
GluR
Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.
Se han encontrado 265 productos de "GluR"
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LY456066
CAS:LY456066 is a mGluR1 receptor-selective, negative allosteric modulator.Fórmula:C19H23N3OSPureza:98%Forma y color:SolidPeso molecular:341.47Z-Cyclopentyl-AP4
CAS:Group III mGlu receptor agonistFórmula:C6H12NO5PPureza:98%Forma y color:SolidPeso molecular:209.14DFMTI
CAS:DFMTI can completely block the rmGlu1 L757V glutamate response.Fórmula:C20H18F2N4OForma y color:SolidPeso molecular:368.38LY382884
CAS:LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.Fórmula:C18H23NO4Pureza:98.32% - 98.71%Forma y color:SolidPeso molecular:317.38GRN-529
CAS:GRN-529 is a selective negative allosteric modulator of the mGluR5 receptor.Fórmula:C22H15F2N3O2Pureza:98%Forma y color:SolidPeso molecular:391.37MAP4
CAS:metabotropic glutamate receptor modulatorFórmula:C5H12NO5PPureza:98%Forma y color:White SolidPeso molecular:197.13mGlu4 receptor agonist 1
CAS:Compound 62, an mGlu4 agonist, has a 308 nM EC50 with anxiolytic and antipsychotic effects.Fórmula:C21H15ClN4O2Forma y color:SolidPeso molecular:390.82ADX71743
CAS:ADX71743 is a potent and selective negative allosteric modulator of metabotropic glutamate receptor 7.Fórmula:C17H19NO2Pureza:99.27%Forma y color:SolidPeso molecular:269.34VU 0360223
CAS:VU 0360223 is a negative allosteric modulator of mGlu5.Fórmula:C15H9FN2SPureza:98%Forma y color:SolidPeso molecular:268.31L-AP4 monohydrate
CAS:L-AP4 (L-APB) is a group III mGluR agonist with EC50s: 0.13μM (mGlu4), 0.29μM (mGlu8), 1.0μM (mGlu6), 249μM (mGlu7).Fórmula:C4H12NO6PForma y color:SolidPeso molecular:201.115VU0366248
CAS:VU0366248 is a mGlu5 negative allosteric modulator.Fórmula:C14H7ClF2N2OPureza:98%Forma y color:SolidPeso molecular:292.673,3'-Difluorobenzaldazine
CAS:allosteric potentiator of mGlu5Fórmula:C14H10F2N2Pureza:98%Forma y color:SolidPeso molecular:244.24TC-N 22A
CAS:TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.Fórmula:C14H13N5SPureza:99.95%Forma y color:SolidPeso molecular:283.35(RS)-MCPG disodium salt
CAS:group I/group II metabotropic glutamate receptor antagonistFórmula:C10H11NNaO4Pureza:98%Forma y color:SolidPeso molecular:232.19CPPHA
CAS:CPPHA, a positive allosteric modulator of glutamate receptors mGluR5 and mGluR1, is commonly used in development for central nervous system diseases.
Fórmula:C22H15ClN2O4Pureza:98.07%Forma y color:SolidPeso molecular:406.82ML289
CAS:ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, >15-fold selectivity over mGlu2, and inactive against mGlu5.Fórmula:C22H23NO3Pureza:99.54%Forma y color:SolidPeso molecular:349.42Ref: TM-T23000
5mg48,00€1mL*10mM (DMSO)49,00€10mg75,00€25mg138,00€50mg212,00€100mg320,00€200mg445,00€LYPLAL1-IN-1
CAS:LYPLAL1-IN-1 is a selective covalent small-molecule inhibitor of Lysophospholipase-like 1 (IC50: 0.006 μM). LYPLAL1-IN-1 also enhances glucose production.Fórmula:C29H29N7O4Pureza:98%Forma y color:SolidPeso molecular:539.59Methoxy-PEPy
CAS:Methoxy-PEPy is a potent and selective mGlu5 receptor inhibitor with an IC50 value of 1 nM.Fórmula:C13H10N2OPureza:98.66%Forma y color:SolidPeso molecular:210.23(1R,2S)-VU0155041
CAS:(1R,2S)-VU0155041 is the cis regioisomer of VU0155041 and a partial agonist of mGluR4.Fórmula:C14H15Cl2NO3Pureza:98.85%Forma y color:SolidPeso molecular:316.18VU 0469650
CAS:VU 0469650 is a potent and selective negative allosteric modulator of mGluR1 (IC50 = 99 nM).Fórmula:C22H28N4OPureza:98.03%Forma y color:SolidPeso molecular:364.48Ref: TM-T29118
1mg42,00€5mg79,00€1mL*10mM (DMSO)90,00€10mg108,00€25mg210,00€50mg313,00€100mg464,00€200mg640,00€
