Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 385 productos de "Receptor de histamina"
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Zotepine
CAS:Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86SCH-37370
CAS:SCH-37370 is an effective and orally active dual antagonist of platelet-activating factor and histamine.Fórmula:C21H21ClN2OPureza:99.07%Forma y color:SolidPeso molecular:352.86Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Fórmula:C19H23ClN2Forma y color:SolidPeso molecular:314.852H4 Receptor antagonist 1
CAS:H4 Receptor antagonist 1 is a potent and selective histamine H4 receptor inverse agonist, with an IC50 of 19 nM.Fórmula:C16H17ClN4OPureza:98.81%Forma y color:SolidPeso molecular:316.79Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFórmula:C21H28N2O2Pureza:99.53%Forma y color:White Or Similar To White PowderPeso molecular:340.46Psoralenoside
CAS:Psoralenoside: a compound from Psoralea fruit; has estrogenic, osteoblastic, antitumor, and antibacterial properties.Fórmula:C17H18O9Pureza:99.03% - 99.49%Forma y color:SolidPeso molecular:366.32Bilastine
CAS:Bilastine (Bilaxten) is a novel new-generation antihistamine that is highly selective for the H1 histamine receptor, has a rapid onset and prolonged duration ofFórmula:C28H37N3O3Pureza:99.86% - >99.99%Forma y color:SolidPeso molecular:463.61Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Forma y color:SolidPeso molecular:233.18Ritanserin
CAS:Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.Fórmula:C27H25F2N3OSPureza:99.77% - 99.89%Forma y color:SolidPeso molecular:477.57cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Fórmula:C16H14O2Pureza:98.15%Forma y color:SolidPeso molecular:238.2812C-Type Natriuretic Peptide (CNP) (1-22), human
CAS:C-Type Natriuretic Peptide (CNP) (1-22), human is the 1-22 fragment of C-Type Natriuretic Peptide.Fórmula:C93H157N27O28S3Pureza:>99.99%Forma y color:SolidPeso molecular:2197.6Niaprazine
CAS:<p>Niaprazine is a histamine H1-receptor antagonist with marked sedative properties.</p>Fórmula:C20H25FN4OPureza:99.56%Forma y color:SolidPeso molecular:356.44Tiaramide hydrochloride
CAS:Tiaramide hydrochloride (FK-1160) is an anti-inflammatory that blocks mast cell mediators and relaxes smooth muscles.Fórmula:C15H19Cl2N3O3SPureza:98.48%Forma y color:SolidPeso molecular:392.3Irdabisant hydrochloride
CAS:Irdabisant (CEP-26401) is a selective H3R inverse agonist, BBB-penetrable, with cognition-enhancing effects.Fórmula:C18H24ClN3O2Forma y color:SolidPeso molecular:349.86Talastine HCl
CAS:Talastine is an antihistamine drug.Fórmula:C19H22ClN3OPureza:98%Forma y color:SolidPeso molecular:343.86Tribenoside
CAS:Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.Fórmula:C29H34O6Pureza:≥98%Forma y color:LiquidPeso molecular:478.58Clobenpropit 2HBr
CAS:Clobenpropit 2HBr is a histamine H3 receptor antagonist. It has neuroprotective effects via stimulation of GABA release in the brain.Fórmula:C14H17ClN4SForma y color:SolidPeso molecular:308.83Lodoxamide
CAS:<p>Lodoxamide (Lodoxamidum) is an antiallergic drug acting as a mast-cell stabilizer. It is effective in the treatment of asthma and allergic conjunctivitis.</p>Fórmula:C11H6ClN3O6Pureza:99.13% - 99.81%Forma y color:SolidPeso molecular:311.63Dimaprit dihydrochloride
CAS:Dimaprit dihydrochloride: selective H2 agonist, inhibits nNOS (IC50: 49 μM), boosts gastric acid.Fórmula:C6H15N3S·2HClPureza:99.79%Forma y color:SolidPeso molecular:234.19HTMT dimaleate
CAS:HTMT dimaleate (Histamine Trifluoromethyl Toluidide Dimaleate) is an H1 and H2 receptor agonist.Fórmula:C27H33F3N4O9Pureza:99.51%Forma y color:SolidPeso molecular:614.57
