GluR
Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.
Se han encontrado 255 productos de "GluR"
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Org-26576
CAS:<p>Org-26576 is a positive allosteric modulator of the AMPA receptor.</p>Fórmula:C11H12N2O2Pureza:99.67%Forma y color:SolidPeso molecular:204.23AZD-8529 mesylate
CAS:<p>AZD-8529 mesylate is a highly selective, and orally bioavailable positive allosteric modulator of mGluR2 (EC50: 285 nM).</p>Fórmula:C25H28F3N5O6SPureza:99.19%Forma y color:SolidPeso molecular:583.58DHPG
CAS:<p>DHPG is a potent Group I mGluR agonist; doesn't affect Group II/III; linked to phospholipase D.</p>Fórmula:C8H9NO4Pureza:99.55%Forma y color:SolidPeso molecular:183.16NBQX disodium
CAS:<p>NBQX Disodium (FG9202 disodium) is a highly selective, competitive AMPA receptor antagonist with neuroprotective and anticonvulsant activity.</p>Fórmula:C12H6N4Na2O6SPureza:97.6% - 98.22%Forma y color:SolidPeso molecular:380.2415LY339434 HCl
<p>LY339434 HCl is a low affinity GluR5 erythrocyte receptor agonist.LY339434 HCl causes rapid neuronal death primarily by affecting N-methyl-D-aspartate (NMDA)</p>Fórmula:C18H20ClNO4Pureza:97.96% - 99.68%Forma y color:SoildPeso molecular:349.81Decoglurant
CAS:<p>Decoglurant (RO4995819) is a negative allosteric modulator of mGluR2 and mGluR3 and it also is developed as an antidepressant.</p>Fórmula:C21H11F6N5Pureza:99.77%Forma y color:SolidPeso molecular:447.34Piracetam
CAS:<p>Piracetam (UCB-6215), a cyclic derivative of the neurotransmitter gamma-aminobutyric acid (GABA), is used in therapy of the extensive cognitive disorders.</p>Fórmula:C6H10N2O2Pureza:97.16%Forma y color:Crystals From Isopropanol SolidPeso molecular:142.16(R)-3,4-DCPG HCl
<p>(R)-3,4-DCPG HCl is a potent and selective mGlu8a receptor agonist that activates metabotropic glutamate receptors on primary afferent terminals in the neonatal</p>Fórmula:C10H10ClNO6Pureza:98.80% - 99.89%Forma y color:SoildPeso molecular:275.64VU0650786
CAS:<p>VU0650786: selective mGlu3 NAM, CNS-penetrant, IC50 392 nM, shows antidepressant/anxiolytic effects in rodents.</p>Fórmula:C18H15ClFN5O2Pureza:99.09%Forma y color:SolidPeso molecular:387.8KM02894
CAS:<p>KM02894 inhibits glutamate release, potentially reducing cancer-induced bone pain in tumor studies.</p>Fórmula:C7H9N3OS2Pureza:99.98%Forma y color:SolidPeso molecular:215.3γ-DGG acetate(6729-55-1 free base)
CAS:<p>gamma-DGG acetate(6729-55-1 free base) (γ-D-Glutamylglycine) is a competitive blocker of AMPA receptor.</p>Fórmula:C9H16N2O7Pureza:99.81%Forma y color:SolidPeso molecular:264.23Basimglurant
CAS:<p>Basimglurant (CTEP Derivative) is a potent, selective and orally available modulator of mGlu5 negative allosteric(Kd of 1.1 nM).</p>Fórmula:C18H13ClFN3Pureza:98.35%Forma y color:SolidPeso molecular:325.77(R)-ADX-47273
CAS:<p>(R)-ADX-47273 is a potent mGluR5 positive allosteric modulator(EC50 of 168 nM for potentiation ).</p>Fórmula:C20H17F2N3O2Pureza:99.87%Forma y color:SolidPeso molecular:369.36GYKI-47261 dihydrochloride
CAS:<p>GYKI-47261 dihydrochloride is an AMPA receptor antagonist and CYP2E1 inducer, demonstrating broad-spectrum anticonvulsant and neuroprotective activities.</p>Fórmula:C18H17Cl3N4Pureza:98.32% - 99.14%Forma y color:SolidPeso molecular:395.71MMPIP hydrochloride
