Transferasa
Las transferasas son una gran clase de enzimas que catalizan la transferencia de grupos funcionales, como grupos metilo, glicosilo y fosfato, de una molécula a otra. Los inhibidores de transferasas se utilizan para estudiar una amplia gama de procesos biológicos, incluyendo la transducción de señales, el metabolismo y la expresión génica. Estos inhibidores son herramientas esenciales en áreas de investigación como el cáncer, las enfermedades metabólicas y la epigenética, donde está implicada la disfunción de la actividad de las transferasas. En CymitQuimica, ofrecemos una selección integral de inhibidores de transferasas para apoyar su investigación en enzimología, señalización celular y mecanismos de enfermedad.
Se han encontrado 30 productos de "Transferasa"
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Cycloleucine
CAS:<p>Cycloleucine is an antagonist of NMDA receptor associated glycine receptor with a Ki of 600 μM.</p>Fórmula:C6H11NO2Pureza:99.90%Forma y color:SolidPeso molecular:129.16Opicapone
CAS:<p>Opicapone (BIA 9-1067), a potent COMT inhibitor for Parkinson's studies, lowers cell ATP (IC50: 98 μM).</p>Fórmula:C15H10Cl2N4O6Pureza:98.17% - 99.36%Forma y color:SolidPeso molecular:413.17Sinbaglustat
CAS:<p>Sinbaglustat (OGT2378), an oral N-alkyl iminosugar, inhibits GCS/GBA2 and treats lysosomal storage and neurodegenerative disorders.</p>Fórmula:C11H23NO4Pureza:99.93%Forma y color:SolidPeso molecular:233.3Histamine glutarimide
CAS:<p>Histamine glutarimide is a novel QPCT inhibitor that targets inflammatory processes like eosinophil migration, showing anti-asthmatic effects in animal models.</p>Fórmula:C10H13N3O2Pureza:99.79%Forma y color:SolidPeso molecular:207.23FUT8-IN-1
<p>FUT8-IN-1 (Compound 37) is an inhibitor of α-1,6-fucosyltransferase (FUT8), with a dissociation constant (KD) of 49 nM and an IC50 around 50 µM. In the presence of FUT8, FUT8-IN-1 forms a highly active naphthoquinone imine intermediate, thereby inhibiting FUT8's enzymatic activity.</p>Fórmula:C23H25ClN2OForma y color:SolidPeso molecular:380.91β-1,4-GALT1-IN-1
<p>β-1,4-GALT1-IN-1 (Compound 6) is a β-1,4-GALT1 inhibitor with an IC50 value of 6.2 μM. It is applicable in studying various pathological conditions, including cancer, autoimmune diseases, and viral infections.</p>Fórmula:C29H23NO10Forma y color:SolidPeso molecular:545.494ST6 Sialyltransferase 5
<p>ST6Sialyltransferase5 (EC:2.4.3.3, ST6GALNAC5, SIAT7E, ST6 N-acetylgalactosaminide alpha-2,6-sialyltransferase 5) transfers sialic acid to N-acetylgalactosamine (GalNAc) residues. It may serve as a biomarker in cervical screening samples.</p>L-739750 2HCl
<p>L-739750 2HCl is a potent inhibitor of peptidomimetic farnesyltransferase, a novel pseudopeptide mimetic with potential anticancer activity.</p>Fórmula:C23H41Cl2N3O6S2Pureza:98.69% - 99.16%Forma y color:SoildPeso molecular:590.62Tipifarnib
CAS:<p>Tipifarnib (IND 58359), a quinolinone, inhibits farnesyl transferase, blocks Ras activation, arrests cell growth, and curbs angiogenesis.</p>Fórmula:C27H22Cl2N4OPureza:97.1% - 99.22%Forma y color:Off-White To Pale Beige SolidPeso molecular:489.4Ibiglustat
CAS:<p>Ibiglustat (GZ402671) inhibits Glucosylceramide synthase, may treat Fabry disease by preventing GL-3 synthesis.</p>Fórmula:C20H24FN3O2SPureza:97.97% - 98.81%Forma y color:SolidPeso molecular:389.49Entacapone
CAS:<p>Entacapone (OR-611) is a selective and reversible inhibitor of catechol-O-methyltransferase (COMT).</p>Fórmula:C14H15N3O5Pureza:98.80% - >99.99%Forma y color:Yellow Crystalline SolidPeso molecular:305.29Tipifarnib (S enantiomer)
CAS:<p>Tipifarnib S enantiomer ((S)-(-)-R-115777) is the S-enantiomer of Tipifarnib. Tipifarnib is a potent and specific farnesyltransferase inhibitor (IC50: 0.6 nM).</p>Fórmula:C27H22Cl2N4OPureza:99.05%Forma y color:SolidPeso molecular:489.4PD 128042
CAS:<p>PD 128042 (CI 976) is a potent orally active and selective ACAT inhibitor(IC50: 73 nM) and a potent lysophospholipid acyltransferase(LPAT) inhibitor.</p>Fórmula:C23H39NO4Pureza:99.79%Forma y color:SolidPeso molecular:393.56CP-609754
CAS:<p>CP-609754 shows selective inhibition of farnesyltransferase.</p>Fórmula:C29H22ClN3O2Pureza:99.04% - 99.86%Forma y color:SolidPeso molecular:479.96Nitecapone
CAS:<p>Nitecapone is a reversible inhibitor of S-COMT (IC50 values of 300 nM in rat liver)</p>Fórmula:C12H11NO6Pureza:98.39%Forma y color:SolidPeso molecular:265.22Ervogastat
CAS:<p>Ervogastat (PF-06865571) is a potent and well-tolerated diacylglycerol acyltransferase 2 inhibitor.</p>Fórmula:C21H21N5O4Pureza:99.97%Forma y color:SolidPeso molecular:407.423-O-Methyltolcapone
CAS:<p>3-O-Methyltolcapone (Ro 40-7591) is a metabolite of Tolcapone which is a potent COMT inhibitor.</p>Fórmula:C15H13NO5Pureza:98%Forma y color:SolidPeso molecular:287.27AMP-Deoxynojirimycin
CAS:<p>AMP-Deoxynojirimycin (AMP-DNM) is a ceramide glucosyltransferase and GCase 2 inhibitor for the study of Parkinson's and diabetes.</p>Fórmula:C22H39NO5Pureza:>99.99%Forma y color:SolidPeso molecular:397.55Lucerastat
CAS:<p>Lucerastat（NBDGJ） is an orally available inhibitor of GCS for Fabry disease by reducing harmful substrates.. GCS is a key enzyme in sphingolipid synthesiss.</p>Fórmula:C10H21NO4Pureza:98%Forma y color:SolidPeso molecular:219.28P-3FAX-Neu5Ac
CAS:<p>P-3FAX-Neu5Ac is a sialic acid analog and a sialyltransferase inhibitor.</p>Fórmula:C22H30FNO14Pureza:97.08%Forma y color:SolidPeso molecular:551.47
