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Receptor 5-HT

Receptor 5-HT

Los receptores 5-HT, también conocidos como receptores de serotonina, son un grupo de receptores acoplados a proteínas G (GPCR) que median los efectos de la serotonina, un neurotransmisor involucrado en la regulación del estado de ánimo, la ansiedad, el sueño, el apetito y otros procesos fisiológicos. Estos receptores se dividen en varios subtipos, cada uno con funciones y propiedades farmacológicas distintas. Los moduladores de los receptores 5-HT se estudian ampliamente por su papel en el tratamiento de la depresión, los trastornos de ansiedad y otras afecciones neuropsiquiátricas. En CymitQuimica, ofrecemos una gama de moduladores de receptores 5-HT de alta calidad para apoyar su investigación en neurofarmacología, trastornos del estado de ánimo y señalización GPCR.

Se han encontrado 940 productos de "Receptor 5-HT"

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  • Fluvoxamine maleate

    CAS:
    <p>Fluvoxamine maleate (DU-23000 (maleate)) is a selective serotonin reuptake inhibitor that is used in the treatment of depression and a variety of anxiety</p>
    Fórmula:C19H25F3N2O6
    Pureza:99.92% - 99.94%
    Forma y color:White Crystalline Powder
    Peso molecular:434.41
  • Mianserin hydrochloride

    CAS:
    <p>Mianserin HCl (Org GB 94): a tetracyclic antidepressant; blocks alpha-adrenergic, H1, serotonin receptors; may induce drowsiness, hematological issues.</p>
    Fórmula:C18H21ClN2
    Pureza:99.63% - 99.82%
    Forma y color:White And Film Coated Tablet And Seem To Be White Or White-Like After Removing It'S Film Coated
    Peso molecular:300.83
  • JNJ-18038683

    CAS:
    <p>JNJ-18038683 is a 5-Hydroxytryptamine Type 7 (5-HT7) receptor antagonist, with pKis of 8.19, 8.20 for rat and human 5-HT7 in HEK293 cells, respectively.</p>
    Fórmula:C26H28ClN3O7
    Pureza:97.29%
    Forma y color:Solid
    Peso molecular:529.97
  • Mebhydrolin napadisylate

    CAS:
    <p>Mebhydrolin napadisylate (Incidal) is an antihistamine used to relieve allergic symptoms caused by histamine release, including nasal allergies and allergic</p>
    Fórmula:C19H20N2C10H8O6S2
    Pureza:99.35% - 99.96%
    Forma y color:White Or Almost White Crystalline
    Peso molecular:420.52
  • Cyproheptadine hydrochloride sesquihydrate

    CAS:
    <p>Cyproheptadine hydrochloride sesquihydrate (Peritol), an antihistamine, is an antagonist of serotonin and histamine2.</p>
    Fórmula:C21H24ClNO
    Pureza:99.77% - >99.99%
    Forma y color:White To Slightly Yellowish Crystalline Solid
    Peso molecular:341.88
  • Bufotenidine hydrochloride(487-91-2 Free base)

    CAS:
    <p>Bufotenidine hydrochloride(487-91-2 Free base) is a natural product for research related to life sciences.</p>
    Fórmula:C13H19ClN2O
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:254.76
  • Promazine hydrochloride

    CAS:
    <p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>
    Fórmula:C17H21ClN2S
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:320.88
  • Naftidrofuryl oxalate

    CAS:
    <p>Naftidrofuryl oxalate treats peripheral/cerebral vascular issues, boosts cell oxidation, is spasmolytic, and may block 5HT-2 serotonin receptors.</p>
    Fórmula:C26H35NO7
    Pureza:97.12% - 98.38%
    Forma y color:Solid
    Peso molecular:473.56
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Fórmula:C21H26ClN3OS
    Pureza:99.3% - 99.99%
    Forma y color:Solid
    Peso molecular:403.97
  • Vilazodone

    CAS:
    <p>Vilazodone (SB659746A): an SSRI and 5-HT-1A agonist, boosts serotonin to treat depression and anxiety.</p>
    Fórmula:C26H27N5O2
    Pureza:99.61%
    Forma y color:Light Yellow Solid
    Peso molecular:441.52
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:383.51
  • Desipramine hydrochloride

    CAS:
    <p>Desipramine hydrochloride (Norimipramine) ,a secondary amine tricyclic antidepressant (TCA), is the hydrochloride salt form of desipramine.</p>
    Fórmula:C18H23ClN2
    Pureza:99.58% - 99.94%
    Forma y color:White To Off-White Powder
    Peso molecular:302.842
  • Dexchlorpheniramine Maleate

    CAS:
    <p>Dexchlorpheniramine Maleate, an antihistamine with anticholinergic effects, treats allergies like hay fever. It's the active isomer of chlorpheniramine.</p>
    Fórmula:C20H23ClN2O4
    Pureza:99.58%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:390.86
  • NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Fórmula:C20H24ClN3O
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:357.88
  • Granisetron hydrochloride

    CAS:
    <p>Granisetron hydrochloride (Granisetron HCl) is a serotonin receptor (5HT-3 selective) antagonist that has been used as an antiemetic for cancer chemotherapy</p>
    Fórmula:C18H25ClN4O
    Pureza:99.88% - 99.93%
    Forma y color:White To Off-White Crystalline Solid
    Peso molecular:348.87
  • Alosetron hydrochloride

    CAS:
    <p>Alosetron hydrochloride (GR 68755), a selective 5-HT3 receptor antagonist, can block the actions of serotonin at 5-HT3 sites in the peripheral nervous system.</p>
    Fórmula:C17H19ClN4O
    Pureza:99.90%
    Forma y color:Off-White Powder
    Peso molecular:330.81
  • Molindone hydrochloride

    CAS:
    <p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>
    Fórmula:C16H24N2O2·HCl
    Pureza:99% - 99.99%
    Forma y color:Solid
    Peso molecular:312.84
  • Aniracetam

    CAS:
    <p>Aniracetam (Ro 13-5057)(Ro 13-5057), a nootropic and neuroprotective drug, selectively modulates the AMPA receptor and nAChR.</p>
    Fórmula:C12H13NO3
    Pureza:99.88% - 99.89%
    Forma y color:White Crystalline Or Crystalline Powde
    Peso molecular:219.24
  • Cericlamine

    CAS:
    <p>Cericlamine is a selective 5-hydroxytryptamine (5-HT) reuptake blocker with antidepressant activity.</p>
    Fórmula:C12H17Cl2NO
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:262.18
  • Pimethixene

    CAS:
    <p>Pimethixene (Calmixen) blocks 5-HT1A, 2A/B/C, H1, D2/D4.4 &amp; muscarinic M1/M2 receptors; potent with pKis 7.54-10.44.</p>
    Fórmula:C19H19NS
    Pureza:97.50%
    Forma y color:Solid
    Peso molecular:293.43