CAS:<p>MMPIP hydrochloride is a selective antagonist of allosteric mGluR7.</p>Fórmula:C19H16ClN3O3Pureza:99.88%Forma y color:SolidPeso molecular:369.8(S)-3,4-DCPG HCl
<p>(S)-3,4-DCPG HCl is a selective mGluR8a agonist, impacting AV12-664 cells with an EC50 of 31 nM.</p>Fórmula:C10H10ClNO6Pureza:99.53% - 99.9%Forma y color:SoildPeso molecular:275.64(S)-3,4-DCPG
CAS:<p>(S)-3,4-DCPG ((S)-3,4-Dicarboxyphenylglycine) is a selective agonist of human metabotropic glutamate receptor 8a (mGluR8a).</p>Fórmula:C10H9NO6Pureza:98%Forma y color:SolidPeso molecular:239.18STX-107
CAS:<p>STX-107 is a potent and selective mGluR5 agonist for the study of Fragile X Syndrome.</p>Fórmula:C18H10FN3SPureza:99.17%Forma y color:SolidPeso molecular:319.36(S)-AMPA HCl
<p>(S)-AMPA HCl (L-AMPA HCl) is a selective AMPA receptor agonist with potential antidepressant activity. It can be used in research on Parkinson's disease.</p>Fórmula:C7H11ClN2O4Pureza:99.18%Forma y color:SolidPeso molecular:222.63MGS0274
CAS:<p>MGS0274, a lipophilic prodrug of mGlu2/3 agonist MGS0008, enhances oral bioavailability, potentially aiding schizophrenia research.</p>Fórmula:C21H32FNO7Forma y color:SolidPeso molecular:429.485ML353
<p>ML353 activates TREK-1/2, binds mGlu5 SAM (Ki=18.2 nM), surpasses 5mpep, may address SAM activity/blocking.</p>Fórmula:C19H15FN2OPureza:99.98% - 99.98%Forma y color:SoildPeso molecular:306.331H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)-
CAS:<p>1H-Pyrrolo[2,1-c][1,2,4]benzothiadiazine, 2,3,3a,4-tetrahydro-, 5,5-dioxide, (3aR)- is a low activity isomer of S 18986.</p>Fórmula:C10H12N2O2SPureza:99.96%Forma y color:SoildPeso molecular:224.28VU0483605
CAS:<p>VU0483605 is an effective and selective positive allosteric modulator of mGluR1 with EC50s of 390 and 356 nM for human and rat, respectively.</p>Fórmula:C20H10Cl3N3O3Pureza:99.61%Forma y color:SolidPeso molecular:446.67(S,S)-BMS-984923
CAS:<p>(S,S)-BMS-984923 is a weak mGluR5 modulator with EC50 >1μM; less active than its potent counterpart.</p>Fórmula:C22H15ClN2O2Forma y color:SolidPeso molecular:374.82KRP-199 sodium
<p>KRP-199 sodium sodium is highly potent and selective for AMPA-R in vitro and exhibits good neuroprotection in vivo.</p>Fórmula:C22H12F3N5Na2O7Pureza:97.27%Forma y color:SoildPeso molecular:561.33(±)-LY367385
CAS:<p>(±)-LY367385 is the racemic form of LY367385, and LY367385 is a highly potent and selective mGluR1a antagonist.</p>Fórmula:C10H11NO4Forma y color:SolidPeso molecular:209.201Pomaglumetad methionil anhydrous
CAS:<p>LY2140023, potential schizophrenia treatment, is an oral prodrug of LY404039, a selective mGlu2/3 agonist.</p>Fórmula:C12H18N2O7S2Pureza:98%Forma y color:SolidPeso molecular:366.41LY2812223
CAS:<p>LY2812223: selective mGlu2 agonist; binds mGlu2/mGlu3 (Ki=144/156 nM).</p>Fórmula:C10H12N4O4SPureza:98%Forma y color:SolidPeso molecular:284.29LY3027788 hydrochloride
CAS:<p>LY3027788 HCl, potent oral prodrug of LY3020371, targets mGlu2/3 with antidepressant effects.</p>Fórmula:C25H32ClF2NO11SForma y color:SolidPeso molecular:628.03MGS0028
