selective V1b agonist, K i 1.2 nM, favors V1b over V1a, V2, oxytocin receptors.</p>Fórmula:C52H72F3N13O13S2Forma y color:SolidPeso molecular:1208.33Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin
CAS:<p>Desamino(D-3-(3′-pyridyl)-Ala2,Arg8)-Vasopressin, a synthetic analog of vasopressin (AVP), acts as a weak agonist at the antidiuretic receptor but is a potent</p>Fórmula:C45H63N15O11S2Forma y color:SolidPeso molecular:1054.21[Asu1,6-Arg8]Vasopressin
CAS:<p>[Asu1,6-Arg8]Vasopressin, a vasopressin agonist, boosts cAMP and ACTH release in cultured rat pituitary cells.</p>Fórmula:C48H68N14O12Forma y color:SolidPeso molecular:1033.14(Phe2,Orn8)-Oxytocin acetate
<p>(Phe2,Orn8)-Oxytocin acetate: V1 agonist with EC50 of 280 nM for rabbit epididymis contractility.</p>Fórmula:C44H69N13O13S2Forma y color:SolidPeso molecular:1052.23Selepressin acetate
<p>Selepressin acetate is a useful organic compound for research related to life sciences and the catalog number is T73654.</p>Fórmula:C48H77N13O13S2Forma y color:SolidPeso molecular:1108.33(Phe2,Orn8)-Oxytocin
CAS:<p>(Phe2,Orn8)-Oxytocin: Selective V1 agonist, induces rabbit epididymis contractility, EC50=280 nM.</p>Fórmula:C42H65N13O11S2Forma y color:SolidPeso molecular:992.18D[LEU4,LYS8]-VP TFA
<p>D[LEU4,LYS8]-VP TFA: V1b receptor agonist; K_i: 0.16 nM (rat), 0.52 nM (human), 1.38 nM (mouse); weak antidiuretic/vasopressor/oxytocic.</p>Fórmula:C49H68F3N11O13S2Forma y color:SolidPeso molecular:1140.25(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin
CAS:<p>Potent VP V1R antagonist, lowers rat MAP: '(Phenylac1,D-Tyr(Et)2,Lys6,Arg8,des-Gly9)-Vasopressin'.</p>Fórmula:C54H76N14O11Forma y color:SolidPeso molecular:1097.27[8-L-arginine] deaminovasopressin
CAS:<p>[8-L-arginine] deaminovasopressin (dAVP) is a vasopressin analog [1] .</p>Fórmula:C46H64N14O13S2Forma y color:SolidPeso molecular:1085.22Endolide F
<p>Endolide F (Compound 2) is a proline-containing lactone that serves as a moderate antagonist of the arginine vasopressin V1A receptor.</p>Fórmula:C25H32N4O6Peso molecular:484.23218Velmupressin acetate
CAS:<p>Potent, selective, short-acting peptidic V2R agonist; EC50: 0.07 nM (hV2R), 0.02 nM (rV2R).</p>Fórmula:C44H64ClN11O10S2Pureza:98%Forma y color:SolidPeso molecular:1006.63d[Leu4,Lys8]-VP acetate
<p>d[Leu4,Lys8]-VP acetate: Vasopressin V1b agonist. Ki: rat 0.16 nM, human 0.52 nM, mouse 1.38 nM. Low antidiuretic/vasopressor effects.</p>Fórmula:C49H71N11O13S2Pureza:98.86%Forma y color:SolidPeso molecular:1086.28Dp[Tyr(methyl)2,Arg8]-Vasopressin
CAS:<p>Dp[Tyr(Me)2,Arg8]-Vasopressin is a non-selective antagonist of the peptide arginine vasopressin V1b receptor [1].</p>Fórmula:C49H70N14O12S2Pureza:98%Forma y color:SolidPeso molecular:1111.3Invopressin
CAS:<p>Invopressin (Compound 42), a vasopressin V1A receptor partial agonist (EC50: 1.0 nM), is utilized in research related to cirrhosis conditions such as bacterial</p>Fórmula:C110H161N31O27S2Pureza:98%Forma y color:SolidPeso molecular:2413.78[Deamino-Pen1,Val4,D-Arg8]-vasopressin
