Serina proteasa
Los inhibidores de serina proteasa son compuestos que inhiben las serina proteasas, un grupo de enzimas caracterizadas por un residuo de serina en su sitio activo. Estas proteasas están involucradas en numerosos procesos fisiológicos, incluyendo la digestión, la respuesta inmunitaria, la coagulación sanguínea y la inflamación. Los inhibidores de serina proteasa son fundamentales para estudiar enfermedades en las que estas enzimas están desreguladas, como enfermedades cardiovasculares, cáncer y condiciones inflamatorias. En CymitQuimica, ofrecemos inhibidores de serina proteasa para apoyar su investigación en enzimología, mecanismos de enfermedades e intervenciones terapéuticas.
Se han encontrado 85 productos para "Serina proteasa".
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TAO Kinase inhibitor 2
CAS:TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.Fórmula:C25H24N2O3Pureza:98.58%Forma y color:SolidPeso molecular:400.4697Chlorobenzothiazolinone
CAS:Chlorobenzothiazolinone blocks human chymase at 90 μM, assessed by fluorescence using a specific peptide substrate after 1 hr.Fórmula:C7H4ClNOSPureza:99.42% - 99.77%Forma y color:SolidPeso molecular:185.631BAY-85-8501
CAS:BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)Fórmula:C22H17F3N4O3SPureza:99.16%Forma y color:SolidPeso molecular:474.456Tilpisertib fosmecarbil TFA
CAS:Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.Fórmula:C37H37ClF3N8O9PForma y color:SolidPeso molecular:861.16Chymotrypsinogen
CAS:Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .Forma y color:SolidLonodelestat TFA
Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.Fórmula:C73H112F3N15O21Forma y color:SolidPeso molecular:1592.75Roseltide rT1
CAS:Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.Fórmula:C110H177N31O31S6Forma y color:SolidPeso molecular:2622.16KKI-5
CAS:KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.Fórmula:C35H55N11O9Pureza:98%Forma y color:SolidPeso molecular:773.88α 1 Antichymotrypsin, Human Plasma
CAS:Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.Forma y color:SolidSafflower oil (from Carthamus tinctorius seed)
CAS:Safflower oil (from Carthamus tinctorius seed) contains unsaturated fatty acids, tocopherols and phenolic compounds, which has antioxidant and lipid metabolism regulating activities, can scavenge free radicals and inhibit collagenase and elastase activities, and is often used in skin aging, atherosclerosis and functional oil-related research.CDD-3290
CDD-3290 serves as a functional therapeutic tool specifically designed to enable the precise detection and inhibition of the proteolytic activity of PSA which plays a pivotal role in the progression of prostate cancer during strictly monitored laboratory observation periods and molecular investigations to evaluate the pharmacological potential of targeted kallikrein inhibition in specialized preclinical research environments.Fórmula:C17H14N6O2Pureza:99.06% - 99.13%Forma y color:White SolidPeso molecular:334.33Kallikrein 5-IN-2 TFA
Kallikrein5-IN-2 TFA is the trifluoroacetate salt form of Kallikrein5-IN-2. It acts as a selective inhibitor of kallikrein5 (KLK5), with a pIC50 value of 7.1. Kallikrein5-IN-2 TFA exhibits no phototoxicity at 100 μg/mL and is non-irritating. The compound remains stable in non-oxidative conditions within a pH range of 4 to 8. Kallikrein5-IN-2 shows potential for improving Netherton syndrome.Fórmula:C25H23F3N6O3Forma y color:SolidPeso molecular:512.17837hCAXII-IN-10
hCAXII-IN-10 (Compound 18b) acts as a dual inhibitor of human carbonic anhydrase isoenzyme XII (hCAXII) and cathepsin B, with a Ki value of 2.2 nM. It inhibits the function of hCAXII in creating a pH microenvironment conducive to tumor growth, showing promise for use in cancer research.Forma y color:Odour SolidSuc-AAP-Abu-pNA
CAS:Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,Fórmula:C25H34N6O9Forma y color:SolidPeso molecular:562.57Tiprelestat
CAS:Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.Fórmula:C254H416N72O75S10Forma y color:SolidPeso molecular:5999.09Z-APF-CMK
CAS:Z-APF-CMK is a selective inhibitor of the calcium (Ca2+)-regulated nuclear scaffold protease (CRNSP), as reported in reference [1].Fórmula:C26H30ClN3O5Forma y color:SolidPeso molecular:499.99SFTI-1
CAS:SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.Fórmula:C67H104N18O18S2Forma y color:SolidPeso molecular:1513.78Protease Inhibitor Library
A unique collection of xnum protease and proteasome inhibitors for research in chemical genomics, and drug screening;Forma y color:Odour SolidMeOSuc-AAPA-CMK
MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].Fórmula:C20H31ClN4O8Forma y color:SolidPeso molecular:490.94Dansyl-Glu-Gly-Arg-Chloromethylketone
CAS:Dansyl-Glu-Gly-Arg-Chloromethylketone is a protease inhibitor that specifically impedes serine/threonine proteases and has been shown to inhibit activatedFórmula:C26H36ClN7O7SForma y color:SolidPeso molecular:626.12
