
Canal de calcio
Los canales de calcio son proteínas de membrana que regulan el flujo de iones de calcio hacia dentro y fuera de las células, lo cual es esencial para diversas funciones celulares, como la contracción muscular, la liberación de neurotransmisores y la expresión génica. La desregulación de la actividad de los canales de calcio está asociada con condiciones como la hipertensión, las arritmias cardíacas y los trastornos neurológicos. En CymitQuimica, ofrecemos una amplia selección de moduladores de canales de calcio para apoyar su investigación en salud cardiovascular, neurobiología y transducción de señales.
Se han encontrado 562 productos de "Canal de calcio"
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AJG-049 HCl
CAS:AJG-049 HCl is a calcium channel antagonist that inhibits L-type Ca2+ channels via diltiazem-binding site(s).Fórmula:C27H31ClN2O2Forma y color:SolidPeso molecular:451.01PD-151307
CAS:PD-151307 is used as an N-type calcium channel blocker.Fórmula:C33H47N3O5Pureza:98%Forma y color:SolidPeso molecular:565.74(Rac)-MEM 1003
CAS:MEM-1003, a calcium channel blocker, is used potentially for the treatment of bipolar disorders.Fórmula:C22H25ClN2O5Forma y color:SolidPeso molecular:432.9RyRs activator 3
CAS:RyRs activator 3 (compound A4) serves as an insecticide highly effective against both the diamondback moths, M.Fórmula:C23H19BrCl2N6O3Pureza:98%Forma y color:SolidPeso molecular:578.25AMG-1
CAS:AMG-1 inhibits CRAC channels, blocks effector T cells, not regulatory ones, and reduces EAE progression.Fórmula:C18H9ClF5N3OForma y color:SolidPeso molecular:413.73RQ-00311651
CAS:RQ-00311651 is a novel T-type Ca2+ channel blocker. RQ-00311651 also inhibited high K-induced Ca signaling in those cells.Fórmula:C19H18F3N5O2Forma y color:SolidPeso molecular:405.37β-Amino Acid Imagabalin Hydrochloride
CAS:β-Amino Acid Imagabalin Hydrochloride is the voltage-dependent calcium channel ligand for the α2δ subunit.Fórmula:C9H20ClNO2Pureza:98%Forma y color:SolidPeso molecular:209.71Lidoflazine
CAS:Lidoflazine: antianginal, blocks HERG K+ & Ca channels, risks QT prolongation & arrhythmia.Fórmula:C30H35F2N3OPureza:98%Forma y color:SolidPeso molecular:491.62Semotiadil recemate fumarate
CAS:Semotiadil recemate fumarate is the recemate of Semotiadil fumarate. Semotiadil fumarate is a novel antagonist of vasoselective Ca2+ channel.Fórmula:C33H36N2O10SPureza:98%Forma y color:SolidPeso molecular:652.71Carboxyamidotriazole
CAS:Carboxyamidotriazole is a cytostatic inhibitor of non-voltage-operated calcium channels and calcium channel-mediated signaling pathways.Fórmula:C17H12Cl3N5O2Pureza:98%Forma y color:SolidPeso molecular:424.67Halofuginone hydrobromide
CAS:Halofuginone specifically inhibits collagen type I and MMP-2 gene expression, which may result in the suppression of angiogenesis and tumor cell growth.Fórmula:C16H17BrClN3O3·HBrPureza:97.01% - 99.73%Forma y color:SolidPeso molecular:495.59Ref: TM-T3524
1mg34,00€2mg49,00€5mg74,00€10mg106,00€25mg207,00€50mg310,00€100mg469,00€500mg897,00€1mL*10mM (DMSO)84,00€18:0 LYSO-PE
CAS:18:0 LYSO-PE is a compound that induces an increase in [Ca2+]i and can be used as a phospholipid (PL) standard for lipid analysis by electrospray mass spectrometry (ESI-MS)/MS.Fórmula:C23H48NO7PPureza:98%Forma y color:SolidPeso molecular:481.6DHP-218
CAS:DHP-218, a calcium channel blocker, inhibits rat aorta contractions; pA2: 9.11, IC50: 6.3 nmol/L (high K+) & 66 nmol/L (phenylephrine).Fórmula:C18H21N2O7PPureza:98%Forma y color:SolidPeso molecular:408.34AH-1058 HCl
CAS:AH-1058 HCl is a lipophilic antiarrhythmic calcium channel blocker.Fórmula:C30H29ClN2O3Pureza:98%Forma y color:SolidPeso molecular:501.02A 39355
CAS:A 39355 may specifically overcome multidrug resistance without the serious hypotensive effects associated with calcium antagonists.Fórmula:C28H39Cl2N3OPureza:98%Forma y color:SolidPeso molecular:504.54NP-252
CAS:NP-252 is a calcium channel antagonist potentially for the treatment of angina pectoris and congestive heart failure.Fórmula:C26H35N3O5Pureza:98%Forma y color:SolidPeso molecular:469.57KB-130015
CAS:KB-130015, a activator of hERG1 potassium channels, blocks native and recombinant hERG1 channels at high voltages.Fórmula:C18H14I2O4Pureza:98%Forma y color:SolidPeso molecular:548.11Watanidipine dihydrochloride
CAS:Watanidipine dihydrochloride is a novel dihydropyridine (DHP)-type calcium channel blocker with slow-onset pharmacological actions.Fórmula:C41H44Cl2N4O6Pureza:98%Forma y color:SolidPeso molecular:759.73Gallopamil, (-)-
CAS:Gallopamil, (-)- is an L-type calcium channel blocker. It is used in the treatment of abnormal heart rhythms.Fórmula:C28H40N2O5Pureza:98%Forma y color:SolidPeso molecular:484.63