CAS:<p>[Deamino-Pen1,Val4,D-Arg8]-vasopressin (AVP-A) is an antagonist of arginine-vasopressin (AVP).</p>Fórmula:C48H69N13O11S2Pureza:98%Forma y color:SolidPeso molecular:1068.27Val9-Oxytocin
CAS:<p>Val9-Oxytocin, an Oxytocin analog where Gly9 is substituted with Val9 [1], functions as a complete antagonist of the vasopressin (V1a) receptor.</p>Fórmula:C46H72N12O12S2Pureza:98%Forma y color:SolidPeso molecular:1049.27(d(CH2)51,Tyr(Me)2,Dab5,Arg8)-Vasopressin
CAS:<p>(d(CH2)5[Tyr(Me)2, Dab5]AVP), a vasopressin V1a receptor-specific antagonist, demonstrates a pA2 value of 6.71 [1].</p>Fórmula:C52H76N14O11S2Pureza:98%Forma y color:SolidPeso molecular:1137.38V1a/V2 antagonist 1
<p>V1a/V2 antagonist 1 (Compound 18j) is an orally active dual-target antagonist of V1a and V2 receptors, exhibiting high binding affinity toward these receptors [Ki values are hV1a: 0.13 nM, hV2: 0.53 nM, and mV1a: 0.5 nM; IC50 for hV1a is 2.2 nM]. This compound can inhibit oxytocin-induced scratching behavior in mice.</p>Fórmula:C25H26ClN5O3Forma y color:SolidPeso molecular:479.96Fedovapagon
CAS:<p>Fedovapagon (VA106483) is a pressin V2 receptor (V2R) agonist for the study of overactive bladder syndrome.</p>Fórmula:C27H34N4O3Pureza:99.33%Forma y color:SolidPeso molecular:462.58Argipressin
CAS:<p>Argipressin is a vasoconstrictive and antidiuretic hormone, binding to V1 receptors with Kd ~1.4 nM in rat heart and aortic cells.</p>Fórmula:C46H65N15O12S2Pureza:98%Forma y color:White PowderPeso molecular:1084.23Atosiban
CAS:<p>Atosiban (RW22164), an oxytocin/vasopressin inhibitor, halts premature labor as an intravenous tocolytic, reducing uterine contractions rapidly.</p>Fórmula:C43H67N11O12S2Pureza:98%Forma y color:SolidPeso molecular:994.19Fuscoside
CAS:<p>Fuscoside (OPC-21268) is a non-peptide arginine vasopressin (AVP) receptor VI antagonist with an IC50 value of 0.4 μM.Cost-effective and quality-assured.</p>Fórmula:C26H31N3O4Pureza:98.13% - 99.66%Forma y color:SolidPeso molecular:449.54d[Cha4]-AVP acetate(500170-27-4 free base)
<p>'d[Cha4]-AVP acetate: strong V1B agonist, weak on V1A/Oxytocin/V2. Boosts ACTH, corticosterone; low blood pressure effect.'</p>Fórmula:C52H75N13O13S2Pureza:99.86%Forma y color:SolidPeso molecular:1154.37Atosiban acetate
CAS:<p>Atosiban acetate (RW22164) is an inhibitor of the hormones oxytocin and vasopressin.</p>Fórmula:C45H71N11O14S2Pureza:99.84% - 99.92%Forma y color:SolidPeso molecular:1054.24Conopressin S acetate(111317-90-9 free base)
<p>Conopressin S acetate(111317-90-9 free base) (Con-S acetate) is a natural product isolated from Conus striatus, shows high affinity with vasopressin V1b</p>Fórmula:C43H77N17O12S2Pureza:99.79%Forma y color:SolidPeso molecular:1088.32LIXIVAPTAN
