
Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 549 productos de "Canal de calcio"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Mci 176
CAS:Mci 176 is a quinazolinone calcium antagonist.Fórmula:C24H32ClN3O4Forma y color:SolidPeso molecular:461.98Lemildipine
CAS:Lemildipine is a new blocker of dihydropyridine calcium entry.Fórmula:C20H22Cl2N2O6Forma y color:SolidPeso molecular:457.3BA 41899
CAS:BA 41899 is a positive inotropic Ca(2+)-sensitizing agent.Fórmula:C18H16N2O2Forma y color:SolidPeso molecular:292.33GSK-5503A
CAS:GSK-5503A is a novel channel blocker of CRAC.Fórmula:C23H17F2N3O2Pureza:98%Forma y color:SolidPeso molecular:405.4MRS2690
CAS:MRS2690 is a potent P2Y14 receptor agonist (EC50 = 49 nM) that displays 7-fold higher potency than UDP-glucose.Fórmula:C15H24N2O16P2SForma y color:SolidPeso molecular:582.37SIM-6080
CAS:SIM-6080 is a calcium channel antagonist. SIM-6080 inhibits the proliferation of rat aortic myocytes.Fórmula:C29H36F2N2O3Forma y color:SolidPeso molecular:498.6RS-93522
CAS:RS-93522: Calcium channel antagonist, inhibits phosphodiesterase (IC50=1.6x10^-5M), like milrinone, and has a negative inotropic effect.Fórmula:C27H30N2O9Pureza:98%Forma y color:SolidPeso molecular:526.54Diproteverine
CAS:Diproteverine is a calcium antagonist, it has antianginal property.Fórmula:C26H35NO4Pureza:98%Forma y color:SolidPeso molecular:425.56BMS-192364
CAS:BMS-192364 is a bio-active chemical.Fórmula:C15H9ClF3N3O2Forma y color:SolidPeso molecular:355.70AJG-049 free base
CAS:AJG-049 free base is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Fórmula:C27H30N2O2Forma y color:SolidPeso molecular:414.54Azelnidipine, (S)-
CAS:Azelnidipine, a selective L-type CCB, improves HF severity and cardiac function in HT and HFpEF compared to N-type CCB cilnidipine.Fórmula:C33H34N4O6Forma y color:SolidPeso molecular:582.65ORM-10962
CAS:ORM-10962 is a potent, highly selective inhibitor of sodium-calcium exchanger (NCX) (for the reverse and forward mode inhibition with IC50 values of 67 and 55Fórmula:C27H29N3O4Pureza:98%Forma y color:SolidPeso molecular:459.54PPZ2
CAS:PPZ2 is a novel DAG-activated TRPC3/TRPC6/TRPC7 channels activator.Fórmula:C22H29N3O2Forma y color:SolidPeso molecular:367.48Aladorian sodium
CAS:Aladorian sodium is used for Treatment of Cardiovascular Diseases.Fórmula:C12H13NNaO4SForma y color:SolidPeso molecular:290.29Hyperforin dicyclohexylammonium salt
CAS:Hyperforin dicyclohexylammonium is a TRPC6 activator and antidepressant that modulates Ca2+ levels.Fórmula:C47H75NO4Pureza:98%Forma y color:SolidPeso molecular:718.10PAQ
CAS:PAQ protects neurons in Parkinson's models at 10 μM; prevents neuron loss in mice substantia nigra with 25-50 mg/kg doses.Fórmula:C14H11N3Forma y color:SolidPeso molecular:221.26Ro 18-3981
CAS:Ro 18-3981 inhibits myocardial Ca2+ channels; KD is 1.0 nM, close to IC50 for ICa block (2.3 nM).Fórmula:C24H33N3O8SForma y color:SolidPeso molecular:523.6Azelnidipine, (R)-
CAS:Azelnidipine is an L-type CCB that improves HF severity and cardiac nerve activity in HT and HFpEF compared to cilnidipine.Fórmula:C33H34N4O6Forma y color:SolidPeso molecular:582.65SR-33805
CAS:SR-33805: calcium channel blocker for atherosclerosis/heart failure, enhances myocyte function, modulates myofilament phosphorylation.Fórmula:C32H40N2O5SForma y color:SolidPeso molecular:564.74TTA-Q6(isomer)
CAS:TTA-Q6(isomer) is an isomer of TTA-Q6. TTA-Q6 is a selective antagonist of the T-type Ca2+ channel.Fórmula:C20H15ClF3N3OPureza:98%Forma y color:SolidPeso molecular:405.8
