Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 381 productos de "Receptor de histamina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Carcinine ditrifluoroacetate Acetate
<p>Carcinine ditrifluoroacetate Acetate (β-Alanylhistamine dihydrochloride) is an H3 receptor antagonist.</p>Fórmula:C14H20F6N4O7Pureza:98.18%Forma y color:SolidPeso molecular:470.32Histamine Phosphate
CAS:Histamine Phosphate (Histamine acid phosphate) acts directly on the blood vessels to dilate arteries and capillaries mediated by both H 1- and H 2-receptors.Fórmula:C5H9N·2H3O4PPureza:>99.99%Forma y color:White Crystal PowderPeso molecular:307.14Buclizine
CAS:Buclizine is an orally active antihistamine, antiallergic compound. buclizine is also a strong teratogen in rats and exhibits antitumour effects.Fórmula:C28H33ClN2Forma y color:SolidPeso molecular:433.03Desloratadine
CAS:Desloratadine (Sch34117) is a long-acting piperidine derivate with selective H1 antihistaminergic and non-sedating properties.Fórmula:C19H19ClN2Pureza:99.79% - >99.99%Forma y color:SolidPeso molecular:310.82Decloxizine
CAS:Decloxizine is a H1 receptor antagonistFórmula:C21H28N2O2Pureza:99.53%Forma y color:White Or Similar To White PowderPeso molecular:340.46Fexofenadine
CAS:Fexofenadine, a non-sedating antihistamine, treats allergies like hay fever and urticaria.Fórmula:C32H39NO4Pureza:99.35%Forma y color:White To Off-White SolidPeso molecular:501.66JNJ-5207852 dihydrochloride
CAS:JNJ-5207852 dihydrochloride is a novel, non-imidazole histamine H3 receptor antagonist, with high affinity at the rat (pKi=8.9) and human (pKi=9.24) H3 receptorFórmula:C20H34Cl2N2OPureza:99.51%Forma y color:SolidPeso molecular:389.4Bepotastine Besilate
CAS:Bepotastine Besilate (TAU 284) is a non-sedating and selective H1 receptor antagonist (pIC50: 5.7).Fórmula:C21H25ClN2O3·C6H6O3SPureza:99.83% - 99.9%Forma y color:Brown Viscous LiquidPeso molecular:547.062-Pyridylethylamine dihydrochloride
CAS:2-Pyridylethylamine dihydrochloride is a Histamine H1 receptor agonist.Fórmula:C7H12Cl2N2Pureza:99.42%Forma y color:SolidPeso molecular:195.09Zotepine
CAS:<p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>Fórmula:C18H18ClNOSPureza:99.78%Forma y color:SolidPeso molecular:331.86cicloprofen
CAS:cicloprofen is Cell division cycle 7-related protein kinase (human) inhibitor.Fórmula:C16H14O2Pureza:98.15%Forma y color:SolidPeso molecular:238.2812Acitazanolast
CAS:<p>Acitazanolast (WP-871) is an anti-allergic drug candidate.</p>Fórmula:C9H7N5O3Pureza:98.25%Forma y color:SolidPeso molecular:233.18BMY-25368
CAS:BMY-25368 is a long-acting antagonist of the H2-receptor.Fórmula:C19H25N3O3Forma y color:SolidPeso molecular:343.42Alcaftadine
CAS:<p>Alcaftadine (Lastacaft) is an H1 histamine receptor antagonist indicated for the prevention of itching associated with allergic conjunctivitis.</p>Fórmula:C19H21N3OPureza:98% - 98.65%Forma y color:SolidPeso molecular:307.39GSK189254A
CAS:<p>GSK189254A (GSK189254) is a potent and specific histamine H3 receptor antagonist (pKi values: 9.59-9.90 and 8.51-9.17 for human and rat H3).</p>Fórmula:C21H25N3O2Pureza:98.71% - 99.858%Forma y color:SolidPeso molecular:351.44Tribenoside
CAS:<p>Tribenoside (BG-356) is a vasoprotectant with mild anti-inflammatory, analgesic, and wound healing properties.</p>Fórmula:C29H34O6Pureza:≥98%Forma y color:LiquidPeso molecular:478.58Clemizole
CAS:<p>Clemizole is an H1 histamine receptor antagonist, can inhibit NS4B's RNA binding and hepatitis C virus (HCV) replication.</p>Fórmula:C19H20ClN3Pureza:98% - 99.65%Forma y color:SolidPeso molecular:325.84Mebhydrolin
CAS:<p>Mebhydrolin (Mebhydroline) is a specific histamine H1 receptor antagonist.</p>Fórmula:C19H20N2Pureza:99.3% - ≥98%Forma y color:SolidPeso molecular:276.38Triprolidine hydrochloride
CAS:Triprolidine hydrochloride anhydrous, a Histamine H1 antagonist, is used in asthma, allergic rhinitis, and urticaria.Fórmula:C19H23ClN2Forma y color:SolidPeso molecular:314.852Pitolisant hydrochloride
CAS:Pitolisant hydrochloride (Ciproxidine) is a potent and selective inverse agonist of the histamine H3 receptor(Ki : 0.16 nM).Fórmula:C17H27Cl2NOPureza:99.72% - 99.91%Forma y color:SolidPeso molecular:332.31
