
Receptor de opioides
Los receptores opioides son un grupo de receptores acoplados a proteínas G que median los efectos de los opioides endógenos y exógenos. Estos receptores desempeñan un papel central en la modulación del dolor, la regulación del estado de ánimo y los comportamientos adictivos. Los agonistas y antagonistas de los receptores opioides se utilizan ampliamente en el manejo del dolor y el tratamiento de adicciones, así como en la investigación de trastornos neurológicos y psiquiátricos. En CymitQuimica, ofrecemos una selección integral de moduladores de receptores opioides de alta calidad para apoyar su investigación en neurobiología, manejo del dolor y terapia de adicciones.
Se han encontrado 296 productos de "Receptor de opioides"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
ORL1 antagonist 1
CAS:<p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>Fórmula:C20H22ClN5Pureza:98.92%Forma y color:SolidPeso molecular:367.88ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Fórmula:C34H46N4O6SPureza:98%Forma y color:SolidPeso molecular:638.82JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Fórmula:C26H25N3O2Pureza:98%Forma y color:SolidPeso molecular:411.5LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Fórmula:C28H41N5O4Forma y color:SolidPeso molecular:511.66SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Fórmula:C25H37FN4Pureza:98%Forma y color:SolidPeso molecular:412.59BMS-986124
CAS:<p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>Fórmula:C16H15BrClNO3S2Forma y color:SolidPeso molecular:448.78DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Fórmula:C20H20N2Pureza:98%Forma y color:SolidPeso molecular:288.39Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Fórmula:C21H31ClN2OPureza:98%Forma y color:SolidPeso molecular:362.94Ici 174865
CAS:<p>Ici 174865 is a delta opioid receptor antagonist agent.</p>Fórmula:C38H53N5O7Forma y color:SolidPeso molecular:691.86Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Fórmula:C36H42N6O7Forma y color:SolidPeso molecular:670.75Axomadol
CAS:<p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>Fórmula:C16H25NO3Pureza:98%Forma y color:SolidPeso molecular:279.37LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Fórmula:C32H42N4O6Pureza:98%Forma y color:SolidPeso molecular:578.7Diallyl G
CAS:<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Fórmula:C38H53N5O8Forma y color:SolidPeso molecular:707.86Loperamide oxide
CAS:<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Fórmula:C29H33ClN2O3Forma y color:SolidPeso molecular:493.04CR-665 Acetate
CAS:<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Fórmula:C38H53N9O6Forma y color:SolidPeso molecular:731.899AZD7268
CAS:<p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>Fórmula:C29H30N4O2SForma y color:SolidPeso molecular:498.64AT-076
CAS:<p>AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.</p>Fórmula:C26H35N3O3Forma y color:SolidPeso molecular:437.57GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Fórmula:C24H23F2N4O4PPureza:98%Forma y color:SolidPeso molecular:500.43Dup 747
CAS:<p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>Fórmula:C24H28Cl2N2O2Pureza:98%Forma y color:SolidPeso molecular:447.4σ1 Receptor/μ Opioid receptor modulator 1
CAS:<p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>Fórmula:C24H31FN2O2Forma y color:SolidPeso molecular:398.51
