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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Se han encontrado 265 productos de "GluR"

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productos por página.
  • VU0418506

    CAS:
    VU0418506 is a positive allosteric modulator (PAM) of the metabotropic glutamate receptor 4 (mGlu4).
    Fórmula:C12H8ClFN4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:262.67

    Ref: TM-T29134

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • ACDPP hydrochloride

    CAS:
    mGlu5 receptor antagonist
    Fórmula:C12H13ClN6O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:292.72

    Ref: TM-T22543

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • Ro 64-5229

    CAS:
    mGlu2 antagonist
    Fórmula:C17H19Cl2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:352.26

    Ref: TM-T23247

    10mg
    888,00€
    50mg
    3.574,00€
  • DL-AP4 Sodium salt

    CAS:
    Broad spectrum EAA ligand
    Fórmula:C4H10NNaO5P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:206.09

    Ref: TM-T22731

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU6001966

    CAS:
    VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.
    Fórmula:C17H15FN4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:326.33

    Ref: TM-T29142

    5mg
    982,00€
  • VU6010572

    CAS:
    VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.
    Fórmula:C20H18FNO3
    Forma y color:Solid
    Peso molecular:339.36

    Ref: TM-T61070

    25mg
    1.927,00€
    50mg
    2.507,00€
    100mg
    3.168,00€
  • VU0463841

    CAS:
    VU0463841 is a mGlu5 negative allosteric modulators.
    Fórmula:C13H8ClFN4O
    Forma y color:Solid
    Peso molecular:290.68

    Ref: TM-T29138

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU 0360172 hydrochloride

    CAS:
    positive allosteric modulator of mGlu5 receptors
    Fórmula:C18H16ClFN2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:330.78

    Ref: TM-T23510

    5mg
    251,00€
    10mg
    470,00€
    25mg
    1.108,00€
  • ACPT-II

    CAS:
    metabotropic receptor antagonist
    Fórmula:C8H11NO6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:217.18

    Ref: TM-T22550

    10mg
    697,00€
    50mg
    2.673,00€
  • mGluR2 modulator 4

    CAS:
    Compound 47 is a potent mGluR2 enhancer with an EC50 of 0.8 μM, potentially useful for antipsychotic research.
    Fórmula:C18H18BrN3
    Forma y color:Solid
    Peso molecular:356.26

    Ref: TM-T61277

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU0400195

    CAS:
    VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).
    Fórmula:C21H16ClN3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:393.82

    Ref: TM-T29129

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU0404251

    CAS:
    VU0404251 is a positive allosteric modulator of mGlu5.
    Fórmula:C19H23FN2O2
    Forma y color:Solid
    Peso molecular:330.4

    Ref: TM-T29130

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU0364289

    CAS:
    VU0364289 is a positive allosteric modulator of mGlu5.
    Fórmula:C20H21N3O2
    Forma y color:Solid
    Peso molecular:335.4

    Ref: TM-T29128

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • VU0361747

    CAS:
    VU0361747 is a positive allosteric modulators (PAM) of metabotropic glutamate receptor subtype 5 (mGlu5).
    Fórmula:C19H17FN2O2
    Forma y color:Solid
    Peso molecular:324.35

    Ref: TM-T29127

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • MSOP

    CAS:
    MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).
    Fórmula:C4H10NO6P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:199.1

    Ref: TM-T12118

    5mg
    470,00€
    25mg
    1.728,00€
  • LY487379 hydrochloride

    CAS:
    Positive allosteric modulator of mGlu2 receptors
    Fórmula:C21H20ClF3N2O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:488.91

    Ref: TM-T22955

    10mg
    747,00€
  • AZ12216052

    CAS:
    AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to study obesity and metabolic disorders.
    Fórmula:C19H22BrNOS
    Pureza:99.29%
    Forma y color:Solid
    Peso molecular:392.35

    Ref: TM-T26701

    1mg
    34,00€
    2mg
    49,00€
    5mg
    77,00€
    10mg
    111,00€
    25mg
    187,00€
    50mg
    279,00€
    100mg
    396,00€
    200mg
    560,00€
  • CFMMC

    CAS:

    CFMMC is an allosteric mGluR1 antagonist agent.

    Fórmula:C22H28FNO4
    Forma y color:Solid
    Peso molecular:389.46

    Ref: TM-T25227

    25mg
    1.444,00€
    50mg
    1.882,00€
    100mg
    2.375,00€
  • YM 230888

    CAS:
    Selective mGlu1 antagonist
    Fórmula:C19H28N4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:360.52

    Ref: TM-T23545

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€
  • LY2607540

    CAS:
    LY2607540 is a metabotropic glutamate 2 potentiator with potential anxiolytic/antidepressant properties (EC(50) = 23 and 13 nM, respectively).
    Fórmula:C24H24F3N3O4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:475.46

    Ref: TM-T27935

    25mg
    1.369,00€
    50mg
    1.783,00€
    100mg
    2.250,00€