
Canal de potasio
Los canales de potasio son un grupo diverso de proteínas de membrana que facilitan el flujo de iones de potasio (K+) a través de la membrana celular. Estos canales desempeñan un papel crucial en el mantenimiento del potencial de membrana en reposo, la regulación del volumen celular y el control de la excitabilidad de las neuronas y las células musculares. Los canales de potasio están involucrados en varios procesos fisiológicos, incluyendo la regulación del ritmo cardíaco, la secreción de insulina y la liberación de neurotransmisores. La disfunción de los canales de potasio está relacionada con condiciones como arritmias, epilepsia e hipertensión. En CymitQuimica, ofrecemos una amplia gama de moduladores de canales de potasio para apoyar su investigación en electrofisiología, salud cardiovascular y neurobiología.
Se han encontrado 276 productos de "Canal de potasio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Kv2-IN-A1
CAS:<p>Kv2-IN-A1 is an inhibitor of Kv2.1 and Kv2.2.</p>Fórmula:C20H17ClN4OSPureza:98.83%Forma y color:SolidPeso molecular:396.89Almitrine mesylate
CAS:<p>Almitrine mesylate targets Ca2+-dependent K+ channels in rat cells, used for chronic lung hypoxemia.</p>Fórmula:C28H37F2N7O6S2Pureza:99.96%Forma y color:CoaPeso molecular:669.76Azimilide Dihydrochloride
CAS:<p>Azimilide Dihydrochloride (NE-10064 Dihydrochloride), a novel class III antiarrhythmic agent, blocks both the IKs and IKr with antiarrhythmic activity.</p>Fórmula:C23H30Cl3N5O3Pureza:97.59% - ≥95%Forma y color:SolidPeso molecular:530.88ML365
CAS:<p>ML365 is a novel selective small molecule inhibitor of TASK1(KCNK3).</p>Fórmula:C22H20N2O3Pureza:98.78%Forma y color:SolidPeso molecular:360.41VU0071063
CAS:<p>VU0071063 is a Kir6.2/SUR1 activator.</p>Fórmula:C18H22N4O2Pureza:99.33%Forma y color:SolidPeso molecular:326.39Quinine dihydrochloride
CAS:<p>Quinine dihydrochloride (Quinine bimuriate) is a primary alkaloid of various species of Cinchona (Rubiaceae).</p>Fórmula:C20H26Cl2N2O2Pureza:99.79% - 99.97%Forma y color:White SolidPeso molecular:397.34Sematilide hydrochloride
CAS:<p>Sematilide hydrochloride (CK-1752) is a class III antiarrhythmic. It is a selectively delayed rectifier K+ current (IKr) channel blocker.</p>Fórmula:C14H24ClN3O3SPureza:99.14%Forma y color:SolidPeso molecular:349.87Dofetilide
CAS:<p>Dofetilide (UK 68789), a class III antiarrhythmic sulfonamide, blocks Ikr cardiac channels, prolongs action potential, and treats atrial fibrillation/flutter.</p>Fórmula:C19H27N3O5S2Pureza:97.85% - 99.06%Forma y color:Off-White Or Yellowish Crystalline PowderPeso molecular:441.56AUT1
CAS:<p>AUT1 (AUT-1) is a novel specific modulator of Kv3 channels (EC50: 4.7 and 4.9 uM for Kv3.1b and Kv3.2a).</p>Fórmula:C18H19N3O4Pureza:99.8% - 99.95%Forma y color:SolidPeso molecular:341.36Iptakalim Hydrochloride
CAS:<p>Iptakalim, a lipophilic para-amino compound, is a novel ATP-sensitive potassium channel (KATP) opener, as well as an α4β2-containing nicotinic acetylcholine</p>Fórmula:C9H22ClNPureza:98%Forma y color:SolidPeso molecular:179.731GSK369796 Dihydrochloride
CAS:<p>GSK369796 Dihydrochloride (N-tert-butylisoquine),is an anti-malaria drug candidate.</p>Fórmula:C20H24Cl3N3OPureza:>99.99%Forma y color:SolidPeso molecular:428.78PAP-1
CAS:<p>PAP-1 (5-(4-Phenoxybutoxy)psoralen) is a selective, and orally active Kv1.3 blocker (EC50: 2 nM).</p>Fórmula:C21H18O5Pureza:99.35% - 99.75%Forma y color:White SolidPeso molecular:350.36Nigericin sodium salt
CAS:<p>Nigericin sodium salt, an antibiotic and NLRP3 activator from S. hygroscopicus, inhibits Golgi and gram-positive bacteria, blocking viral activation.</p>Fórmula:C40H67NaO11Pureza:98.2% - 99.52%Forma y color:SolidPeso molecular:746.94Atpenin A5
CAS:<p>Atpenin A5 is a potent and highly specific complex II inhibitor (IC50 ~10 nM).</p>Fórmula:C15H21Cl2NO5Pureza:97.33% - 99.91%Forma y color:SolidPeso molecular:366.24LY 303511 hydrochloride
CAS:<p>LY 303511 hydrochloride is a potent mTOR inhibitor</p>Fórmula:C19H19ClN2O2Pureza:98.47%Forma y color:SolidPeso molecular:342.82Mitiglinide Calcium
CAS:<p>Mitiglinide Calcium (KAD-1229) is a blood glucose-lowering drugs, stimulating insulin secretion by closing the ATP-sensitive K+ channels in pancreatic beta-</p>Fórmula:(C19H24NO3)2·CaPureza:99.83%Forma y color:White Crystal PosderPeso molecular:668.88Flupirtine maleate
CAS:<p>Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. Flupirtine is an NMDA receptor antagonist.</p>Fórmula:C15H17FN4O2·C4H4O4Pureza:99.5% - 99.9%Forma y color:Off-White Crystalline PowderPeso molecular:420.39Senicapoc
CAS:<p>Senicapoc (ICA-17043) blocks Gardos channel, reduces RBC dehydration, IC50: 11 nM for rubidium flux, 30 nM for dehydration. Used in Sickle Cell therapy.</p>Fórmula:C20H15F2NOPureza:95.7% - 99.47%Forma y color:SolidPeso molecular:323.34E-4031 dihydrochloride
CAS:<p>E-4031 is a methanesulfonanilide class III antiarrhythmic agent that prolongs cardiac action potential duration by blocking ERG K+ channels (IC50 = 29 nM)</p>Fórmula:C21H29Cl2N3O3SPureza:99.31% - 99.87%Forma y color:SolidPeso molecular:474.44Allocryptopine
CAS:<p>Allocryptopine (Thalictrimine) induces muscle contraction and relaxation in urinary bladder and ileum, respectively.</p>Fórmula:C21H23NO5Pureza:99.41% - ≥95%Forma y color:SolidPeso molecular:369.41
