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Receptor de opioides

Receptor de opioides

Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.

Se han encontrado 296 productos de "Receptor de opioides"

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  • ORL1 antagonist 1

    CAS:
    <p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>
    Fórmula:C20H22ClN5
    Pureza:98.92%
    Forma y color:Solid
    Peso molecular:367.88
  • ICI 154,129

    CAS:
    <p>Selective δ opioid antagonist</p>
    Fórmula:C34H46N4O6S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:638.82
  • JTC-801 free base

    CAS:
    <p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>
    Fórmula:C26H25N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:411.5
  • LY 164929

    CAS:
    <p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>
    Fórmula:C28H41N5O4
    Forma y color:Solid
    Peso molecular:511.66
  • SR8993

    CAS:
    <p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>
    Fórmula:C25H37FN4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:412.59
  • BMS-986124

    CAS:
    <p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>
    Fórmula:C16H15BrClNO3S2
    Forma y color:Solid
    Peso molecular:448.78
  • DDD028

    CAS:
    <p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>
    Fórmula:C20H20N2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:288.39
  • Viminol

    CAS:
    <p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>
    Fórmula:C21H31ClN2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:362.94
  • Ici 174865

    CAS:
    <p>Ici 174865 is a delta opioid receptor antagonist agent.</p>
    Fórmula:C38H53N5O7
    Forma y color:Solid
    Peso molecular:691.86
  • Endomorphin 1 acetate

    CAS:
    <p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>
    Fórmula:C36H42N6O7
    Forma y color:Solid
    Peso molecular:670.75
  • Axomadol

    CAS:
    <p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>
    Fórmula:C16H25NO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:279.37
  • LY 281217

    CAS:
    <p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>
    Fórmula:C32H42N4O6
    Pureza:98%
    Forma y color:Solid
    Peso molecular:578.7
  • Diallyl G

    CAS:
    <p>Diallyl G is a delta-opioid receptor antagonist agent.</p>
    Fórmula:C38H53N5O8
    Forma y color:Solid
    Peso molecular:707.86
  • Loperamide oxide

    CAS:
    <p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>
    Fórmula:C29H33ClN2O3
    Forma y color:Solid
    Peso molecular:493.04
  • CR-665 Acetate

    CAS:
    <p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>
    Fórmula:C38H53N9O6
    Forma y color:Solid
    Peso molecular:731.899
  • AZD7268

    CAS:
    <p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>
    Fórmula:C29H30N4O2S
    Forma y color:Solid
    Peso molecular:498.64
  • AT-076

    CAS:
    <p>AT-076: κ-opioid (Ki=1.14 nM) &amp; nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) &amp; δ-opioid (Ki=19.6 nM) competitive antagonist.</p>
    Fórmula:C26H35N3O3
    Forma y color:Solid
    Peso molecular:437.57
  • GSK1521498

    CAS:
    <p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>
    Fórmula:C24H23F2N4O4P
    Pureza:98%
    Forma y color:Solid
    Peso molecular:500.43
  • Dup 747

    CAS:
    <p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>
    Fórmula:C24H28Cl2N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:447.4
  • σ1 Receptor/μ Opioid receptor modulator 1

    CAS:
    <p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>
    Fórmula:C24H31FN2O2
    Forma y color:Solid
    Peso molecular:398.51