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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Se han encontrado 265 productos de "GluR"

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productos por página.
  • CFMTI

    CAS:
    CFMTI: potent mGluR1 allosteric antagonist, 2000x selectivity over mGluR5, IC50: 2.6 nM.
    Fórmula:C19H16FN5O
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:349.36

    Ref: TM-T3482

    1mg
    57,00€
    2mg
    82,00€
    5mg
    120,00€
    1mL*10mM (DMSO)
    133,00€
    10mg
    170,00€
    25mg
    304,00€
    50mg
    432,00€
    100mg
    602,00€
  • pep2-SVKI acetate


    Pep2-SVKI acetate(pep2-SVKI acetate (328944-75-8 free base)) is a synthetic peptide salt that prevents internalization of AMPA-type glutamate receptor.
    Fórmula:C62H97N13O20
    Pureza:97.14%
    Forma y color:Solid
    Peso molecular:1344.51

    Ref: TM-TP1944L1

    1mg
    124,00€
    5mg
    271,00€
    10mg
    408,00€
    25mg
    672,00€
    50mg
    945,00€
    100mg
    1.279,00€
  • VU0361737

    CAS:
    VU0361737 (ML-128) is a mGlu4 PAM; EC50 is 240 nM (human) and 110 nM (rat), weak at mGlu5/8, inactive at mGlu1/2/3/6/7, CNS-penetrant.
    Fórmula:C13H11ClN2O2
    Pureza:99.60% - 99.85%
    Forma y color:Solid
    Peso molecular:262.69

    Ref: TM-T6726

    1mL*10mM (DMSO)
    33,00€
    25mg
    44,00€
    50mg
    69,00€
    100mg
    100,00€
    500mg
    236,00€
  • LY-404187

    CAS:
    LY404187 is a positive allosteric modulator of AMPA receptors
    Fórmula:C19H22N2O2S
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:342.46

    Ref: TM-T7706

    2mg
    35,00€
    5mg
    52,00€
    1mL*10mM (DMSO)
    58,00€
    10mg
    90,00€
    25mg
    164,00€
    50mg
    239,00€
    100mg
    339,00€
    200mg
    472,00€
  • 1-BCP

    CAS:
    1-BCP (Piperonylic acid piperidide) is a centrally active drug that modulates AMPA receptor gated currents.
    Fórmula:C13H15NO3
    Pureza:99.60%
    Forma y color:Solid
    Peso molecular:233.26

    Ref: TM-T7579

    5mg
    34,00€
    1mL*10mM (DMSO)
    38,00€
    10mg
    50,00€
    25mg
    95,00€
    50mg
    156,00€
    100mg
    231,00€
    200mg
    334,00€
  • CX614

    CAS:
    CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.
    Fórmula:C13H13NO4
    Pureza:97.37%
    Forma y color:Solid
    Peso molecular:247.25

    Ref: TM-T19698

    5mg
    52,00€
    1mL*10mM (DMSO)
    55,00€
    10mg
    78,00€
    25mg
    119,00€
    50mg
    172,00€
    100mg
    259,00€
    200mg
    388,00€
  • ADX-47273

    CAS:
    ADX-47273 (BA 94673139) is a positive and selective allosteric modulator for the metabotropic glutamate receptor subtype mGluR5(EC50=170 nM).
    Fórmula:C20H17F2N3O2
    Pureza:97% - 99.22%
    Forma y color:Solid
    Peso molecular:369.36

    Ref: TM-T2053

    2mg
    37,00€
    5mg
    52,00€
    1mL*10mM (DMSO)
    56,00€
    10mg
    82,00€
    25mg
    158,00€
    50mg
    284,00€
    100mg
    512,00€
  • AZD-8529

    CAS:
    AZD-8529: selective, oral mGluR2 modulator, EC50 285 nM; inactive on mGluR1,3-8 at 20-25 M.
    Fórmula:C24H24F3N5O3
    Forma y color:Solid
    Peso molecular:487.47

    Ref: TM-T10432

    25mg
    1.603,00€
    50mg
    2.088,00€
    100mg
    3.168,00€
  • NBQX

    CAS:
    NBQX (FG9202) is a potent, selective and competitive AMPA receptor antagonist. Neuroprotective and anticonvulsant; active in vivo.
    Fórmula:C12H8N4O6S
    Pureza:97.66% - 99.93%
    Forma y color:Solid
    Peso molecular:336.28

    Ref: TM-T4113

    1mg
    38,00€
    2mg
    50,00€
    5mg
    84,00€
    1mL*10mM (DMSO)
    92,00€
    10mg
    114,00€
    25mg
    222,00€
    50mg
    334,00€
    100mg
    497,00€
    200mg
    717,00€
  • XAP044

    CAS:
    XAP044 blocks mGlu7, inhibiting long-term potentiation in mouse brain with a half-maximal effect at 88nm.
    Fórmula:C15H9IO4
    Pureza:97.41%
    Forma y color:Solid
    Peso molecular:380.13

    Ref: TM-T21995

    1mg
    58,00€
    2mg
    82,00€
    5mg
    107,00€
    1mL*10mM (DMSO)
    146,00€
    10mg
    197,00€
    25mg
    350,00€
    50mg
    528,00€
    100mg
    755,00€
  • trans-ACPD

