AChR
Los inhibidores del receptor de acetilcolina (AChR) son compuestos que bloquean la actividad de los receptores de acetilcolina, que son críticos para la neurotransmisión en los sistemas nerviosos central y periférico. Los AChRs juegan un papel vital en la contracción muscular, la memoria y las funciones cognitivas. Los inhibidores de los AChRs se utilizan para estudiar afecciones como la miastenia gravis, la enfermedad de Alzheimer y otros trastornos neurológicos. Al modular la actividad de los AChRs, estos inhibidores pueden ayudar a desentrañar las complejidades de la señalización colinérgica en el cerebro. En CymitQuimica, ofrecemos una gama de inhibidores de AChR para apoyar su investigación en neurociencia, farmacología y enfermedades neurodegenerativas.
Se han encontrado 575 productos de "AChR"
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DBO-83
CAS:<p>DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.</p>Fórmula:C10H15Cl3N4Pureza:98%Forma y color:SolidPeso molecular:297.61ADX-10061
CAS:<p>ADX-10061 is a dopamine D1 receptor antagonist.</p>Fórmula:C19H20N2O4Forma y color:SolidPeso molecular:340.37JN403
CAS:<p>JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.</p>Fórmula:C16H21FN2O2Forma y color:SolidPeso molecular:292.35Tebanicline tosylate
CAS:<p>Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.</p>Fórmula:C16H19ClN2O4SPureza:98%Forma y color:SolidPeso molecular:370.85Terodiline hydrochloride
CAS:<p>Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),</p>Fórmula:C20H28ClNPureza:98%Forma y color:SolidPeso molecular:317.9YM-46303
CAS:<p>YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia in</p>Fórmula:C20H23ClN2O2Pureza:>99.99%Forma y color:SolidPeso molecular:358.86CHF5407
CAS:<p>CHF5407（SVT-47060） is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on</p>Fórmula:C27H25BrF4N2O3SPureza:>99.99%Forma y color:SolidPeso molecular:613.46YM-58790
CAS:<p>YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.</p>Fórmula:C27H31N3O2Pureza:98.59%Forma y color:SoildPeso molecular:429.55Metixene hydrochloride
CAS:<p>Metixene hydrochloride is an anticholinergic antiparkinsonian agent.</p>Fórmula:C20H24ClNSPureza:98%Forma y color:SolidPeso molecular:345.93PQCA
CAS:<p>PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.</p>Fórmula:C22H20N4O3Pureza:99.88%Forma y color:SolidPeso molecular:388.42Penehyclidine hydrochloride
CAS:<p>Penehyclidine hydrochloride: M1/M3 antagonist, activates NF-κB, anti-inflammatory, anticholinergic.</p>Fórmula:C20H30ClNO2Pureza:99.79%Forma y color:SolidPeso molecular:351.91PD-102807
CAS:<p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>Fórmula:C23H24N2O4Pureza:98.90%Forma y color:SolidPeso molecular:392.45S 24795
CAS:<p>S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.</p>Fórmula:C14H13BrINOPureza:99.934%Forma y color:SolidPeso molecular:418.07S16961
CAS:<p>S16961 (S169611) is an agonist of nicotinic receptor.</p>Fórmula:C41H71NO6Pureza:99.69%Forma y color:SolidPeso molecular:674.01Afacifenacin
CAS:<p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>Fórmula:C27H26F3N3O2Pureza:99.83%Forma y color:SolidPeso molecular:481.51UP202-56
CAS:<p>UP202-56 is an adenosinergic agonist and is an adenosine analog.</p>Fórmula:C33H37N7O4Pureza:98%Forma y color:SolidPeso molecular:595.69CB-7921220
CAS:<p>CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.</p>Fórmula:C14H12N2O2Pureza:99.59%Forma y color:SolidPeso molecular:240.26Cimetropium Bromide
CAS:<p>Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.</p>Fórmula:C21H28BrNO4Forma y color:SolidPeso molecular:438.36GP531
CAS:<p>GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.</p>Fórmula:C16H21N5O4Forma y color:SolidPeso molecular:347.37GAT107
CAS:<p>GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.</p>Fórmula:C18H17BrN2O2SPureza:99.33%Forma y color:SolidPeso molecular:405.31
