
Receptor de andrógenos
El receptor de andrógenos (AR) es un receptor hormonal nuclear que se activa al unirse a andrógenos, como la testosterona y la dihidrotestosterona. Este receptor juega un papel crucial en el desarrollo y mantenimiento de las características masculinas, así como en la regulación de varios procesos fisiológicos, incluyendo el crecimiento muscular, la libido y la densidad ósea. Los inhibidores del receptor de andrógenos son ampliamente estudiados en el contexto del cáncer de próstata, donde la señalización del AR a menudo está sobreexpresada. En CymitQuimica, ofrecemos una gama de moduladores del receptor de andrógenos de alta calidad para apoyar su investigación en endocrinología, biología del cáncer y regulación hormonal.
Se han encontrado 229 productos de "Receptor de andrógenos"
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Darolutamide
CAS:Darolutamide (BAY-1841788) is an androgen receptor (AR) antagonist that blocks AR nuclear translocation (Ki: 11 nM).Fórmula:C19H19ClN6O2Pureza:97.36% - >99.99%Forma y color:SolidPeso molecular:398.85Ref: TM-T6915
1mg49,00€2mg70,00€5mg105,00€10mg166,00€25mg264,00€50mg378,00€100mg540,00€200mg772,00€1mL*10mM (DMSO)106,00€Dimethylcurcumin
CAS:Dimethylcurcumin (ASC-J9) (ASC-J9) is an androgen receptor degradation enhancer.Fórmula:C23H24O6Pureza:97.36% - 98.96%Forma y color:SolidPeso molecular:396.43Testosterone acetate
CAS:Testosterone acetate (NSC-523836) is a hormone with in vitro antitumor activity.Fórmula:C21H30O3Pureza:99.6%Forma y color:White To Off-White Crystalline PowderPeso molecular:330.46GSK-2881078
CAS:GSK-2881078 is a selective androgen receptor modulato (SARM) that is being evaluated for effects on muscle growth and strength in subjects with muscle wasting.Fórmula:C14H13F3N2O2SPureza:98.16% - 98.81%Forma y color:SolidPeso molecular:330.33MI-136
CAS:MI-136 inhibits expression of androgen receptor (AR) target genes that DHT induced.Fórmula:C23H21F3N6SPureza:98.63% - 99.12%Forma y color:SolidPeso molecular:470.51Ref: TM-T6889
1mg47,00€5mg87,00€10mg147,00€25mg279,00€50mg472,00€100mg730,00€200mg1.017,00€1mL*10mM (DMSO)97,00€Nandrolone phenylpropionate
CAS:Nandrolone phenylpropionate (Nandrolone phenpropionate) is an androgen receptor agonist. It mainly used to treat women with breast cancer and osteoporosisFórmula:C27H34O3Pureza:99.2% - 99.46%Forma y color:White Or Milky Crystalline PowderPeso molecular:406.56YK11
CAS:YK11 is an androgen receptor partial agonist that activates androgen receptor transcriptional activity in HEK293 cells overexpressing androgen receptors when used at a concentration of 0.1 μM, with osteogenic activity.Fórmula:C25H34O6Pureza:98.91%Forma y color:SoildPeso molecular:430.533-(7,7-dimethyl-5-oxo-6,7-dihydro-5H-pyrrolo[3,4-b]pyridin-2-yl)-1H-indole-7-carbonitrile
CAS:3-[7 ,7- dimethyl-5-oxo -6H-pyrrolo[3,4-b]pyridin-2-yI]-1H-indole-7 -carbonitrile is an androgen receptor modulator.Fórmula:C18H14N4OPureza:98.41%Forma y color:SolidPeso molecular:302.332-hydroxy Flutamide
CAS:2-hydroxy Flutamide is competitive inhibition of androgen receptor (AR) for the treatment of prostate cancerFórmula:C11H11F3N2O4Pureza:99.45% - 99.82%Forma y color:SolidPeso molecular:292.21Testosterone undecanoate
CAS:Testosterone undecanoate is a metabolite of Testosterone, which is a promising androgen for male hormonal contraception.Fórmula:C30H48O3Pureza:99.45% - 99.788%Forma y color:White Crystalline PowderPeso molecular:456.7Apalutamide
CAS:<p>Apalutamide (ARN-509) is a small molecule and androgen receptor (AR) antagonist with potential antineoplastic activity.</p>Fórmula:C21H15F4N5O2SPureza:99.03% - 99.91%Forma y color:SolidPeso molecular:477.43AH-3960
CAS:AH-3960 是一种甲状腺激素受体 1 (PTHR1) 激动剂。Fórmula:C13H22N4O3Pureza:98.44%Forma y color:SolidPeso molecular:282.34VPC-13163
CAS:VPC-13566 inhibits growth in LNCaP, Enzalutamide-resistant MR49F, lowers AR gene, PSA, TMPRSS2 expression, but not in AR-independent PC3 cells.Fórmula:C16H14N2Pureza:98.02%Forma y color:SolidPeso molecular:234.3Ref: TM-T29110
1mg89,00€2mg117,00€5mg187,00€10mg284,00€25mg452,00€50mg645,00€100mg867,00€200mg1.130,00€1mL*10mM (DMSO)168,00€S-23
CAS:S-23 ((S)-3-(4-chloro-3-fluorophenoxy)-N-(4-cyano-3-(trifluoromethyl)phenyl)-2-hydroxy-2-methylpropanamide) is an oral selective androgen receptor modulator (Fórmula:C18H13ClF4N2O3Pureza:99.55%Forma y color:SolidPeso molecular:416.75Iprodione
CAS:Iprodione is a fungicide. Iprodione is also used in cannabis testing kits as a component of pesticide mixes.Fórmula:C13H13Cl2N3O3Pureza:98.82%Forma y color:Colorless Crystals Cream To Colorless Odorless PowderPeso molecular:330.17Bavdegalutamide
CAS:Bavdegalutamide (ARV-110) is a PROTAC degrader of androgen receptor (AR).Fórmula:C41H43ClFN9O6Pureza:97.17% - 99.04%Forma y color:SolidPeso molecular:812.29N-desmethyl Enzalutamide
CAS:N-desmethyl Enzalutamide (N-desmethyl MDV 3100) is the active Enzalutamide metabolite.It is the active metabolite of Enzalutamide.Fórmula:C20H14F4N4O2SPureza:99.74%Forma y color:SolidPeso molecular:450.41Ref: TM-T19450
2mg34,00€5mg52,00€10mg74,00€25mg138,00€50mg255,00€100mg375,00€200mg532,00€1mL*10mM (DMSO)58,00€Enzalutamide carboxylic acid
CAS:<p>Enzalutamide carboxylic acid is an antagonist of androgen receptor (AR) .</p>Fórmula:C20H13F4N3O3SPureza:97.88%Forma y color:SolidPeso molecular:451.39Lupeol
CAS:Lupeol (Monogynol B) is a novel androgen receptor inhibitor with anti-inflammatory and antioxidant activity.Fórmula:C30H50OPureza:98% - 99.96%Forma y color:Needles From Alcohol Acetone White PowderPeso molecular:426.72VPC-13566
CAS:<p>VPC-13566 is a BF3-specific small molecule, which effectively inhibited the androgen receptor transcriptional activity and displaced the BAG1L peptide from the</p>Fórmula:C18H14N2Pureza:99.55%Forma y color:SolidPeso molecular:258.32
