
Canal de potasio
Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.
Se han encontrado 276 productos de "Canal de potasio"
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NS1643
CAS:<p>NS1643 is a potent human ether-a-go-go related gene (hERG) KV11.1 channel activator with EC50 of 10.5 μM.</p>Fórmula:C15H10F6N2O3Pureza:98.37% - 99.31%Forma y color:SolidPeso molecular:380.24GAL-021
CAS:<p>GAL-021 an intravenous BKCa-channel blocker.</p>Fórmula:C11H22N6OPureza:97.71% - 99.66%Forma y color:SolidPeso molecular:254.33Daurisoline
CAS:<p>Daurisoline ((R,R)-Daurisoline) is a hERG inhibitor. Daurisoline is also an autophagy blocker.</p>Fórmula:C37H42N2O6Pureza:98% - 99.96%Forma y color:Light Yellow PowderPeso molecular:610.74NS-1619
CAS:NS1619 have cardio-protective effects after ischemia-reperfusion injury.Fórmula:C15H8F6N2O2Pureza:97.66% - 98%Forma y color:SolidPeso molecular:362.23GW9508
CAS:<p>GW9508(GW 9508) is a potent and selective agonist for FFA1 (GPR40), stimulates insulin secretion in a glucose-sensitive manner.</p>Fórmula:C22H21NO3Pureza:97.89% - 99.19%Forma y color:SolidPeso molecular:347.41JNJ 303
CAS:<p>JNJ 303 is a potent blocker of IKs (IC50 : 64 nM).</p>Fórmula:C21H29ClN2O4SPureza:99.28%Forma y color:SolidPeso molecular:440.98TRAM-34
CAS:<p>TRAM-34 (Triarylmethane-34), an effective and specific inhibitor of the intermediate-conductance Ca2+-activated K+ channel, does not block cytochrome P450.</p>Fórmula:C22H17ClN2Pureza:99.01% - 99.91%Forma y color:SolidPeso molecular:344.84ML335
CAS:<p>ML335 is a selective activator of TREK-1 and TREK-2.</p>Fórmula:C15H14Cl2N2O3SPureza:99.73% - 99.79%Forma y color:SolidPeso molecular:373.25ICA 110381
CAS:<p>ICA 110381 is a KCNQ2/Q3 potassium channel opener for the treatment of epilepsy</p>Fórmula:C12H8Cl2N2OPureza:97.72%Forma y color:SolidPeso molecular:267.11Flecainide hydrochloride
CAS:<p>Flecainide is a medication used to prevent and treat abnormally fast heart rates. This includes ventricular and supraventricular tachycardias.</p>Fórmula:C17H21ClF6N2O3Pureza:97.79%Forma y color:SolidPeso molecular:450.81Minoxidil sulfate
CAS:<p>Minoxidil sulfate (U-58838) is the active metabolite required to exert the vasodilatory and hair growing effects of minoxidil.</p>Fórmula:C9H15N5O4SPureza:99.01% - 99.72%Forma y color:White Crystalline SolidPeso molecular:289.31ASP2905
CAS:<p>ASP-2905 is a potent and selective inhibitor of potassium channel Kv12.2 encoded by the Kcnh3/BEC1 gene.</p>Fórmula:C20H17FN8Pureza:97.29%Forma y color:SolidPeso molecular:388.4AM-92016 hydrochloride
CAS:AM-92016 is a specific blocker of rectifier potassium current.Fórmula:C19H24Cl2N2O4S·HClPureza:98.68%Forma y color:SolidPeso molecular:483.84NS6180
CAS:<p>NS6180 is a potent and selective KCa3.1 channel inhibitor(IC50= 9 nM). It prevents T-cell activation and inflammation.</p>Fórmula:C16H12F3NOSPureza:99.83% - ≥95%Forma y color:SolidPeso molecular:323.33Tetraethylammonium chloride
CAS:<p>Tetraethylammonium chloride is a quaternary ammonium compound.</p>Fórmula:C8H20ClNPureza:≥95%Forma y color:White Solid Solid Particulate/PowderPeso molecular:165.7RY785
CAS:<p>RY785 is a potent and selective inhibitor of voltage-gated potassium channel such as KV2.2 (IC50 = 50 nM). RY785 may be used in pain relief studies.</p>Fórmula:C21H20N4O2SPureza:99.78%Forma y color:SolidPeso molecular:392.47Enflurane
CAS:<p>Enflurane (Efrane), a volatile anaesthetic, inhibits Ca2+-activated K+ channels and is used to gauge anesthesia levels in gas chromatography.</p>Fórmula:C3H2ClF5OPureza:99.64%Forma y color:Clear Colorless Liquid Ordinary Temperature And Pressure Bp 56 8°C Density 1 50 G Cm-3 At Room Temperature Used As AnPeso molecular:184.49SCH-23390 hydrochloride
CAS:<p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>Fórmula:C17H19Cl2NOPureza:98% - 99.83%Forma y color:SolidPeso molecular:324.24ICA-105574
CAS:<p>ICA-105574 activates hERG, enhancing peak current and shortening action potential, while modulating activation kinetics.</p>Fórmula:C19H14N2O4Pureza:98.89%Forma y color:SolidPeso molecular:334.33Branaplam
CAS:<p>Branaplam (LMI 070) is a highly potent, selective and orally active small molecule SMN2 splicing modulator.</p>Fórmula:C22H27N5O2Pureza:98.28% - 99.72%Forma y color:SolidPeso molecular:393.48