CAS:<p>MGS0028 is a selective agonist of metabotropic glutamate 2/3 receptor, it could reverse abnormal behaviors in mice induced by isolation rearing.</p>Fórmula:C8H8FNO5Forma y color:SolidPeso molecular:217.15LY3020371
CAS:<p>LY3020371: potent, selective mGlu 2/3 receptor antagonist with Ki of 5.26 nM (hmGluR2) and 2.50 nM (hmGluR3); key in depression studies.</p>Fórmula:C15H15F2NO5SForma y color:SolidPeso molecular:359.34L-AP3
CAS:<p>L-AP3 blocks mGluR, inhibits D/L-phosphoserine (IC50: 368/2087 μM).</p>Fórmula:C3H8NO5PForma y color:White Hygroscopic SolidPeso molecular:169.073JF-NP-26
<p>Releases pain-blocking raseglurant under 405 nm light. Inhibits Quisqualate. Analgesic in vivo. Quantum yield: 0.18.</p>Forma y color:SolidLY3027788
CAS:<p>LY3027788, potent oral prodrug of LY3020371, is a strong mGlu2/3 antagonist with notable antidepressant effects.</p>Fórmula:C25H31F2NO11SForma y color:SolidPeso molecular:591.58mGluR5 modulator 1
CAS:<p>mGluR5 modulator 1 is a positive modulator for mGluR5, used in schizophrenia and cognitive research.</p>Fórmula:C18H19ClFN3O2Forma y color:SolidPeso molecular:363.82MPPG
CAS:<p>MPPG is a selective L-AP4-sensitive receptor antagonist (kD=9.2 μM).</p>Fórmula:C9H12NO5PForma y color:SolidPeso molecular:245.171mGluR3 modulator-1
CAS:<p>1-ethyl-3-morpholin-4-yl tetrahydroisoquinoline: mGluR3 modulator, potential for Parkinson's.</p>Fórmula:C16H21N3OPureza:98.99%Forma y color:SolidPeso molecular:271.36VU0364770 hydrochloride
CAS:<p>VU0364770 hydrochloride: potent, selective mGlu4 PAM; EC50=290 nM (rat), 1.1 μM (human).</p>Fórmula:C12H10Cl2N2OPureza:98%Forma y color:SolidPeso molecular:269.13NS-102
CAS:<p>NS-102 is a glutamate receptor and NMDA receptor antagonist that inhibits erythrocyanine (GluK2) and inhibits specific binding to the glur6 receptor.</p>Fórmula:C12H11N3O4Pureza:98.48% - 98.95%Forma y color:SolidPeso molecular:261.23AMN082
CAS:<p>AMN082 is an mGluR7 agonist with antidepressant effects. Neuroprotective effect of AMN082 on neuronal apoptosis in rats with traumatic brain injury.</p>Fórmula:C28H30Cl2N2Pureza:97.13% - 98.63%Forma y color:SolidPeso molecular:465.46LY487379
CAS:<p>LY487379: human mGluR2 PAM, boosts glutamate binding, aids cognitive flexibility, may treat schizophrenia. EC50: 1.7 μM (mGlu2), >10 μM (mGlu3).</p>Fórmula:C21H19F3N2O4SForma y color:SolidPeso molecular:452.45VU0422288
CAS:<p>VU0422288 (ML396) is a type III mGlu receptor (mGlus) orthosteric modulator with inhibitory effects on mGluR4.VU0422288 can be used to study Rett syndrome.</p>Fórmula:C17H11Cl2N3O2Pureza:95.48%Forma y color:SolidPeso molecular:360.19GYKI 52466 dihydrochloride
CAS:<p>GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used to study neurological diseases.</p>Fórmula:C17H17Cl2N3O2Pureza:99.38%Forma y color:SolidPeso molecular:366.24GYKI 53655 hydrochloride
CAS:<p>GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the study of neurological disorders.</p>Fórmula:C19H21ClN4O3Pureza:98.02%Forma y color:SolidPeso molecular:388.85JNJ-46778212
CAS:<p>JNJ-46778212 (VU 0409551) is a selective and potent mGlu5 allosteric modulator (EC50: 260 nM) for the study of neurodissection.</p>Fórmula:C20H17FN2O3Pureza:99.24%Forma y color:SolidPeso molecular:352.36Ro 01-6128
