Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 358 productos de "Receptor de histamina"
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Betazole
CAS:<p>Betazole, an oral H2 receptor agonist, stimulates gastric acid and raises bile duct pressure, used for gastric secretory testing.</p>Fórmula:C5H9N3Forma y color:SolidPeso molecular:111.15Betazole dihydrochloride
CAS:<p>Betazole dihydrochloride (Betazole hydrochloride) is an agonist of H2 receptor.</p>Fórmula:C5H11Cl2N3Pureza:99.12%Forma y color:SolidPeso molecular:184.067Mequitazine
CAS:<p>Mequitazine (Virginan) is an effective, nonsedative and long-acting histamine H1 antagonist.</p>Fórmula:C20H22N2SPureza:99.98%Forma y color:SolidPeso molecular:322.47Ciproxifan maleate
CAS:<p>Ciproxifan maleate (FUB 359)(FUB-359 maleate) is a highly potent and selective histamin H3-receptor antagonist with IC50 of 9.2 nM, with low apparent affinity</p>Fórmula:C20H22N2O6Pureza:99.39%Forma y color:SolidPeso molecular:386.4Epinastine hydrochloride
CAS:<p>Epinastine hydrochloride (WAL-801CL HCl) is an antihistamine and mast cell stabilizer that is used in eye drops to treat allergic conjunctivitis.</p>Fórmula:C16H15N3·HClPureza:99.26% - 99.62%Forma y color:White SolidPeso molecular:285.77Mecamylamine hydrochloride
CAS:<p>Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.</p>Fórmula:C11H22ClNPureza:99.76% - >99.99%Forma y color:White SolidPeso molecular:203.75JNJ-7777120
CAS:<p>JNJ-7777120 is the first potent and selective non-imidazole histamine H4 receptor antagonist, exhibits >1000-fold selectivity over the other histamin receptors.</p>Fórmula:C14H16ClN3OPureza:99.83% - 99.96%Forma y color:SolidPeso molecular:277.75Chlorcyclizine
CAS:<p>CHLORCYCLIZINE is a histamine H1 antagonist and a potent hepatitis C virus (HCV) entry inhibitor.</p>Fórmula:C18H21ClN2Pureza:98.75%Forma y color:SolidPeso molecular:300.83Chlorprothixene
CAS:<p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>Fórmula:C18H18ClNSPureza:98.77% - 99.756%Forma y color:Pale Yellow Crystals SolidPeso molecular:315.86VUF10460
CAS:<p>VUF10460 is a non-imidazole histamine H4 receptor agonist.</p>Fórmula:C15H19N5Pureza:99.44% - 99.57%Forma y color:SolidPeso molecular:269.34Dimaprit dihydrochloride
CAS:<p>Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.</p>Fórmula:C6H15N3S·2HClPureza:99.79%Forma y color:SolidPeso molecular:234.19Talastine HCl
CAS:<p>Talastine is an antihistamine drug.</p>Fórmula:C19H22ClN3OPureza:98%Forma y color:SolidPeso molecular:343.86C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:<p>C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.</p>Fórmula:C93H157N27O28S3Pureza:>99.99%Forma y color:SolidPeso molecular:2197.6Tiaramide hydrochloride
CAS:<p>Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.</p>Fórmula:C15H19Cl2N3O3SPureza:98.48%Forma y color:SolidPeso molecular:392.3Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Fórmula:C29H34O6Pureza:≥98%Forma y color:LiquidPeso molecular:478.58cicloprofen
CAS:<p>cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.</p>Fórmula:C16H14O2Pureza:98.15%Forma y color:SolidPeso molecular:238.2812Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Forma y color:SolidPeso molecular:233.182-Pyridylethylamine dihydrochloride
CAS:<p>2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.</p>Fórmula:C7H12Cl2N2Pureza:99.42%Forma y color:SolidPeso molecular:195.09Decloxizine
CAS:<p>Decloxizine is a H1 receptor antagonist</p>Fórmula:C21H28N2O2Pureza:99.53%Forma y color:White Or Similar To White PowderPeso molecular:340.46Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86Clemizole hydrochloride
CAS:<p>Clemizole hydrochloride blocks H1 histamine receptors and inhibits HCV replication and NS4B RNA binding.</p>Fórmula:C19H21Cl2N3Pureza:>99.99%Forma y color:SolidPeso molecular:362.3Antazoline
CAS:<p>Antazoline has antihistamine and anticholinergic effects.It used to treat a variety of arrhythmias.</p>Fórmula:C17H19N3Pureza:≥95%Forma y color:White Crystalline Powder SolidPeso molecular:265.35Psoralenoside
CAS:<p>Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.</p>Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Betahistine EP Impurity C
CAS:<p>Betahistine EP Impurity C (NSC19005) is structurally related to Betahistine. Betahistine EP Impurity C is a dimer of Betahistine.</p>Fórmula:C15H19N3Pureza:≥95%Forma y color:SolidPeso molecular:241.33Betahistine
CAS:<p>Betahistine treats vertigo and balance issues in Ménière's disease; it's a histamine analog and H1 receptor agonist.</p>Fórmula:C8H12N2Pureza:99.87% - 99.87%Forma y color:Yellowish Liquid Liquid LiquidPeso molecular:136.19Buclizine dihydrochloride
CAS:<p>Buclizine dihydrochloride (Buclina) is the hydrochloride salt form of buclizine, a piperazine histamine H1 receptor antagonist with primarily antiemetic and</p>Fórmula:C28H33ClN2·2HClPureza:98.05%Forma y color:Off-White PowderPeso molecular:505.95S 38093
