AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Pentolinium Tartrate
CAS:<p>Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.</p>Fórmula:C15H32N2·2C4H5O6Pureza:98%Forma y color:SolidPeso molecular:538.6AF-DX 384 free base
CAS:<p>AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.</p>Fórmula:C27H38N6O2Pureza:98%Forma y color:SolidPeso molecular:478.63Pozanicline
CAS:<p>Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.</p>Fórmula:C11H16N2OPureza:98%Forma y color:SolidPeso molecular:192.26CB-6673567
CAS:<p>CB-6673567 is a selective inhibitor of adenylyl cyclase.</p>Fórmula:C19H14N4O3Forma y color:SolidPeso molecular:346.34NGX-267
CAS:<p>NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.</p>Fórmula:C10H18N2OSForma y color:SolidPeso molecular:214.33Dac 5945
CAS:<p>DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.</p>Fórmula:C19H30ClN3OPureza:98%Forma y color:SolidPeso molecular:351.91Hexocyclium metilsulfate
CAS:<p>Hexocyclium metilsulfate has anti-gastric secretory effects in humans.</p>Fórmula:C21H36N2O5SPureza:98%Forma y color:SolidPeso molecular:428.59GS 283
CAS:<p>GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.</p>Fórmula:C17H17NO3Forma y color:SolidPeso molecular:283.32(R)-VU 6008667
CAS:<p>(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).</p>Fórmula:C24H17ClF2N2O2Forma y color:SolidPeso molecular:438.85Anisodine hydrobromide
CAS:<p>Anisodine hydrobromide is an inhibitor of adenosine kinase.</p>Fórmula:C17H22BrNO5Forma y color:White Crystals Or Crystalline PowderPeso molecular:400.27Btm 1042
CAS:<p>Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.</p>Fórmula:C21H26ClN3OSForma y color:SolidPeso molecular:403.97Hyoscyamine hydrobromide
CAS:<p>Hyoscyamine hydrobromide is an agent of anticholinergic.</p>Fórmula:C17H24BrNO3Pureza:98%Forma y color:SolidPeso molecular:370.28Sazetidine A dihydrochloride
CAS:<p>α4β2 nicotinic acetylcholine receptor ligand</p>Fórmula:C15H21ClN2O2Pureza:98%Forma y color:SolidPeso molecular:296.79FR 121196
CAS:<p>FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.</p>Fórmula:C12H16FN3O3SForma y color:SolidPeso molecular:301.34Prifuroline
CAS:<p>Prifuroline is an agent of antiarrhythmic.</p>Fórmula:C14H16N2OPureza:98%Forma y color:SolidPeso molecular:228.29Epibatidine 2HCl
CAS:<p>Epibatidine 2HCl is a potent nicotinic agonist.</p>Fórmula:C11H15Cl3N2Pureza:98%Forma y color:SolidPeso molecular:281.61Flutropium Bromide
CAS:<p>Flutropium Bromide is a competitive antagonist of acetylcholine. It is used to treat asthma and chronic obstructive pulmonary.</p>Fórmula:C24H29BrFNO3Pureza:98%Forma y color:SolidPeso molecular:478.39Vesamicol
CAS:Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.Fórmula:C17H25NOPureza:98%Forma y color:SolidPeso molecular:259.39Siltenzepine
CAS:<p>Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.</p>Fórmula:C19H20ClN3O4Pureza:98%Forma y color:SolidPeso molecular:389.83L 858051
CAS:<p>L 858051 activates adenylate cyclase. It also inhibits glucose transport in rat adipocytes.</p>Fórmula:C29H48N2O7Forma y color:SolidPeso molecular:536.7
