Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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Bamirastine
CAS:Bamirastine inhibits ligand binding to recombinant human histamine H1 receptor (rhH1R) with an IC50 value of 17.3 nM.Bamirastine has an inhibitory effect onFórmula:C31H37N5O3Pureza:96.68%Forma y color:SolidPeso molecular:527.66CP-66948
CAS:CP-66948 is a potent histamine H2 receptor antagonist with inhibitory effect on gastric acid secretion and can be used to protect gastric and intestinal mucosa.Fórmula:C13H20N6SPureza:99.14%Forma y color:SolidPeso molecular:292.4PF-03654764
CAS:PF-03654764, an oral H3 receptor blocker, Ki: human 1.2 nM, rat 7.9 nM, used with Fexofenadine for allergic rhinitis.Fórmula:C20H28F2N2OPureza:>99.99%Forma y color:SolidPeso molecular:350.45Lavoltidine
CAS:Lavoltidine (Loxtidine) is potent and selective H2 receptor antagonist, oral and irreversible,inhibits gastric acid secretion, gastroesophageal reflux disease.Fórmula:C19H29N5O2Pureza:98.30% - 98.36%Forma y color:SolidPeso molecular:359.47H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Fórmula:C19H24ClN3O3Pureza:98%Forma y color:SolidPeso molecular:377.86Propiomazine HCl
CAS:Propiomazine HCl is an analgesia adjunct.Fórmula:C20H25ClN2OSForma y color:SolidPeso molecular:376.94Vapitadine dihydrochloride
CAS:Vapitadine dihydrochloride(R-129160 2HCl) is a novel, potent, selective and non-sedating compound with inhibitory effects on histamine H1.Fórmula:C17H22Cl2N4OPureza:98.28% - 99.30%Forma y color:SolidPeso molecular:369.29JNJ 10191584 maleate
CAS:JNJ 10191584 maleate (VUF6002 maleate) is an orally active and selective antagonist of H4 receptor (Ki = 26 nM).Fórmula:C17H19ClN4O5Pureza:99.37%Forma y color:SolidPeso molecular:394.81Azatadine
CAS:Azatadine is histamine and cholinergic inhibitor (IC50: 6.5 nM and 10 nM, respectively).Fórmula:C20H22N2Pureza:98%Forma y color:SolidPeso molecular:290.4Impromidine
CAS:Impromidine is a highly potent and specific agonist of the histamine H2 receptor.Fórmula:C14H23N7SPureza:98%Forma y color:SolidPeso molecular:321.44VUF14862
CAS:VUF14862 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Fórmula:C26H32N4O2Forma y color:SolidPeso molecular:432.56Sch 44643
CAS:Sch 44643 is an antagonist of platelet activating factor with oral activity.Fórmula:C25H22ClN3O2Forma y color:SolidPeso molecular:431.91UR-PI376
CAS:UR-PI376 is a selective histamine H4 receptor agonist with low H1/H2 activity and moderate H3 affinity.Fórmula:C17H22N6SForma y color:SolidPeso molecular:342.46Brl 22321
CAS:Brl 22321 is a mast cell stabilizer.Fórmula:C12H9N3O2Forma y color:SolidPeso molecular:227.22BL 6341A
CAS:BL 6341A is related to Tumor data and H2-antagonists or anti-histaminsFórmula:C9H14N8OS3Forma y color:SolidPeso molecular:346.46(R)-Azelastine
CAS:(R)-Azelastine, an antihistamine, reduces H1R, M1R, M3R levels and inhibits HNEpC growth.Fórmula:C22H24ClN3OForma y color:SolidPeso molecular:381.9Aceprometazine
CAS:Aceprometazine (1664CB) is an antipsychotic which is orally active. Aceprometazine can be used in psychiatric disorders research, for example, depression [1].Fórmula:C19H22N2OSForma y color:SolidPeso molecular:326.46Noberastine maleate
CAS:Noberastine maleate, a fast-acting furan-derived H1 antagonist, peaks at 4 hours with minimal CNS effects and maximal efficacy at 30 mg/day.Fórmula:C25H29N5O9Forma y color:SolidPeso molecular:543.53ROS 234 dioxalate
CAS:ROS 234 dioxalate is a potent antagonist of H3(pKB of 9.46 for Guinea-pig ileum H3-receptor)Fórmula:C17H19N5O8Pureza:98%Forma y color:SolidPeso molecular:421.37Fenspiride-d5
CAS:Fenspiride-d5: internal standard for GC/LC-MS quantification, H1 antagonist, NSAID, anti-inflammatory, selective PDE4,5,3 inhibitor.Fórmula:C15H15D5N2O2Forma y color:SolidPeso molecular:265.36