CAS:<p>S 38093 is a brain-penetrant antagonist of the H3 receptor (Ki: 8.8/1.44/1.2 μM, for rat/mouse/human).</p>Fórmula:C17H24N2O2Pureza:99.95%Forma y color:SolidPeso molecular:288.38Dioxopromethazine
CAS:<p>Dioxopromethazine (Dioxoprothazine) is a drug for the treatment of a cough and expectoration. It also can be used in local anesthesia.</p>Fórmula:C17H20N2O2SPureza:98%Forma y color:SolidPeso molecular:316.42Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Fórmula:C14H20F6N4O7Pureza:98.18%Forma y color:SolidPeso molecular:470.32Decloxizine dihydrochloride
CAS:<p>Decloxizine dihydrochloride (UCB 1402 dihydrochloride) is a histamine 1 receptor antagonist.</p>Fórmula:C21H28N2O2·2ClHPureza:99.73%Forma y color:SolidPeso molecular:413.39Histamine Phosphate
CAS:<p>Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.</p>Fórmula:C5H9N·2H3O4PPureza:>99.99%Forma y color:White Crystal PowderPeso molecular:307.14Alginic acid
CAS:<p>Alginic acid, a polysaccharide from brown seaweed, has anti-anaphylactic and anti-inflammatory properties and is used in food industry.</p>Fórmula:C14H22O13Pureza:≥98%Forma y color:SolidPeso molecular:398.317Betahistine dihydrochloride
CAS:<p>Betahistine dihydrochloride (Betahistine 2HCl) is a histamine analog and H1 receptor agonist that serves as a vasodilator.</p>Fórmula:C8H14Cl2N2Pureza:99.34% - 99.88%Forma y color:White To Light Yellow Crystalline PowderPeso molecular:209.12Thonzylamine
CAS:<p>Thonzylamine is an antihistamine/anticholinergic, combined with Clofedanol or Phenylephrine for cold, hay fever, or allergy relief.</p>Fórmula:C16H22N4OPureza:99.45%Forma y color:SolidPeso molecular:286.37Alimemazine hemitartrate
CAS:<p>Alimemazine hemitartrate (Trimeprazine hemitartrate) is aphenothiazine derivative that is used as an antipruritic.</p>Fórmula:C18H22N2SC4H6O6Pureza:98.16% - 99.69%Forma y color:SolidPeso molecular:448.53JNJ-5207852
CAS:<p>JNJ-5207852 is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptor.</p>Fórmula:C20H32N2OPureza:97.19%Forma y color:SolidPeso molecular:316.48LML134
CAS:<p>LML134 (LML-134) is an inverse agonist of Histamine 3 receptor (H3R)(hH3R cAMP and hH3R bdg with Kis of 0.3 nM and 12 nM).</p>Fórmula:C19H29N5O3Pureza:99.36%Forma y color:SolidPeso molecular:375.47S 38093 HCl
CAS:<p>S 38093 is a novel brain-penetrant antagonist/inverse agonist of H3 receptors.</p>Fórmula:C17H25ClN2O2Pureza:97.91%Forma y color:SolidPeso molecular:324.85Hydroxyzine dihydrochloride
CAS:<p>Hydroxyzine dihydrochloride treats allergies, pruritus, anxiety; causes drowsiness; also an antiemetic and sedative.</p>Fórmula:C21H27ClN2O2·2HClPureza:99.46% - 99.79%Forma y color:Oil PowderPeso molecular:447.83OXOMEMAZINE
CAS:<p>Oxomemazine: a phenothiazine antihistamine H1-blocker with strong antimuscarinic and selective M1 antagonist properties, used in cough research.</p>Fórmula:C18H22N2O2SPureza:99.58%Forma y color:SolidPeso molecular:330.44Ranitidine
CAS:<p>Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion (H2 receptors).</p>Fórmula:C13H22N4O3SPureza:99.52%Forma y color:Solid SolidPeso molecular:314.40Bepotastine
CAS:<p>Bepotastine (Bepotastine free base) free base is a histamine 1 (H1) receptor antagonis.</p>Fórmula:C21H25ClN2O3Pureza:99.75%Forma y color:SolidPeso molecular:388.89Latrepirdine dihydrochloride
CAS:<p>Latrepirdine dihydrochloride (Dimebolin dihydrochloride) is an orally active, and neuroactive antagonist of multiple drug targets.</p>Fórmula:C21H25N3·2HClPureza:98.45%Forma y color:SolidPeso molecular:392.37Levocetirizine Dihydrochloride
CAS:<p>Levocetirizine Dihydrochloride is a third-gen antihistamine targeting H1-receptors, treating allergies and urticaria.</p>Fórmula:C21H27Cl3N2O3Pureza:99.89%Forma y color:White Or Off-White Crystalline PowderPeso molecular:461.81Methaphenilene hydrochloride
CAS:<p>Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.</p>Fórmula:C15H21ClN2SPureza:99.84%Forma y color:SolidPeso molecular:296.86Ciproxifan
CAS:<p>Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).</p>Fórmula:C16H18N2O2Pureza:98.00%Forma y color:SolidPeso molecular:270.33Amthamine
CAS:<p>Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.</p>Fórmula:C6H11N3SForma y color:SoildPeso molecular:157.24Roxatidine acetate
CAS:<p>Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.</p>Fórmula:C19H28N2O4Pureza:98%Forma y color:White Or Off-White PowderPeso molecular:348.44Lodoxamide tromethamine
CAS:<p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>Fórmula:C19H28ClN5O12Pureza:98.8%Forma y color:SolidPeso molecular:553.91GT 2016
CAS:<p>GT 2016 is a H3 receptor antagonist.</p>Fórmula:C19H31N3OPureza:98%Forma y color:SolidPeso molecular:317.47
