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Canal de cloruro

Canal de cloruro

Los canales de cloruro son proteínas de membrana que controlan el movimiento de los iones de cloruro a través de las membranas celulares, desempeñando un papel vital en el mantenimiento del volumen celular, la excitabilidad eléctrica y el equilibrio ácido-base. La desregulación de los canales de cloruro está relacionada con enfermedades como la fibrosis quística, la epilepsia y los trastornos renales. En CymitQuimica, ofrecemos una variedad de moduladores de canales de cloruro para apoyar su investigación en el transporte de iones, la homeostasis celular y los mecanismos de enfermedades.

Se han encontrado 49 productos de "Canal de cloruro"

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  • Stepronin

    CAS:
    <p>Stepronin (TTPG) shows expectorant activities and inhibits airway secretion.</p>
    Fórmula:C10H11NO4S2
    Pureza:99.59%
    Forma y color:White Or Off White Crystalline
    Peso molecular:273.33
  • ANO1-IN-1

    CAS:
    <p>ANO1-IN-1 blocks ANO1/2 channels (IC50: 2.56/15.43 μM) and hinders glioma cell growth.</p>
    Fórmula:C18H28N2O2S
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:336.49
  • Ani9

    CAS:
    <p>Ani9 selectively blocks ANO1/TMEM16A with a 77 nM IC50, useful for ANO1 research and treating cancer, hypertension, pain, diarrhea, asthma.</p>
    Fórmula:C17H17ClN2O3
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:332.78
  • ARN 11391

    CAS:
    <p>ARN 11391 enhances the function of the IP3-gated calcium channel ITPR1 (Inositol 1,4,5-trisphosphate (IP3) receptor type 1), boosting intracellular calcium ion</p>
    Fórmula:C22H29N3O3
    Forma y color:Solid
    Peso molecular:383.49
  • OADS

    CAS:
    <p>OADS is an inhibitor of ClC-ec1 with low micromolar affinity. OADS has no specific effect on a CLC channel (ClC-1).</p>
    Fórmula:C30H42N2O8S2
    Forma y color:Solid
    Peso molecular:622.79
  • S9-A13

    CAS:
    <p>S9-A13 is a potent and selective inhibitor of SLC26A9, exhibiting an IC50 of 90.9 nM without inhibiting other members of the SLC26 family, such as SLC26A3, SLC26A4, and SLC26A6. It also inhibits the SLC26A9 Cl- current in cells lacking CFTR expression.</p>
    Fórmula:C20H18ClN3O2S
    Forma y color:Solid
    Peso molecular:399.89
  • NMD670

    CAS:
    <p>NMD670 is an orally active, partial inhibitor of the skeletal muscle-specific chloride channel ClC-1. It enhances muscle excitability and neuromuscular transmission, restoring muscle function and mobility. NMD670 has a favorable safety profile and improves muscle function in rats, particularly in an MG rat model [1].</p>
    Fórmula:C12H10BrNO4
    Forma y color:Solid
    Peso molecular:312.12
  • DFBTA


    <p>DFBTA inhibits ANO1 with IC50 of 24 nM, effectively treating inflammatory pain orally.</p>
    Fórmula:C18H10ClF2NO3S
    Forma y color:Solid
    Peso molecular:393.79
  • T16A(inh)-C01

    CAS:
    <p>T16A(inh)-C01 is the Ca(2+)-activated Cl(-) Channel, Ano1 class C inhibitor.</p>
    Fórmula:C18H16O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:312.32

    Ref: TM-T24846

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