
Fosfolipasa
Las fosfolipasas son un grupo de enzimas que hidrolizan fosfolípidos en ácidos grasos y otras sustancias lipofílicas, desempeñando un papel crítico en la biología de las membranas y la generación de moléculas de señalización. Los inhibidores de fosfolipasas se utilizan para estudiar su papel en enfermedades inflamatorias, trastornos cardiovasculares y neurodegeneración. Estos inhibidores también son valiosos para explorar las vías de señalización de lípidos y sus implicaciones en los mecanismos de enfermedades. En CymitQuimica, ofrecemos una variedad de inhibidores de fosfolipasas para apoyar su investigación en inflamación, metabolismo de lípidos y señalización celular.
Se han encontrado 86 productos para "Fosfolipasa".
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ST271
CAS:ST271 is an effective protein tyrosine kinase (PTK) inhibitor.Fórmula:C16H20N2O2Pureza:98.49%Forma y color:SolidPeso molecular:272.34Darapladib
CAS:Darapladib (SB-480848) is a lipoprotein-associated phospholipase A2 (Lp-PLA2) inhibitor with an IC50 value of 0.25 nM.Cost-effective and quality-assured.Fórmula:C36H38F4N4O2SPureza:99.82% - >99.99%Forma y color:SolidPeso molecular:666.77Ref: TM-T6109
1mg39,00€2mg50,00€5mg82,00€1mL*10mM (DMSO)110,00€10mg118,00€25mg170,00€50mg294,00€100mg472,00€200mg673,00€RHC 80267
CAS:RHC 80267 (U-57908) is a selective inhibitor of DAGL (IC50 : 4 μM in canine platelets)Fórmula:C20H34N4O4Pureza:99.54%Forma y color:White SolidPeso molecular:394.51GW4869
CAS:GW4869 (GW69A) is a selective and non-competitive inhibitor of neutral sphingomyelinase N-SMase (IC50=1 μM).Fórmula:C30H30Cl2N6O2Pureza:98.12% - 98.47%Forma y color:SolidPeso molecular:577.5Anti-Inflammatory Peptide 1 Acetate
Anti-Inflammatory Peptide 1 Acetate (C45H82N12O14S2) inhibits PLA2 to reduce inflammation and pain.Fórmula:C47H86N12O16S2Pureza:98.95%Forma y color:White SolidPeso molecular:1139.391-Linoleoyl Glycerol
CAS:1-Linoleoyl Glycerol (Monolinolein) is fatty acid glycerol that has been isolated from Saururus Chinensis roots.Fórmula:C21H38O4Pureza:98.95% - 99.9%Forma y color:SolidPeso molecular:354.52ONO-RS-082
CAS:ONO-RS-082 is a Ca2+-independent phospholipase A2 inhibitor.Fórmula:C21H22ClNO3Pureza:99.35%Forma y color:SolidPeso molecular:371.86AA26-9
CAS:AA26-9 is an effective and broad-spectrum inhibitor of serine hydrolase.Fórmula:C7H10N4OPureza:99.88%Forma y color:White SolidPeso molecular:166.18Ref: TM-T3990
1mg34,00€2mg49,00€5mg74,00€1mL*10mM (DMSO)82,00€10mg113,00€25mg200,00€50mg333,00€100mg495,00€ML-211
CAS:ML-211 is a carbamate-based dual inhibitor of LYPLA1 (IC50 = 17 nM) and the related LYPLA2 (IC50 = 30 nM)Fórmula:C25H30N4O2Pureza:97.07%Forma y color:SolidPeso molecular:418.53Ref: TM-T8974
1mg114,00€1mL*10mM (DMSO)219,00€5mg222,00€10mg313,00€25mg497,00€50mg670,00€100mg888,00€1-Naphthaleneacetic acid potassium salt
CAS:1-Naphthaleneacetic acid potassium salt (1-NAA Potassium Salt) is a synthetic phytogrowth hormone that promotes plant growth and a PLA2 inhibitor.Fórmula:C12H9O2·KPureza:97.68%Forma y color:Off-White To Beige PowderPeso molecular:224.3Difluprednate
CAS:Difluprednate (Myser)(Durezol) is a corticosteroid, approved for the treatment of post-operative ocular inflammation and pain.Fórmula:C27H34F2O7Pureza:99.23% - 99.86%Forma y color:SolidPeso molecular:508.55Cambinol
CAS:Cambinol is a SIRT1/2 inhibitor (IC50: 56/59 μM), non-competitive with NAD, weak on SIRT5, and prompts apoptosis in lymphoma cells.Fórmula:C21H16N2O2SPureza:98.02% - 99.83%Forma y color:SolidPeso molecular:360.43Ref: TM-T4019
1mg38,00€2mg50,00€1mL*10mM (DMSO)63,00€5mg80,00€10mg117,00€25mg207,00€50mg333,00€100mg495,00€500mg1.071,00€CAY10594
CAS:CAY10594, a PLD2 inhibitor, mitigates acetaminophen liver damage via the p-GSK-3β/JNK pathway.Fórmula:C26H28N4O2Pureza:97.76%Forma y color:White SolidPeso molecular:428.53trans-Benzylideneacetone
CAS:trans-Benzylideneacetone (Acetocinnamone) is used in various synthetic preparations.Fórmula:C10H10OPureza:97.48%Forma y color:SolidPeso molecular:146.19Aristolochic acid C
CAS:Aristolochic acid C is a derivative of Aristolochic acid which is a phospholipase A2 inhibitor.Fórmula:C16H9NO7Pureza:99.8%Forma y color:Orange SolidPeso molecular:327.25N-(p-amylcinnamoyl) Anthranilic Acid
CAS:N-(p-amylcinnamoyl) Anthranilic Acid (ACA) is a broad spectrum Phospholipase A2 (PLA2) inhibitor and TRP channel blocker.Fórmula:C21H23NO3Pureza:99.35% - 99.75%Forma y color:White SolidPeso molecular:337.41U-73122
CAS:U-73122 (U73122) , an effective PLC inhibitor, reduces agonist-induced Ca2+ increases in platelets and PMN.Fórmula:C29H40N2O3Pureza:97.50% - 98.66%Forma y color:White SolidPeso molecular:464.64m-3M3FBS
CAS:m-3M3FBS is a phospholipase C (PLC) activator.Fórmula:C16H16F3NO2SPureza:99.66%Forma y color:SolidPeso molecular:343.36Melittin
CAS:Melittin: principal bee venom toxin, 26 amino acids, activates low-weight PLA2, not high-weight PLA2.Fórmula:C131H229N39O31Pureza:98.37% - 99.92%Forma y color:SolidPeso molecular:2846.46Neomycin sulfate
CAS:Neomycin sulfate (Framycin sulfate) is a broad-spectrum aminoglycoside antibiotic that blocks the synthesis of bacterial proteins in order to exertFórmula:C23H46N6O13·3H2SO4Pureza:99.4% - 99.88%Forma y color:Yellow SolidPeso molecular:908.87
