
GluR
Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.
Se han encontrado 265 productos de "GluR"
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CX614
CAS:CX614 is a positive allosteric modulator of the AMPA receptor concerning AMPA.Fórmula:C13H13NO4Pureza:97.37%Forma y color:SolidPeso molecular:247.25Ref: TM-T19698
5mg52,00€1mL*10mM (DMSO)55,00€10mg78,00€25mg119,00€50mg172,00€100mg259,00€200mg388,00€MTEP
CAS:MTEP: potent, selective mGluR5 antagonist; IC50=5 nM, Ki=16 nM; may have antidepressant/anxiolytic effects; useful in Parkinson's research.Fórmula:C11H8N2SForma y color:SolidPeso molecular:200.26JNJ-42153605
CAS:JNJ-42153605 is a mGlu2 receptor positive allosteric modulator (EC50: 17 nM).
Fórmula:C22H23F3N4Pureza:97.25% - 98.57%Forma y color:SolidPeso molecular:400.44LY-404187
CAS:LY404187 is a positive allosteric modulator of AMPA receptorsFórmula:C19H22N2O2SPureza:99.34%Forma y color:SolidPeso molecular:342.46Ref: TM-T7706
2mg35,00€5mg52,00€1mL*10mM (DMSO)58,00€10mg90,00€25mg164,00€50mg239,00€100mg339,00€200mg472,00€CX717
CAS:CX 717 is a positive allosteric modulator of AMPA receptor which has an antidepressant-like effect.Fórmula:C11H11N3O3Pureza:99.81%Forma y color:SoildPeso molecular:233.23(S)-4CPG
CAS:(S)-4CPG ((S)-4-Carboxyphenylglycine) is a competitive mGlu1 receptor antagonist that attenuates nociceptive hypersensitivity and nociceptive abnormalities associated with sciatic nerve constriction injuries in rats, and may be used in the study of neurological disorders.Fórmula:C9H9NO4Pureza:99.96%Forma y color:SolidPeso molecular:195.17VU0477886
CAS:VU0477886: Potent mGlu4 PAM, effective in preclinical Parkinson's model HIC.Fórmula:C20H13ClN4O3Pureza:98%Forma y color:SolidPeso molecular:392.80IEM 1754 2HBr
CAS:IEM 1754 2HBr (IEM 1754 dihydrobromide) is a selective AMPA/kainate receptor blockers for GluR1 and GluR3 with IC50 of 6 μM.Fórmula:C16H30N2·2HBrPureza:99.04% - 99.72%Forma y color:SolidPeso molecular:412.25LY456066
CAS:LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.Fórmula:C19H23N3OSPureza:98%Forma y color:SolidPeso molecular:341.47Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Fórmula:C13H10N2OPureza:98.66%Forma y color:SolidPeso molecular:210.23Z-Cyclopentyl-AP4
CAS:Group III mGlu receptor agonistFórmula:C6H12NO5PPureza:98%Forma y color:SolidPeso molecular:209.14Talaglumetad hydrochloride
CAS:Talaglumetad hydrochloride, a prodrug of Eglumegad, targets mGluR2/3 to treat psychiatric disorders.Fórmula:C11H17ClN2O5Forma y color:SolidPeso molecular:292.72DFMTI
CAS:DFMTI can completely block the rmGlu1 L757V glutamate response.Fórmula:C20H18F2N4OForma y color:SolidPeso molecular:368.38LY392098
CAS:LY392098 (AMPA receptor modulator-3) is an allosteric modulator of AMPA receptor with EC50 of 4.4 μM and can be used in studies about mammalian nervous system.Fórmula:C18H22FNO2SPureza:99.86%Forma y color:SolidPeso molecular:335.44Ref: TM-T27951
1mg39,00€5mg93,00€1mL*10mM (DMSO)96,00€10mg133,00€25mg215,00€50mg306,00€100mg414,00€200mg573,00€RO5488608
CAS:RO5488608 is a new type of high-efficiency mGlu2/3 NAM.Fórmula:C23H17F3N2O4SForma y color:SolidPeso molecular:474.45GRN-529
CAS:GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.Fórmula:C22H15F2N3O2Pureza:98%Forma y color:SolidPeso molecular:391.37A 841720
CAS:Potent, selective mGlu1 antagonist A-841720; IC50: 10 nM; 34x selectivity vs mGlu5; analgesic potential.Fórmula:C17H21N5OSForma y color:SolidPeso molecular:343.45NPEC-caged-LY379268
CAS:NPEC-caged-LY379268 is a type II mGluR agonist [1].Fórmula:C16H16N2O9Forma y color:SolidPeso molecular:380.31MAP4
CAS:metabotropic glutamate receptor modulatorFórmula:C5H12NO5PPureza:98%Forma y color:White SolidPeso molecular:197.13mGluR2 modulator 1
CAS:Potent mGluR2 modulator 1 crosses blood-brain barrier, EC50: 0.03 μM, useful for psychiatric research.Fórmula:C21H20F3N3O3Forma y color:SolidPeso molecular:419.4
