Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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Adriforant
CAS:Adriforant (PF-3893787,ZPL-3893797) is a competitive histamine receptor 4 h4 antagonist that antagonizes histamine-induced phosphorylation of ERK, inflammation.Fórmula:C13H22N6Pureza:99.84%Forma y color:SolidPeso molecular:262.35FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Fórmula:C22H30N2O4SPureza:98%Forma y color:SolidPeso molecular:418.55ReN-1869 hydrochloride
CAS:ReN 1869 hydrochloride is a novel, selective antagonist of histamine H1 receptor.Fórmula:C24H28ClNO2Pureza:98%Forma y color:SolidPeso molecular:397.94H4R antagonist 1
CAS:H4R antagonist 1: selective histamine H4R inhibitor, IC50 27 nM, no affinity for H1R, H2R, H3R.Fórmula:C11H11BrN8Forma y color:SolidPeso molecular:335.16(±)-Tazifylline
CAS:(±)-Tazifylline is a selective and long-acting antagonist of histamine H1 receptor.Fórmula:C23H32N6O3SPureza:99.54%Forma y color:SolidPeso molecular:472.6Azelastine
CAS:<p>Azelastine (Azelastinum) is a phthalazine derivative, and is an histamine antagonist and mast cell stabilizer.</p>Fórmula:C22H24ClN3OPureza:99.35%Forma y color:White Crystal PowderPeso molecular:381.90Zaltidine
CAS:Zaltidine is an antagonist of H2-receptor, and has the antisecretory action.Fórmula:C8H10N6SPureza:98%Forma y color:SolidPeso molecular:222.27JNJ-10191584
CAS:JNJ-10191584, a potent and selective antagonist at the histamine H4 receptor, has antiinflammatory and analgesic effects in animal studies of acute inflammationFórmula:C13H15ClN4OForma y color:SolidPeso molecular:278.74Alimemazine
CAS:Alimemazine, an antipruritic and HA-receptor antagonist, also partially activates H1R and other GPCRs.Fórmula:C18H22N2SPureza:98%Forma y color:Crystals SolidPeso molecular:298.45Aminopotentidine
CAS:H2 antagonistFórmula:C26H35N7O2Pureza:98%Forma y color:SolidPeso molecular:477.6Zolantidine dimaleate
CAS:H2 receptor antagonistFórmula:C26H31N3O5SPureza:98%Forma y color:SolidPeso molecular:497.61BMY-25271
CAS:BMY-25271 is an antagonist of histamine H2 receptor.Fórmula:C12H19N5O2S2Pureza:98%Forma y color:SolidPeso molecular:329.44ABT-239
CAS:ABT-239 is a novel, highly efficacious antagonist belonging to the non-imidazole class of histamine H3 receptor (H3R) antagonists.Fórmula:C22H22N2OPureza:99.94%Forma y color:SolidPeso molecular:330.42(R)-Mequitazine
CAS:(R)-Mequitazine, a muscarinic acetylcholine receptor (M-AChRs) antagonist, is used potentially for the treatment of asthma.Fórmula:C20H22N2SForma y color:SolidPeso molecular:322.47A-304121
CAS:A-304121 is a histamine H(3) receptor.Fórmula:C20H29N3O3Forma y color:SolidPeso molecular:359.46OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Fórmula:C19H30ClN3SForma y color:SolidPeso molecular:367.98JNJ 10181457 dihydrochloride
CAS:JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.Fórmula:C20H28N2OPureza:98%Forma y color:SolidPeso molecular:312.45Mianserin
CAS:Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family.Fórmula:C18H20N2Pureza:99.85%Forma y color:SolidPeso molecular:264.36Wy 49051
CAS:Wy 49051 is an orally active antagonist of H1 receptor(IC50 of 44 nM).Fórmula:C28H33N5O3Pureza:99.89%Forma y color:SolidPeso molecular:487.59ROS 234
CAS:ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.Fórmula:C13H15N5Forma y color:SolidPeso molecular:241.29
