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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Se han encontrado 255 productos de "GluR"

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  • LY341495

    CAS:
    <p>LY341495 is a potent metabotropic glutamate receptor antagonist and can be used to study neurological disorders.</p>
    Fórmula:C20H19NO5
    Pureza:98.53% - 99.37%
    Forma y color:Solid
    Peso molecular:353.37
  • GYKI 53655 hydrochloride

    CAS:
    <p>GYKI 53655 hydrochloride (LY300168 hydrochloride) is an antagonist of AMPA and is used in the study of neurological disorders.</p>
    Fórmula:C19H21ClN4O3
    Pureza:98.02%
    Forma y color:Solid
    Peso molecular:388.85
  • JNJ-46778212

    CAS:
    <p>JNJ-46778212 (VU 0409551) is a selective and potent mGlu5 allosteric modulator (EC50: 260 nM) for the study of neurodissection.</p>
    Fórmula:C20H17FN2O3
    Pureza:99.24%
    Forma y color:Solid
    Peso molecular:352.36
  • GYKI 52466 dihydrochloride

    CAS:
    <p>GYKI 52466 dihydrochloride is an AMPA/Kainate receptor antagonist with anticonvulsant activity and can be used to study neurological diseases.</p>
    Fórmula:C17H17Cl2N3O2
    Pureza:99.38%
    Forma y color:Solid
    Peso molecular:366.24
  • γ-DGG

    CAS:
    <p>gamma-DGG is a competitive blocker of AMPA receptor.</p>
    Fórmula:C7H12N2O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:204.18
  • VU0364770 hydrochloride

    CAS:
    <p>VU0364770 hydrochloride: potent, selective mGlu4 PAM; EC50=290 nM (rat), 1.1 μM (human).</p>
    Fórmula:C12H10Cl2N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:269.13
  • Ro 01-6128

    CAS:
    <p>Positive allosteric modulator of mGlu1 receptors</p>
    Fórmula:C17H17NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:283.32
  • VU0422288

    CAS:
    <p>VU0422288 (ML396) is a type III mGlu receptor (mGlus) orthosteric modulator with inhibitory effects on mGluR4.VU0422288 can be used to study Rett syndrome.</p>
    Fórmula:C17H11Cl2N3O2
    Pureza:95.48%
    Forma y color:Solid
    Peso molecular:360.19
  • AMN082

    CAS:
    <p>AMN082 is an mGluR7 agonist with antidepressant effects. Neuroprotective effect of AMN082 on neuronal apoptosis in rats with traumatic brain injury.</p>
    Fórmula:C28H30Cl2N2
    Pureza:97.13% - 98.63%
    Forma y color:Solid
    Peso molecular:465.46
  • CFMTI

    CAS:
    <p>CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.</p>
    Fórmula:C19H16FN5O
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:349.36
  • (S)-ATPO

    CAS:
    <p>(S)-ATPO is Competitive antagonist at GluR1-4 (AMPA-preferring) receptors.</p>
    Fórmula:C11H19N2O7P
    Pureza:98.37% - 99.41%
    Forma y color:Solid
    Peso molecular:322.25
  • MTEP

    CAS:
    <p>MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.</p>
    Fórmula:C11H8N2S
    Forma y color:Solid
    Peso molecular:200.26
  • Ro0711401

    CAS:
    <p>Ro0711401 is an agonist of mGlu1 receptor.</p>
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Forma y color:Solid
    Peso molecular:360.29
  • DNQX

    CAS:
    <p>DNQX (FG 9041) is a competitive, non-NMDA glutamate receptor antagonist (IC50s = 0.5 and 0.1 μM for AMPA and kainate receptors, respectively)</p>
    Fórmula:C8H4N4O6
    Pureza:97.27% - 99.1%
    Forma y color:Off-White Powder With A Yellow Tinge
    Peso molecular:252.14
  • VU0155041

    CAS:
    <p>VU0155041 is an effective and positive allosteric modulator/allosteric agonist at mGlu4 receptors (EC50: 798/693 nM, at human/rat).</p>
    Fórmula:C14H15Cl2NO3
    Pureza:99.52% - 99.56%
    Forma y color:Solid
    Peso molecular:316.18
  • VU0361737

    CAS:
    <p>VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.</p>
    Fórmula:C13H11ClN2O2
    Pureza:99.60% - 99.85%
    Forma y color:Solid
    Peso molecular:262.69
  • ADX88178

    CAS:
    <p>ADX88178 is a potent positive allosteric modulator for metabotropic glutamate receptor 4 (mGluR4) with EC50 of 4 nM for human mGluR4.</p>
    Fórmula:C12H12N6S
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:272.33
  • JNJ-40411813

    CAS:
    <p>JNJ-40411813 (ADX-71149) (ADX-71149) is a new positive allosteric modulator of the metabotropic glutamate 2 receptor (mGlu2R, EC50: 147 nM).</p>
    Fórmula:C20H25ClN2O
    Pureza:99.74%
    Forma y color:Solid
    Peso molecular:344.88
  • CX614

    CAS:
    <p>CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.</p>
    Fórmula:C13H13NO4
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:247.25
  • ADX-47273

    CAS:
    <p>ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).</p>
    Fórmula:C20H17F2N3O2
    Pureza:97% - 99.18%
    Forma y color:Solid
    Peso molecular:369.36