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GluR

GluR

Inhibidores del Receptor de Glutamato son compuestos que bloquean la actividad de los receptores de glutamato, los principales receptores de neurotransmisores excitatorios en el cerebro. Estos receptores desempeñan un papel crucial en la transmisión sináptica, la plasticidad, el aprendizaje y la memoria. La desregulación de la señalización de glutamato está asociada con varios trastornos neurológicos, como la epilepsia, el accidente cerebrovascular y las enfermedades neurodegenerativas. Los inhibidores de los receptores de glutamato son esenciales para investigar los mecanismos de la excitotoxicidad y desarrollar estrategias neuroprotectoras. En CymitQuimica, ofrecemos una gama de inhibidores de receptores de glutamato para apoyar su investigación en la función sináptica, la neuroprotección y los trastornos cognitivos.

Se han encontrado 255 productos de "GluR"

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  • LSP1-2111

    CAS:
    <p>LSP1-2111 is a mGlu4 receptor subtype agonist.</p>
    Fórmula:C12H17N2O9P
    Forma y color:Solid
    Peso molecular:364.25
  • Lu-AF11205

    CAS:
    <p>Lu-AF11205 is a potent positive allosteric modulator (PAM) of mGlu5 receptor.</p>
    Fórmula:C17H16N2OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:296.39
  • (RS)-4-Carboxyphenylglycine

    CAS:
    <p>(RS)-4-Carboxyphenylglycine is a racemic mixture. (S)-4-Carboxyphenylglycine is a selective mGlu1α receptor antagonist.</p>
    Fórmula:C9H9NO4
    Pureza:99.04% - >99.99%
    Forma y color:Solid
    Peso molecular:195.17
  • (R)-4-Carboxyphenylglycine

    CAS:
    <p>(R)-4-Carboxyphenylglycine is a NMDA receptor antagonist.</p>
    Fórmula:C9H9NO4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:195.17
  • VU0652835

    CAS:
    <p>VU0652835 is a negative allosteric modulator of metabotropic glutamate receptor subtype 5 (mGlu5) (IC50: 81 nM).</p>
    Fórmula:C16H19N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:333.41
  • JNJ-55511118

    CAS:
    <p>JNJ-55511118 is a TARP γ8 allosteric modulator with anticonvulsant activity, which can be used in research on chronic operant alcohol self-administration.</p>
    Fórmula:C14H8ClF3N2O2
    Forma y color:Solid
    Peso molecular:328.67
  • DCB

    CAS:
    <p>DCB is an mGluR5 allosteric ligand that blocks mGluR modulation, countering DMeOB and DFB effects.</p>
    Fórmula:C14H10Cl2N2
    Pureza:99.12% - 99.9%
    Forma y color:Solid
    Peso molecular:277.15
  • ML337

    CAS:
    <p>ML337 is a negative allosteric modulator of mGlu3 with an IC50 of 593 nM.</p>
    Fórmula:C21H20FNO3
    Pureza:99.83%
    Forma y color:Solid
    Peso molecular:353.39
  • LY382884

    CAS:
    <p>LY382884 is a selective and potent GluR5 kainate receptor antagonist with anxiolytic activity.LY382884 blocks blockade of mossy fibre LTP induction.</p>
    Fórmula:C18H23NO4
    Pureza:98.32% - 98.71%
    Forma y color:Solid
    Peso molecular:317.38
  • TC-N 22A

    CAS:
    <p>TC-N 22A is a strong, selective, oral active mGlu4 forward allosteric regulator (PAM) that can cross the blood-brain barrier.</p>
    Fórmula:C14H13N5S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:283.35
  • CPPHA

    CAS:
    <p>CPPHA, a positive allosteric modulator of glutamate receptors mGluR5 and mGluR1, is commonly used in development for central nervous system diseases.</p>
    Fórmula:C22H15ClN2O4
    Pureza:98.07%
    Forma y color:Solid
    Peso molecular:406.82
  • ML289

    CAS:
    <p>ML289 is a potent CNS-penetrant mGlu3 modulator with IC50 of 0.66 μM, &gt;15-fold selectivity over mGlu2, and inactive against mGlu5.</p>
    Fórmula:C22H23NO3
    Pureza:99.54%
    Forma y color:Solid
    Peso molecular:349.42
  • Foliglurax

    CAS:
    <p>Foliglurax is a highly selective brain-penetrant metabotropic glutamate receptor 4 positive allosteric modulator (mGluR4 PAM) (EC50: 79 nM).</p>
    Fórmula:C23H23N3O3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:421.51
  • VU6001376

    CAS:
    <p>VU6001376 is an effective and selective positive allosteric modulator of the metabotropic glutamate receptor 4 (EC50: 50.1 nM).</p>
    Fórmula:C18H14F2N6OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:400.41
  • Ro 67-4853

    CAS:
    <p>Ro 67-4853 is a positive allosteric modulator of mGluR1, selectively enhancing the response to the agonist (S)-3,5-dihydroxy-phenylglycine (DHPG).</p>
    Fórmula:C19H19NO4
    Pureza:98.57%
    Forma y color:Solid
    Peso molecular:325.36
  • VU0155041 sodium

    CAS:
    <p>VU0155041 sodium is a positive allosteric modulator of mGluR4 that promotes extinction in male rats.</p>
    Fórmula:C14H14Cl2NNaO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:338.16
  • HexylHIBO

    CAS:
    <p>HexylHIBO is a type I mGluR antagonist that inhibits mGlu1a and mGlu5a, with Kb values of 140 and 110 μM, respectively.HexylHIBO decreases sEPSC in rats.</p>
    Fórmula:C12H20N2O4
    Pureza:99.55%
    Forma y color:Solid
    Peso molecular:256.3
  • (S)-MCPG

    CAS:
    <p>(S)-MCPG is the active isomer of (RS)-MCPG, non-selective group I/group II metabotropic glutamate receptor antagonist.</p>
    Fórmula:C10H11NO4
    Pureza:98.72%
    Forma y color:Solid
    Peso molecular:209.20
  • DMeOB

    CAS:
    <p>DMeOB (3,3'-Dimethoxybenzaldazine) is a negative regulator with mGluR5 agonist activity and is used in the study of neurological disorders.</p>
    Fórmula:C16H16N2O2
    Pureza:98.34%
    Forma y color:Solid
    Peso molecular:268.31
  • A-794282

    CAS:
    <p>A-794282 is a selective antagonist of mGluR1.</p>
    Fórmula:C19H18N4OS
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:350.44