CAS:<p>Positive allosteric modulator of mGlu1 receptors</p>Fórmula:C17H17NO3Pureza:98%Forma y color:SolidPeso molecular:283.32EGLU
CAS:<p>EGLU, an antidepressant and potent mGluR-2 antagonist, binds with a 66 μM Kd to (lS,3S)-ACPD sites.</p>Fórmula:C7H13NO4Pureza:99.98%Forma y color:SolidPeso molecular:175.18LY341495
CAS:<p>LY341495 is a potent metabotropic glutamate receptor antagonist and can be used to study neurological disorders.</p>Fórmula:C20H19NO5Pureza:98.53% - 99.37%Forma y color:SolidPeso molecular:353.37γ-DGG
CAS:<p>gamma-DGG is a competitive blocker of AMPA receptor.</p>Fórmula:C7H12N2O5Pureza:98%Forma y color:SolidPeso molecular:204.18CFMTI
CAS:<p>CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.</p>Fórmula:C19H16FN5OPureza:97.23%Forma y color:SolidPeso molecular:349.36Chelidamic acid
CAS:<p>Chelidamic acid is a heterocyclic organic acid with a pyran skeleton. Chelidamic acid is inhibitors of glutamate decarboxylase, with a Ki of 33 μM.</p>Fórmula:C7H5NO5Pureza:98.11%Forma y color:Pale Yellow PowderPeso molecular:183.12VU-1545
CAS:<p>VU-1545 is mGlu5 positive allosteric modulator.</p>Fórmula:C22H15FN4O3Pureza:98.8%Forma y color:SolidPeso molecular:402.38(RS)-3-Hydroxyphenylglycine
CAS:<p>(RS)-3-Hydroxyphenylglycine is a PI-linked metabotropic glutamate receptors agonist.</p>Fórmula:C8H9NO3Pureza:99.29%Forma y color:SolidPeso molecular:167.16FTIDC
CAS:<p>FTIDC: potent, selective mGluR1 allosteric antagonist, weak on mGluR5. IC50: human 5.8 nM, mouse 3.1 nM. Noncompetitive.</p>Fórmula:C18H23FN6OPureza:94.58%Forma y color:SolidPeso molecular:358.41E4CPG
CAS:<p>E4CPG is a novel group I/II metabotropic glutamate receptor antagonist, more potent than (RS)-MCPG.</p>Fórmula:C11H13NO4Pureza:99.96%Forma y color:SolidPeso molecular:223.23DNQX
CAS:<p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C8H4N4O6Pureza:97.27% - 99.1%Forma y color:Off-White Powder With A Yellow TingePeso molecular:252.14VU-29
CAS:<p>VU-29 is a positive allosteric mGlu5 receptor modulator with EC50=9 nM and Ki=244 nM for rmGluR5. It is selective for mGluR5 relative to other mGluR subtypes.</p>Fórmula:C22H16N4O3Pureza:99.63%Forma y color:SolidPeso molecular:384.39VU0361737
CAS:<p>VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.</p>Fórmula:C13H11ClN2O2Pureza:99.60% - 99.85%Forma y color:SolidPeso molecular:262.69(S)-ATPO
CAS:<p>(S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.</p>Fórmula:C11H19N2O7PPureza:98.37% - 99.41%Forma y color:SolidPeso molecular:322.25CX614
CAS:<p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>Fórmula:C13H13NO4Pureza:97.37%Forma y color:SolidPeso molecular:247.25ADX-47273
CAS:<p>ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).</p>Fórmula:C20H17F2N3O2Pureza:97% - 99.18%Forma y color:SolidPeso molecular:369.36Farampator
CAS:<p>Farampator (CX-691) (CX-691;Org24448) is a positive modulator of AMPA receptor.</p>Fórmula:C12H13N3O2Pureza:99.84% - >99.99%Forma y color:SolidPeso molecular:231.25AZD-8529
CAS:<p>AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.</p>Fórmula:C24H24F3N5O3Forma y color:SolidPeso molecular:487.47NBQX
CAS:<p>NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.</p>Fórmula:C12H8N4O6SPureza:97.66% - 99.42%Forma y color:SolidPeso molecular:336.28XAP044
