Receptor de histamina
Los receptores de histamina son GPCR que median los efectos de la histamina, una amina biógena involucrada en las respuestas inmunitarias, la secreción de ácido gástrico y la neurotransmisión. Hay cuatro subtipos de receptores de histamina (H1, H2, H3 y H4), cada uno de los cuales desempeña roles distintos en las reacciones alérgicas, la función gástrica y la actividad del sistema nervioso central. Los antagonistas de los receptores de histamina se utilizan ampliamente en el tratamiento de alergias, úlceras pépticas y mareos por movimiento. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores de histamina de alta calidad para apoyar su investigación en inmunología, gastroenterología y neurofarmacología.
Se han encontrado 381 productos de "Receptor de histamina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Hydroxyzine-d8 DiHCl
CAS:Hydroxyzine-d8 DiHCl is a deuterated compound of Hydroxyzine DiHCl. Hydroxyzine DiHCl has a CAS number of 2192-20-3.Fórmula:C21H21D8Cl3N2O2Forma y color:SolidPeso molecular:455.88Methaphenilene hydrochloride
CAS:Methaphenilene hydrochloride is an H1 receptor antagonist with antihistaminic and anticholinergic activity, in allergic inflammation and autonomic research.Fórmula:C15H21ClN2SPureza:99.84%Forma y color:SolidPeso molecular:296.86Mianserin-d3
CAS:Mianserin-d3 is a deuterated compound of Mianserin. Mianserin has a CAS number of 24219-97-4. Mianserin, an H1 receptor reverse agonist, is a psychoactive compound in the tetracyclic antidepressant (TeCA) treatment family. Mianserin has antidepressant, antianxiety, antiemetic, hypotrophic, hypnotic and antihistamine effects, and can be used as a combination of norepinephrine and specific serotonin to treat depression.Fórmula:C18H17D3N2Forma y color:SolidPeso molecular:267.38Roxatidine acetate
CAS:Roxatidine acetate: anti-ulcer, blocks histamine, reduces acid. Safer at lower doses.Fórmula:C19H28N2O4Pureza:98%Forma y color:White Or Off-White PowderPeso molecular:348.44Amthamine
CAS:Compound AMTHAMINE DIHYDROBROMIDE is a useful organic compound for research related to life sciences.Fórmula:C6H11N3SForma y color:SoildPeso molecular:157.24Proxyfan Oxalate
CAS:Proxyfan Oxalate is a potent antagonist of the histamine H3 receptor (histamine H3 receptor), with Ki values of 2.9 nM for rats and 2.7 nM for humans. Its inhibitory effect on H3 receptors is over 1000 times stronger than its effect on other histamine receptors.Fórmula:C15H18N2O5Forma y color:SolidPeso molecular:306.31Ciproxifan
CAS:Ciproxifan (FUB-359) is a highly effective and specific histamin H3-receptor antagonist (IC50: 9.2 nM).Fórmula:C16H18N2O2Pureza:98.00%Forma y color:SolidPeso molecular:270.33Lodoxamide tromethamine
CAS:<p>Lodoxamide tromethamine is a mast cell stabilizer with anti-allergic properties and can be used in studies about the treatment of asthma and allergic</p>Fórmula:C19H28ClN5O12Pureza:98.8%Forma y color:SolidPeso molecular:553.91PF-03654746
CAS:<p>PF-03654746: selective H3 antagonist, boosts cognition in Alzheimer's, may treat allergic rhinitis.</p>Fórmula:C18H24F2N2OPureza:98.85% - 99.57%Forma y color:SolidPeso molecular:322.39A 987306
CAS:<p>A-987306: Potent, oral histamine H4 antagonist; Ki: 3.4 nM (rat), 5.8 nM (human); reduces inflammation in mouse peritonitis.</p>Fórmula:C18H25N5OForma y color:SolidPeso molecular:327.42FRG8701
CAS:FRG8701 is a new Histamine H2-receptor antagonist with an IC50 of ranging from 0.25 to 0.43 μM.Fórmula:C22H30N2O4SPureza:98%Forma y color:SolidPeso molecular:418.55Nedocromil
CAS:Nedocromil (FPL 59002) inhibits the action or formation of multiple mediators. Which including histamine, leukotriene C4 (LTC4), and prostaglandin D2 (PGD2).Fórmula:C19H17NO7Pureza:95% - 97.34%Forma y color:SolidPeso molecular:371.34H3R-IN-1 Hydrochloride
CAS:H3R-IN-1 Hydrochloride is an inverse agonist of histamine receptor 3( H3R ) .Fórmula:C19H24ClN3O3Pureza:98%Forma y color:SolidPeso molecular:377.86Carcinine
CAS:Carcinine ditrifluoroacetate is a H3 receptor antagonist.Fórmula:C8H14N4OPureza:98%Forma y color:SolidPeso molecular:182.22Setastine HCl
CAS:<p>Setastine HCl is a potent antagonist of histamine H1-receptor mediated responses.</p>Fórmula:C22H29Cl2NOForma y color:SolidPeso molecular:394.38Carbinoxamine
CAS:Carbinoxamine: antihistamine for hay fever, angioedema, rhinitis, mild urticaria, dermatographism, allergic conjunctivitis; an H1-antagonist.Fórmula:C16H19ClN2OPureza:98%Forma y color:LiquidPeso molecular:290.79AZD5213
CAS:AZD5213: selective human H3 receptor antagonist, pKi 9.3, for sleep/cognition research.Fórmula:C19H25N3O2Forma y color:SolidPeso molecular:327.42ROS 234
CAS:ROS 234 is a potent H3 antagonist with pKB 9.46 for Guinea-pig ileum and pKi 8.90 for Rat cortex; ED50 of 19.12 mg/kg in rats, but with limited central access.Fórmula:C13H15N5Forma y color:SolidPeso molecular:241.29JNJ 10181457 dihydrochloride
CAS:<p>JNJ 10181457 dihydrochloride is a Histamine H3 receptor antagonist.</p>Fórmula:C20H28N2OPureza:98%Forma y color:SolidPeso molecular:312.45OUP-186
CAS:OUP-186 is a selective H3 receptor antagonist that suppresses breast cancer cell growth with an IC50 of ~50 μM and induces apoptosis.Fórmula:C19H30ClN3SForma y color:SolidPeso molecular:367.98
