
Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 381 productos de "Receptor de histamina"
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A-304121
CAS:A-304121 is a histamine H(3) receptor.Fórmula:C20H29N3O3Forma y color:SolidPeso molecular:359.46(R)-Mequitazine
CAS:<p>(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.</p>Fórmula:C20H22N2SForma y color:SolidPeso molecular:322.47ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Fórmula:C22H22N2OPureza:99.94%Forma y color:SolidPeso molecular:330.42Zolantidine dimaleate
CAS:H2 receptor antagonistFórmula:C26H31N3O5SPureza:98%Forma y color:SolidPeso molecular:497.61Aminopotentidine
CAS:H2 antagonistFórmula:C26H35N7O2Pureza:98%Forma y color:SolidPeso molecular:477.6Alimemazine
CAS:Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.Fórmula:C18H22N2SPureza:98%Forma y color:Crystals SolidPeso molecular:298.45JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFórmula:C13H15ClN4OForma y color:SolidPeso molecular:278.74Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Fórmula:C8H10N6SPureza:98%Forma y color:SolidPeso molecular:222.27Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Fórmula:C13H22N6Pureza:99.84%Forma y color:SolidPeso molecular:262.35VUF 8328
CAS:VUF 8328 is an agonist of histamine H(3) receptor.Fórmula:C7H12N4SPureza:98%Forma y color:SolidPeso molecular:184.26FR-A 19
CAS:FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.Fórmula:C25H34Cl3F2N5Forma y color:SolidPeso molecular:548.93S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFórmula:C6H11NO2SPureza:98%Forma y color:SolidPeso molecular:161.22UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Fórmula:C17H22N6SForma y color:SolidPeso molecular:342.46Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Fórmula:C14H23N7SPureza:98%Forma y color:SolidPeso molecular:321.44Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Fórmula:C20H22N2Pureza:98%Forma y color:SolidPeso molecular:290.4JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Fórmula:C17H19ClN4O5Pureza:99.37%Forma y color:SolidPeso molecular:394.81Setastine
CAS:Setastine, a highly selective H1 receptor antagonist, acts as a non-sedative antihistamine.Fórmula:C22H28ClNOForma y color:SolidPeso molecular:357.92JNJ-28610244
CAS:JNJ-28610244 is a specific agonist of the H4 receptor. It acts by blocking Mac-1-dependent activation of p38 MAPK.Fórmula:C16H21N3OPureza:98%Forma y color:SolidPeso molecular:271.36GT 2016
CAS:GT 2016 is a H3 receptor antagonist.Fórmula:C19H31N3OPureza:98%Forma y color:SolidPeso molecular:317.47Bavisant dihydrochloride
CAS:Bavisant (JNJ-310010740) is an oral, selective H3 receptor antagonist enhancing wakefulness and cognition.Fórmula:C19H29Cl2N3O2Pureza:98%Forma y color:SolidPeso molecular:402.36