    CAS:
    trans-ACPD ((±)-trans-ACPD) is an equimolecular mixture of (1S, 3R)- and (1R, 3S)-ACPD.
    Fórmula:C7H11NO4
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:173.17

    Ref: TM-T3484

    1mg
    46,00€
    2mg
    59,00€
    1mL*10mM (DMSO)
    71,00€
    5mg
    94,00€
    10mg
    140,00€
    25mg
    264,00€
    50mg
    477,00€
    100mg
    692,00€
  • (RS)-MCPG

    CAS:
    (RS)-MCPG ((±)-MCPG) is a non-selective group I/II metabotropic glutamate receptor antagonist.
    Fórmula:C10H11NO4
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:209.2

    Ref: TM-T3479

    1mg
    34,00€
    5mg
    63,00€
    1mL*10mM (DMSO)
    67,00€
    10mg
    88,00€
    25mg
    168,00€
    50mg
    279,00€
    100mg
    452,00€
  • CTEP

    CAS:
    CTEP (RO 4956371) (RO4956371) is a novel, long-acting, orally bioavailable allosteric antagonist of mGlu5 receptor with IC50 of 2.2 nM, shows >1000-fold
    Fórmula:C19H13ClF3N3O
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:391.77

    Ref: TM-T6457

    2mg
    34,00€
    5mg
    50,00€
    1mL*10mM (DMSO)
    55,00€
    10mg
    88,00€
    25mg
    138,00€
    50mg
    244,00€
    100mg
    330,00€
    200mg
    470,00€
  • Ro0711401

    CAS:
    Ro0711401 is an agonist of mGlu1 receptor.
    Fórmula:C18H11F3N2O3
    Pureza:97.57%
    Forma y color:Solid
    Peso molecular:360.29

    Ref: TM-T9021

    2mg
    34,00€
    5mg
    49,00€
    1mL*10mM (DMSO)
    50,00€
    10mg
    75,00€
    25mg
    145,00€
    50mg
    225,00€
    100mg
    371,00€
  • MPEP

    CAS:
    MPEP is a selective mGlu5 receptor antagonist with IC50 of 36 nM, exhibits no appreciable activity at mGlu1b/2/3/4a/7b/8a/6 receptors.
    Fórmula:C14H11N
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:193.24

    Ref: TM-T6598

    10mg
    46,00€
    25mg
    80,00€
    50mg
    130,00€
    100mg
    200,00€
    200mg
    295,00€
    500mg
    497,00€
  • YM90K

    CAS:
    YM90K (6-(1H-imidazol-1-yl)-7-nitro-2,3(1H,4H)-) hydrochloride is an antagonist of AMPA receptor.
    Fórmula:C11H8ClN5O4
    Pureza:98.23%
    Forma y color:Solid
    Peso molecular:309.66

    Ref: TM-T8435

    1mg
    73,00€
    5mg
    160,00€
    1mL*10mM (DMSO)
    170,00€
    10mg
    245,00€
    25mg
    404,00€
    50mg
    567,00€
    100mg
    767,00€
    200mg
    1.018,00€
  • VU0364770

    CAS:
    VU0364770 (VU 0364770)(EC50=1.1 μM), a positive allosteric modulator(PAM) of mGlu4, shows insignificant activity at 68 other receptors, including other mGlu
    Fórmula:C12H9ClN2O
    Pureza:99.65% - >99.99%
    Forma y color:Solid
    Peso molecular:232.67

    Ref: TM-T6727

    1mL*10mM (DMSO)
    33,00€
    10mg
    34,00€
    25mg
    44,00€
    50mg
    73,00€
    100mg
    103,00€
    500mg
    245,00€
  • 3-MATIDA

    CAS:
    3-MATIDA is an effective mGluR-1 antagonist (IC50: 6.3 μM, rat mGluR-1a).
    Fórmula:C8H9NO4S
    Pureza:99.75% - 99.96%
    Forma y color:Solid
    Peso molecular:215.23

    Ref: TM-T3486

    2mg
    34,00€
    5mg
    49,00€
    1mL*10mM (DMSO)
    49,00€
    10mg
    79,00€
    25mg
    145,00€
    50mg
    227,00€
    100mg
    339,00€
    200mg
    482,00€
  • VU 0357121

    CAS:
    VU0357121, a positive allosteric modulator of mGlu5 (EC50: 33 nM), is inactive or very weakly antagonizing at other mGlu receptor subtypes.
    Fórmula:C17H17F2NO2
    Pureza:99% - >99.99%
    Forma y color:Solid
    Peso molecular:305.32

    Ref: TM-T6725

    2mg
    39,00€
    5mg
    56,00€
    1mL*10mM (DMSO)
    56,00€
    10mg
    90,00€
    25mg
    172,00€
    50mg
    266,00€
    100mg
    416,00€
  • HBT1

    CAS:
    HBT1 is an AMPA receptor potentiator that induces production of brain-derived neurotrophic factor (BDNF) and exhibits little agonistic effect in primary neurons
    Fórmula:C16H17F3N4O2S
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:386.39

    Ref: TM-T8779

    10mg
    46,00€
    1mL*10mM (DMSO)
    46,00€
    25mg
    82,00€
    50mg
    110,00€
    100mg
    178,00€
    200mg
    266,00€