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Canal de potasio

Canal de potasio

Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.

Se han encontrado 276 productos de "Canal de potasio"

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  • NS1643

    CAS:
    <p>NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator with EC50 of 10.5 μM.</p>
    Fórmula:C15H10F6N2O3
    Pureza:98.37% - 99.31%
    Forma y color:Solid
    Peso molecular:380.24
  • GAL-021

    CAS:
    <p>GAL-021 an intravenous BKCa-channel blocker.</p>
    Fórmula:C11H22N6O
    Pureza:97.71% - 99.66%
    Forma y color:Solid
    Peso molecular:254.33
  • Daurisoline

    CAS:
    <p>Daurisoline ((R,R)-Daurisoline) is a hERG inhibitor. Daurisoline is also an autophagy blocker.</p>
    Fórmula:C37H42N2O6
    Pureza:98% - 99.96%
    Forma y color:Light Yellow Powder
    Peso molecular:610.74
  • NS-1619

    CAS:
    NS1619 have cardio-protective effects after ischemia-reperfusion injury.
    Fórmula:C15H8F6N2O2
    Pureza:97.66% - 98%
    Forma y color:Solid
    Peso molecular:362.23
  • GW9508

    CAS:
    <p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>
    Fórmula:C22H21NO3
    Pureza:97.89% - 99.19%
    Forma y color:Solid
    Peso molecular:347.41
  • JNJ 303

    CAS:
    <p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>
    Fórmula:C21H29ClN2O4S
    Pureza:99.28%
    Forma y color:Solid
    Peso molecular:440.98
  • TRAM-34

    CAS:
    <p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>
    Fórmula:C22H17ClN2
    Pureza:99.01% - 99.91%
    Forma y color:Solid
    Peso molecular:344.84
  • ML335

    CAS:
    <p>ML335 is a selective activator of TREK-1 and TREK-2.</p>
    Fórmula:C15H14Cl2N2O3S
    Pureza:99.73% - 99.79%
    Forma y color:Solid
    Peso molecular:373.25
  • ICA 110381

    CAS:
    <p>ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsy</p>
    Fórmula:C12H8Cl2N2O
    Pureza:97.72%
    Forma y color:Solid
    Peso molecular:267.11
  • Flecainide hydrochloride

    CAS:
    <p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>
    Fórmula:C17H21ClF6N2O3
    Pureza:97.79%
    Forma y color:Solid
    Peso molecular:450.81
  • Minoxidil sulfate

    CAS:
    <p>Minoxidil sulfate (U-58838) is the active metabolite required to exert the vasodilatory and hair growing effects of minoxidil.</p>
    Fórmula:C9H15N5O4S
    Pureza:99.01% - 99.72%
    Forma y color:White Crystalline Solid
    Peso molecular:289.31
  • ASP2905

    CAS:
    <p>ASP-2905 is a potent and selective inhibitor of potassium channel Kv12.2 encoded by the Kcnh3/BEC1 gene.</p>
    Fórmula:C20H17FN8
    Pureza:97.29%
    Forma y color:Solid
    Peso molecular:388.4
  • AM-92016 hydrochloride

    CAS:
    AM-92016 is a specific blocker of rectifier potassium current.
    Fórmula:C19H24Cl2N2O4S·HCl
    Pureza:98.68%
    Forma y color:Solid
    Peso molecular:483.84
  • NS6180

    CAS:
    <p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>
    Fórmula:C16H12F3NOS
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:323.33
  • Tetraethylammonium chloride

    CAS:
    <p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>
    Fórmula:C8H20ClN
    Pureza:≥95%
    Forma y color:White Solid Solid Particulate/Powder
    Peso molecular:165.7
  • RY785

    CAS:
    <p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>
    Fórmula:C21H20N4O2S
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:392.47
  • Enflurane

    CAS:
    <p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>
    Fórmula:C3H2ClF5O
    Pureza:99.64%
    Forma y color:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As An
    Peso molecular:184.49
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Forma y color:Solid
    Peso molecular:324.24
  • ICA-105574

    CAS:
    <p>ICA-105574 activates hERG, enhancing peak current and shortening action potential, while modulating activation kinetics.</p>
    Fórmula:C19H14N2O4
    Pureza:98.89%
    Forma y color:Solid
    Peso molecular:334.33
  • Branaplam

    CAS:
    <p>Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.</p>
    Fórmula:C22H27N5O2
    Pureza:98.28% - 99.72%
    Forma y color:Solid
    Peso molecular:393.48