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Canal de potasio

Canal de potasio

Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.

Se han encontrado 276 productos de "Canal de potasio"

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  • Kv2-IN-A1

    CAS:
    <p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>
    Fórmula:C20H17ClN4OS
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:396.89
  • Almitrine mesylate

    CAS:
    <p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>
    Fórmula:C28H37F2N7O6S2
    Pureza:99.96%
    Forma y color:Coa
    Peso molecular:669.76
  • Azimilide Dihydrochloride

    CAS:
    <p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>
    Fórmula:C23H30Cl3N5O3
    Pureza:97.59% - ≥95%
    Forma y color:Solid
    Peso molecular:530.88
  • ML365

    CAS:
    <p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>
    Fórmula:C22H20N2O3
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:360.41
  • VU0071063

    CAS:
    <p>VU0071063 is a Kir6.2/SUR1 activator.</p>
    Fórmula:C18H22N4O2
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:326.39
  • Quinine dihydrochloride

    CAS:
    <p>Quinine dihydrochloride (Quinine bimuriate) is a primary alkaloid of various species of Cinchona (Rubiaceae).</p>
    Fórmula:C20H26Cl2N2O2
    Pureza:99.79% - 99.97%
    Forma y color:White Solid
    Peso molecular:397.34
  • Sematilide hydrochloride

    CAS:
    <p>Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker.</p>
    Fórmula:C14H24ClN3O3S
    Pureza:99.14%
    Forma y color:Solid
    Peso molecular:349.87
  • Dofetilide

    CAS:
    <p>Dofetilide (UK 68789), a class III antiarrhythmic sulfonamide, blocks Ikr cardiac channels, prolongs action potential, and treats atrial fibrillation/flutter.</p>
    Fórmula:C19H27N3O5S2
    Pureza:97.85% - 99.06%
    Forma y color:Off-White Or Yellowish Crystalline Powder
    Peso molecular:441.56
  • AUT1

    CAS:
    <p>AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).</p>
    Fórmula:C18H19N3O4
    Pureza:99.8% - 99.95%
    Forma y color:Solid
    Peso molecular:341.36
  • Iptakalim Hydrochloride

    CAS:
    <p>Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine</p>
    Fórmula:C9H22ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:179.731
  • GSK369796 Dihydrochloride

    CAS:
    <p>GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.</p>
    Fórmula:C20H24Cl3N3O
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:428.78
  • PAP-1

    CAS:
    <p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>
    Fórmula:C21H18O5
    Pureza:99.35% - 99.75%
    Forma y color:White Solid
    Peso molecular:350.36
  • Nigericin sodium salt

    CAS:
    <p>Nigericin sodium salt, an antibiotic and NLRP3 activator from S. hygroscopicus, inhibits Golgi and gram-positive bacteria, blocking viral activation.</p>
    Fórmula:C40H67NaO11
    Pureza:98.2% - 99.52%
    Forma y color:Solid
    Peso molecular:746.94
  • Atpenin A5

    CAS:
    <p>Atpenin A5 is a potent and highly specific complex II inhibitor (IC50 ~10 nM).</p>
    Fórmula:C15H21Cl2NO5
    Pureza:97.33% - 99.91%
    Forma y color:Solid
    Peso molecular:366.24
  • LY 303511 hydrochloride

    CAS:
    <p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>
    Fórmula:C19H19ClN2O2
    Pureza:98.47%
    Forma y color:Solid
    Peso molecular:342.82
  • Mitiglinide Calcium

    CAS:
    <p>Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-</p>
    Fórmula:(C19H24NO3)2·Ca
    Pureza:99.83%
    Forma y color:White Crystal Posder
    Peso molecular:668.88
  • Flupirtine maleate

    CAS:
    <p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>
    Fórmula:C15H17FN4O2·C4H4O4
    Pureza:99.5% - 99.9%
    Forma y color:Off-White Crystalline Powder
    Peso molecular:420.39
  • Senicapoc

    CAS:
    <p>Senicapoc (ICA-17043) blocks Gardos channel, reduces RBC dehydration, IC50: 11 nM for rubidium flux, 30 nM for dehydration. Used in Sickle Cell therapy.</p>
    Fórmula:C20H15F2NO
    Pureza:95.7% - 99.47%
    Forma y color:Solid
    Peso molecular:323.34
  • E-4031 dihydrochloride

    CAS:
    <p>E-4031 is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by blocking ERG K+ channels (IC50 = 29 nM)</p>
    Fórmula:C21H29Cl2N3O3S
    Pureza:99.31% - 99.87%
    Forma y color:Solid
    Peso molecular:474.44
  • Allocryptopine

    CAS:
    <p>Allocryptopine (Thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively.</p>
    Fórmula:C21H23NO5
    Pureza:99.41% - ≥95%
    Forma y color:Solid
    Peso molecular:369.41