CAS:<p>XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.</p>Fórmula:C15H9IO4Pureza:97.41%Forma y color:SolidPeso molecular:380.13ADX88178
CAS:<p>ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.</p>Fórmula:C12H12N6SPureza:99.55%Forma y color:SolidPeso molecular:272.33SIB-1757
CAS:<p>SIB-1757 (6-methyl-2-[(E)-phenyldiazenyl]pyridin-3) is a selective antagonist of mGlu5 metabotropic glutamate receptor subtype (hmGlu5, IC50 : 0.4 μM)</p>Fórmula:C12H11N3OPureza:97.37%Forma y color:SolidPeso molecular:213.24MPEP
CAS:<p>MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.</p>Fórmula:C14H11NPureza:99.54%Forma y color:SolidPeso molecular:193.24(RS)-MCPG
CAS:<p>(RS)-MCPG ((±)-MCPG) is a non-selective group I/II metabotropic glutamate receptor antagonist.</p>Fórmula:C10H11NO4Pureza:99.96%Forma y color:SolidPeso molecular:209.2TCN238
CAS:<p>TCN238 is an orally bioavailable positive allosteric modulator of the metabotropic glutamate receptor 4 (mGluR4with an EC50 of 1 μM).</p>Fórmula:C12H11N3Pureza:99.9% - 99.92%Forma y color:SolidPeso molecular:197.24VU0364770
CAS:<p>VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu</p>Fórmula:C12H9ClN2OPureza:99.65% - >99.99%Forma y color:SolidPeso molecular:232.67CNQX
CAS:<p>CNQX (FG9065) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.3 and 1.5 μM for AMPA and kainate receptors, respectively)</p>Fórmula:C9H4N4O4Pureza:99.70%Forma y color:Pale Yellow SolidPeso molecular:232.15PHCCC
CAS:<p>PHCCC is a Group I mGluR antagonist and enhances mGluR4 function; also blocks mGluR2/8.</p>Fórmula:C17H14N2O3Pureza:>99.99%Forma y color:SolidPeso molecular:294.31-BCP
CAS:<p>1-BCP (Piperonylic acid piperidide) is a centrally active drug that modulates AMPA receptor gated currents.</p>Fórmula:C13H15NO3Pureza:99.60%Forma y color:SolidPeso molecular:233.26(S)-3-Hydroxyphenylglycine
CAS:<p>(S)-3-Hydroxyphenylglycine is an agonist of group I metabotropic glutamate receptors (mGluRs).</p>Fórmula:C8H9NO3Pureza:99.65%Forma y color:SolidPeso molecular:167.16JNJ16259685
CAS:<p>JNJ16259685 (TN.T 16259685) is a selective mGluR1 antagonist, and inhibits the synaptic activation of mGluR1 in a concentration-dependent manner with IC50 of 19</p>Fórmula:C20H23NO3Pureza:98.31%Forma y color:SolidPeso molecular:325.4Lu AF21934
CAS:<p>Lu AF21934 is a brain-penetrant and selective mGlu4 receptor positive allosteric modulator (IC50: 500 nM, human).</p>Fórmula:C14H16Cl2N2O2Pureza:99.79%Forma y color:SolidPeso molecular:315.2LY-404187
CAS:<p>LY404187 is a positive allosteric modulator of AMPA receptors</p>Fórmula:C19H22N2O2SPureza:99.34%Forma y color:SolidPeso molecular:342.46IDRA-21
CAS:<p>IDRA-21 is a positive AMPA receptor modulator.</p>Fórmula:C8H9ClN2O2SPureza:99.73%Forma y color:SolidPeso molecular:232.69trans-ACPD
CAS:<p>trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.</p>Fórmula:C7H11NO4Pureza:99.53%Forma y color:SolidPeso molecular:173.17Ro0711401
CAS:<p>Ro0711401 is an agonist of mGlu1 receptor.</p>Fórmula:C18H11F3N2O3Pureza:97.57%Forma y color:SolidPeso molecular:360.29YM90K
CAS:<p>YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.</p>Fórmula:C11H8ClN5O4Pureza:98.23%Forma y color:SolidPeso molecular:309.66HBT1
