
Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
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Dynorphin B (1-13) acetate(83335-41-5 free base)
<p>Dynorphin B (1-13) acetate acts as an agonist on opioid κ-receptor.</p>Fórmula:C76H119N21O19Pureza:99.72%Forma y color:SolidPeso molecular:1630.89Bisacodyl
CAS:<p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>Fórmula:C22H19NO4Pureza:99.45% - 99.78%Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline PowderPeso molecular:361.39LY2795050
CAS:<p>LY2795050 is a novel specific κ-Opioid Receptor antagonist (IC50: 0.72 nM).</p>Fórmula:C23H22ClN3O2Pureza:97.77%Forma y color:SolidPeso molecular:407.89Alvimopan monohydrate
CAS:<p>Alvimopan monohydrate is a mu-opioid receptor antagonist that intended for the treatment of constipation in patients who take opiates for pain.</p>Fórmula:C25H34N2O5Pureza:98%Forma y color:SolidPeso molecular:442.55[Met5]-Enkephalin, amide TFA
<p>[Met5]-Enkephalin, amide TFA (5-Methionine-enkephalin amide (TFA)) is a δ opioid receptors agonist as well as putative ζ (zeta) opioid receptors.</p>Fórmula:C29H37F3N6O8SPureza:99.81%Forma y color:SolidPeso molecular:686.7GRT2932Q
CAS:<p>GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].</p>Fórmula:C25H26ClN3OForma y color:SolidPeso molecular:419.95LY2048978
CAS:<p>LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.</p>Fórmula:C19H24N2O2Pureza:98%Forma y color:SolidPeso molecular:312.41ML138
CAS:<p>ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.</p>Fórmula:C19H14Cl2N4OSForma y color:SolidPeso molecular:417.31SCH 221510
CAS:<p>SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.</p>Fórmula:C28H31NOPureza:99.54%Forma y color:SolidPeso molecular:397.55μ opioid receptor agonist 2
CAS:<p>μ opioid receptor agonist 2 (Compound H-3)is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.</p>Fórmula:C25H34N4OForma y color:SolidPeso molecular:406.56TIPP
CAS:<p>TIPP is an agent of delta opioid antagonist.</p>Fórmula:C37H38N4O6Pureza:98%Forma y color:SolidPeso molecular:634.72Opioid receptor modulator 1
CAS:<p>Opioid receptor modulator 1 is a modulator of opioid receptor.</p>Fórmula:C18H23NO2Pureza:98%Forma y color:SolidPeso molecular:285.38LY2444296
CAS:<p>LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).</p>Fórmula:C24H22F2N2O2Pureza:99.18%Forma y color:SolidPeso molecular:408.44BW 373U86
CAS:<p>BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [</p>Fórmula:C27H37N3O2Forma y color:SolidPeso molecular:435.6ML 190
CAS:<p>ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.</p>Fórmula:C27H32N6O3Pureza:99.88%Forma y color:SolidPeso molecular:488.58GSK1521498 free base (hydrochloride)
CAS:<p>GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H21ClF2N4Pureza:98%Forma y color:SolidPeso molecular:438.9ADL-5859 HCl
CAS:<p>ADL-5859 is a delta-opioid receptor agonist.</p>Fórmula:C24H28N2O3Pureza:98%Forma y color:SolidPeso molecular:392.49DIPPA hydrochloride
CAS:<p>κ receptor antagonist</p>Fórmula:C22H24Cl3N3OSPureza:98%Forma y color:SolidPeso molecular:484.87PF-4455242 HCl
CAS:<p>PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.</p>Fórmula:C21H29ClN2O2SPureza:99.59%Forma y color:SolidPeso molecular:408.99CP-866087
CAS:<p>CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.</p>Fórmula:C24H28N2O2Pureza:99.56% - >99.99%Forma y color:SoildPeso molecular:376.49
