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Receptor CGRP

Receptor CGRP

Los receptores de CGRP están involucrados en la transmisión del dolor y la regulación del flujo sanguíneo. El CGRP es un neuropéptido que desempeña un papel crucial en la fisiopatología de la migraña al dilatar los vasos sanguíneos y modular las vías de señalización del dolor. Dirigirse a los receptores de CGRP se ha convertido en un enfoque prometedor en el desarrollo de terapias para la migraña. En CymitQuimica, ofrecemos una gama de moduladores de receptores de CGRP para apoyar su investigación en el manejo del dolor, neurobiología y salud vascular.

Se han encontrado 51 productos de "Receptor CGRP"

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  • β-CGRP, human acetate


    <p>β-CGRP, human acetate is one of calcitonin peptides and acts via the complex of receptor-activity-modifying protein (RAMP) and calcitonin-receptor-like receptor</p>
    Fórmula:C164H271N51O50S3
    Pureza:99.35%
    Forma y color:Solid
    Peso molecular:3853.46
  • Atogepant

    CAS:
    <p>Atogepant (MK-8031) is an orally available, selective and potent calcitonin gene-related peptide receptor (CGRP) antagonist for the study of migraine.</p>
    Fórmula:C29H23F6N5O3
    Pureza:99.66%
    Forma y color:Solid
    Peso molecular:603.52
  • Fremanezumab

    CAS:
    <p>Fremanezumab (TEV-48125) is a humanised monoclonal antibody targeting CGRP, capable of neutralising human, mouse and rat CGRP, migraine.</p>
    Pureza:95% - 95%
    Forma y color:Liquid
  • Eptinezumab

    CAS:
    <p>Eptinezumab is a humanised monoclonal antibody targeting CGRP (calcitonin gene-related peptide), which prevents CGRP binding to its receptor, migraine.</p>
    Pureza:95% - 95%
    Forma y color:Liquid
  • SB 268262

    CAS:
    <p>CGRP1 antagonist</p>
    Fórmula:C18H15N3O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:401.46
  • CGRP antagonist 1

    CAS:
    <p>CGRP antagonist 1 is a potent CGRP receptor antagonist with Ki values of 35 nM and IC50 values of 57 nM, respectively.CGRP antagonist 1 can be used for the</p>
    Fórmula:C29H26N4O4
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:494.54
  • Ubrogepant

    CAS:
    <p>Ubrogepant (MK-1602) is an antagonist of calcitonin gene-related peptide receptor that can be used in the acute treatment of migraine studies.</p>
    Fórmula:C29H26F3N5O3
    Pureza:99.452% - 99.78%
    Forma y color:Solid
    Peso molecular:549.54
  • MK-3207

    CAS:
    <p>MK-3207 is a potent, oral CGRP receptor antagonist with high selectivity for human and monkey receptors, inhibiting blood flow in vivo.</p>
    Fórmula:C31H29F2N5O3
    Forma y color:Solid
    Peso molecular:557.59
  • MK-3207 Hydrochloride

    CAS:
    <p>MK-3207 Hydrochloride (MK-3207 HCl) is a potent CGRP receptor antagonist with IC50 and Kiof 0.12 nM and 0.022 nM, highly selective versus human AM1, AM2, CTR, and AMY3. Phase 2.</p>
    Fórmula:C31H30ClF2N5O3
    Pureza:98.19%
    Forma y color:Solid
    Peso molecular:594.05
  • BI-44370

    CAS:
    <p>BI-44370, a CGRP (calcitonin gene-related peptide) receptor antagonist, can be used to treat migraines and other chronic pain.</p>
    Fórmula:C35H47N5O6
    Forma y color:Solid
    Peso molecular:633.78
  • MK-8825

    CAS:
    <p>MK-8825 is a CGRP receptor antagonist.</p>
    Fórmula:C31H30F2N6O3
    Forma y color:Solid
    Peso molecular:572.61