CAS:<p>HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons</p>Fórmula:C16H17F3N4O2SPureza:99.52%Forma y color:SolidPeso molecular:386.393-MATIDA
CAS:<p>3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).</p>Fórmula:C8H9NO4SPureza:99.75% - 99.96%Forma y color:SolidPeso molecular:215.23VU 0357121
CAS:<p>VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.</p>Fórmula:C17H17F2NO2Pureza:99% - >99.99%Forma y color:SolidPeso molecular:305.32MTEP hydrochloride
CAS:<p>MTEP hydrochloride (MTEP) is non-competitive mGlu5 antagonist (IC50 and Ki of 5 nM and 16 nM, respectively)</p>Fórmula:C11H9ClN2SPureza:99.58%Forma y color:SolidPeso molecular:236.72FITM
CAS:<p>FITM is a potent negative allosteric modulator of mGlu1 receptor(Ki : 2.5 nM).</p>Fórmula:C18H18FN5OSPureza:97.25%Forma y color:SolidPeso molecular:371.43ML 254
CAS:<p>是一种化学合成中的砌块</p>Fórmula:C18H15FN2O2Pureza:98.09%Forma y color:SolidPeso molecular:310.32AMN082 free base
CAS:<p>AMN082 free base is a metabotropic glutamate receptor 7 allosteric agonist.</p>Fórmula:C28H28N2Pureza:97.75% - 97.79%Forma y color:SolidPeso molecular:392.54MPEP hydrochloride
CAS:<p>MPEP hydrochloride is an effective and highly specific non-competitive antagonist at the mGlu5 receptor subtype (IC50: 36 nM).</p>Fórmula:C14H12ClNPureza:99.87% - >99.99%Forma y color:SolidPeso molecular:229.7CX516
CAS:<p>CX516 (Ampalex), an ampakine and nootropic, acts as an AMPA receptor positive allosteric modulator as a therapy for Alzheimer's disease, schizophrenia and MCI.</p>Fórmula:C14H15N3OPureza:99.04% - ≥95%Forma y color:Tan SolidPeso molecular:241.29MTEP
CAS:<p>MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.</p>Fórmula:C11H8N2SForma y color:SolidPeso molecular:200.26Ro 67-7476
CAS:<p>Ro 67-7476 is a positive allosteric modulator of mGlu1 receptors.</p>Fórmula:C17H18FNO2SPureza:99.69%Forma y color:SolidPeso molecular:319.39CTEP
CAS:<p>CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold</p>Fórmula:C19H13ClF3N3OPureza:99.17%Forma y color:SolidPeso molecular:391.77VU0155094
CAS:<p>VU0155094 (ML 397) is a positive allosteric modulator with differential activity at the various group III mGluRs.</p>Fórmula:C24H24N2O4SPureza:97.21%Forma y color:SolidPeso molecular:436.52Caroverine hydrochloride
CAS:<p>Caroverine HCL: Blocks NMDA/AMPA receptors, antioxidant, calcium-blocker, and vasorelaxant, used for tinnitus research.</p>Fórmula:C22H28ClN3O2Pureza:98.37% - 98.75%Forma y color:SolidPeso molecular:401.9VU 0364439
CAS:<p>VU 0364439 is a mGlu4 positive allosteric modulator (C50: 19.8 nM).</p>Fórmula:C18H13Cl2N3O3SPureza:97.9%Forma y color:SolidPeso molecular:422.29JNJ-42153605
CAS:<p>JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).</p>Fórmula:C22H23F3N4Pureza:97.25% - 98.57%Forma y color:SolidPeso molecular:400.44VU0155041
CAS:<p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>Fórmula:C14H15Cl2NO3Pureza:99.52% - 99.56%Forma y color:SolidPeso molecular:316.18JNJ-40411813
CAS:<p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>Fórmula:C20H25ClN2OPureza:99.74%Forma y color:SolidPeso molecular:344.88
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