Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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GSK-239512
CAS:GSK-239512 is an antagonist of H3 receptor and can be used in studies about the treatment of cognitive dysfunction in neurodegenerative disorders.Fórmula:C23H27N3O2Pureza:99.62% - 99.74%Forma y color:SolidPeso molecular:377.48S-1-Propenyl-L-cysteine
CAS:S-1-Propenyl-L-cysteine, a stereoisomer of S-allyl-l-cysteine, exhibits immunomodulatory effects and has been shown to decrease blood pressure in hypertensiveFórmula:C6H11NO2SPureza:98%Forma y color:SolidPeso molecular:161.22Dacemazine
CAS:Dacemazine is used to treat depression.Fórmula:C16H16N2OSForma y color:SolidPeso molecular:284.38VUF14738
CAS:VUF14738 is a robust and fatigue-resistant photoswitchable GPCR antagonist.Fórmula:C25H32N4O2Forma y color:SolidPeso molecular:420.55Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Fórmula:C19H17NO7Pureza:95% - 97.34%Forma y color:SolidPeso molecular:371.34Dothiepin HCl
CAS:Dothiepin HCl: TCA, SNRI, with antihistamine, antiadrenergic, anticholinergic, and sodium block properties.Fórmula:C19H22ClNSForma y color:SolidPeso molecular:331.9FR-A 19
CAS:FR-A 19: Histamine H2 agonist, nanomolar inhibition of basophil histamine release; potent anti-allergic.Fórmula:C25H34Cl3F2N5Forma y color:SolidPeso molecular:548.93KY 234
CAS:KY 234 is a thromboxane synthetase antagonist.Fórmula:C33H35N5O2Forma y color:SolidPeso molecular:533.676(S)-Azelastine
CAS:(S)-Azelastine is an antihistamine reducing receptors H1R, M1R, M3R, and inhibiting HNEpC cell growth.Fórmula:C22H24ClN3OForma y color:SolidPeso molecular:381.9VUF 8328
CAS:VUF 8328 is an agonist of histamine H(3) receptor.Fórmula:C7H12N4SPureza:98%Forma y color:SolidPeso molecular:184.26ReN-1869
CAS:ReN-1869 is a novel selective histamine H(1) receptor antagonist with anti-neurogenic pain and anti-inflammatory activity for the study of neurological diseasesFórmula:C24H27NO2Pureza:99.83% - 99.98%Forma y color:SolidPeso molecular:361.48Immethridine dihydrobromide
CAS:Immethridine dihydrobromide is a histamine H3 receptor agonist.Fórmula:C9H11Br2N3Pureza:97.61% - 98.14%Forma y color:SolidPeso molecular:321.01Proxyfan
CAS:Proxyfan is a high-affinity protean antagonist/agonist of H3 receptors from full agonist to full inverse agonist, depending on given tissue or brain region.Fórmula:C13H16N2OPureza:99.68%Forma y color:SolidPeso molecular:216.28DF-1111301
CAS:DF-1111301 is a novel anti-allergic compound with anti-histamine H1 and anti-PAF activity.Fórmula:C15H25Cl2N3OPureza:99.17%Forma y color:SolidPeso molecular:334.29Noberastine
CAS:Noberastine (R 64947) is a novel histamine H1 antagonist with potent and specific peripheral antihistamine activity.Fórmula:C17H21N5OPureza:99.72% - >99.99%Forma y color:SolidPeso molecular:311.38KP136
CAS:KP136 is an orally effective antiallergic compound (IC50: 76.1 μg/mL for histamine release and 63 ug/mL for degranulation).Fórmula:C16H18N4O3Pureza:98.3% - 98.61%Forma y color:SolidPeso molecular:314.34JZP-361
CAS:JZP-361: selective MAGL inhibitor (IC50 = 46 nM); weaker on FAAH, hABHD6; anti-histamine; for asthma research.Fórmula:C22H20ClN5OPureza:99.82%Forma y color:SolidPeso molecular:405.88Pitolisant
CAS:Pitolisant is a potent and selective nonimidazole inverse agonist that acts on the recombinant human histamine H3 receptor with Ki of 0.16 nM.Fórmula:C17H26ClNOPureza:99.84%Forma y color:SolidPeso molecular:295.85Ref: TM-T60636
5mg48,00€10mg70,00€25mg120,00€50mg188,00€100mg311,00€500mg747,00€1mL*10mM (DMSO)52,00€KSK94
CAS:KSK94 is an H3 receptor antagonist that inhibits sigma-2 receptors , with a Ki value of 75.2 nM, and can be used to study injurious pain.Fórmula:C25H26N4OPureza:99.60%Forma y color:SolidPeso molecular:398.5Impromidine hydrochloride
CAS:<p>Impromidine hydrochloride is a very potent and specific histamine H2 receptor agonist for conducting cardiovascular studies.</p>Fórmula:C14H26Cl3N7SPureza:99.82%Forma y color:SolidPeso molecular:430.83