CAS:<p>Lixivaptan (VPA-985) is an orally active and selective vasopressin receptor V2 antagonist(Ki = 2.3 nM)</p>Fórmula:C27H21ClFN3O2Pureza:98.36%Forma y color:SolidPeso molecular:473.93Desmopressin acetate (16679-58-6 free base)
CAS:<p>Desmopressin (16679-58-6), a synthetic vasopressin analog, treats nocturia, enuresis, and diabetes insipidus by reducing urine production.</p>Fórmula:C48H68N14O14S2Pureza:98.84% - >99.99%Forma y color:SolidPeso molecular:1129.26Tolvaptan
CAS:<p>Tolvaptan (OPC-41061) is an orally bioavailable, selective, arginine vasopressin receptor 2 (V2, AVPR2) antagonist that can be used to treat hyponatremia.</p>Fórmula:C26H25ClN2O3Pureza:99.78% - >99.99%Forma y color:SolidPeso molecular:448.94Conivaptan hydrochloride
CAS:<p>Conivaptan hydrochloride (Vaprisol) is an orally active vasopressin V2 and V1A receptor antagonist, used in the therapy of hypervolemic hyponatremia and</p>Fórmula:C32H26N4O2·HClPureza:98.33% - 99.86%Forma y color:SolidPeso molecular:535.04RG7713
CAS:<p>RG7713 (RO 5028442) has been used in trials studying Autistic Disorder.</p>Fórmula:C25H28ClN3O2Pureza:99.74%Forma y color:SolidPeso molecular:437.96Mozavaptan
CAS:<p>Mozavaptan (OPC-31260) is a competitive vasopressin receptor antagonist for both V1 and V2 receptors with IC50 of 1.2 μM and 14 nM, respectively.</p>Fórmula:C27H29N3O2Pureza:98.98% - 99.12%Forma y color:SolidPeso molecular:427.54Felypressin
CAS:<p>Felypressin, a Lypressin analog with a phenylalanine substitution, acts as a vasoconstrictor with less antidiuretic effect.</p>Fórmula:C46H65N13O11S2Pureza:99.65%Forma y color:SolidPeso molecular:1040.22Felypressin acetate
CAS:<p>Felypressin acetate (PLV-2) is an agonist of vasopressin 1 and acts on all arginine vasopressin receptors 1AS.</p>Fórmula:C48H69N13O13S2Pureza:97.06%Forma y color:SolidPeso molecular:1100.27OPC-51803
CAS:<p>OPC-51803 is an orally available nonapeptidylpressor (AVP) V(2) receptor selective agonist for the treatment of urinary incontinence and nocturia.</p>Fórmula:C26H32ClN3O2Pureza:98.93% - >99.99%Forma y color:SolidPeso molecular:454TASP0390325
CAS:<p>TASP0390325, a potent and orally active V1B receptor antagonist, has antidepressant and anxiolytic activities in rodents.</p>Fórmula:C25H30Cl2FN5O4Pureza:98.62%Forma y color:SolidPeso molecular:554.44RGH-122
CAS:<p>RGH-122 (compound 43), characterized as an orally active, potent, and selective hV1a receptor antagonist, demonstrates significant affinity with a K i value of 0.3 nM and an IC 50 of 0.9 nM. It exhibits microsomal stability, indicated by a CL int value of 13/28/25 μL/min/mg [1].</p>Fórmula:C24H25ClN4O3Forma y color:SolidPeso molecular:452.93Elsovaptan
CAS:<p>Elsovaptan is an antagonist of the vasopressin receptor and is applicable for research in Alzheimer's disease.</p>Fórmula:C19H20ClN5O2Forma y color:SolidPeso molecular:385.847
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