AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 623 productos para "AChR".
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Btm 1042
CAS:Btm 1042 is an antispasmodic drug. It has been found to depress twitch responses in the ileum of guinea pigs.Fórmula:C21H26ClN3OSForma y color:SolidPeso molecular:403.97Hyoscyamine hydrobromide
CAS:Hyoscyamine hydrobromide is an agent of anticholinergic.Fórmula:C17H24BrNO3Pureza:98%Forma y color:SolidPeso molecular:370.28Sazetidine A dihydrochloride
CAS:α4β2 nicotinic acetylcholine receptor ligandFórmula:C15H21ClN2O2Pureza:98%Forma y color:SolidPeso molecular:296.79FR 121196
CAS:FR 121196, a potential antidementia drug, ameliorates the impaired memory of rat in the Morris water maze.Fórmula:C12H16FN3O3SForma y color:SolidPeso molecular:301.34Prifuroline
CAS:Prifuroline is an agent of antiarrhythmic.Fórmula:C14H16N2OPureza:98%Forma y color:SolidPeso molecular:228.29Epibatidine 2HCl
CAS:Epibatidine 2HCl is a potent nicotinic agonist.Fórmula:C11H15Cl3N2Pureza:98%Forma y color:SolidPeso molecular:281.61Flutropium Bromide
CAS:Flutropium Bromide is a competitive antagonist of acetylcholine. It is used to treat asthma and chronic obstructive pulmonary.Fórmula:C24H29BrFNO3Pureza:98%Forma y color:SolidPeso molecular:478.39Vesamicol
CAS:Vesamicol is an experimental drug. It acting presynaptically by inhibiting acetylcholine uptake into synaptic vesicles and reducing its release.Fórmula:C17H25NOPureza:98%Forma y color:SolidPeso molecular:259.3865Siltenzepine
CAS:Siltenzepine is an agent of anti-acid agent,and used in the treatment of peptic ulcers.Fórmula:C19H20ClN3O4Pureza:98%Forma y color:SolidPeso molecular:389.83L 858051
CAS:L 858051 activates adenylate cyclase. It also inhibits glucose transport in rat adipocytes.Fórmula:C29H48N2O7Forma y color:SolidPeso molecular:536.7LY593093
CAS:LY593093 is a selective partial orthosteric agonist of M1 muscarinic acetylcholine receptor.Fórmula:C32H30FN3O2Pureza:98%Forma y color:SolidPeso molecular:507.6DBO-83
CAS:DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.Fórmula:C10H15Cl3N4Pureza:98%Forma y color:SolidPeso molecular:297.61ADX-10061
CAS:ADX-10061 is a dopamine D1 receptor antagonist.Fórmula:C19H20N2O4Forma y color:SolidPeso molecular:340.37JN403
CAS:JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.Fórmula:C16H21FN2O2Forma y color:SolidPeso molecular:292.35Tebanicline tosylate
CAS:Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.Fórmula:C16H19ClN2O4SPureza:98%Forma y color:SolidPeso molecular:370.85Terodiline hydrochloride
CAS:Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),Fórmula:C20H28ClNPureza:98%Forma y color:SolidPeso molecular:317.9YM-46303
CAS:YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia inFórmula:C20H23ClN2O2Pureza:>99.99%Forma y color:Yellow SolidPeso molecular:358.86CHF5407
CAS:CHF5407（SVT-47060） is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect onFórmula:C27H25BrF4N2O3SPureza:99.54% - >99.99%Forma y color:White SolidPeso molecular:613.46KL8604166
CAS:KL8604166 (UCB-11056) is a potential puzzle compound.UCB-11056 amplifies the formation of inducible cyclic AMP in rat brain tissue.Fórmula:C12H21N5O2Pureza:99.95%Forma y color:White SolidPeso molecular:267.33PF-06767832
CAS:PF-06767832: selective M1 PAM (EC50=60 nM), no M2-M5 activity, good CNS penetration, but has GI and cardiovascular risks.Fórmula:C22H23N3O3SForma y color:SolidPeso molecular:409.5
