
Receptor de bradicinina
Los receptores de bradicinina son GPCR que median los efectos de la bradicinina, un péptido involucrado en las respuestas inflamatorias, la sensación de dolor y la regulación de la presión arterial. Hay dos tipos principales de receptores de bradicinina, B1 y B2, cada uno con roles distintos en procesos fisiopatológicos. Los antagonistas de los receptores de bradicinina se utilizan en el tratamiento de afecciones como el angioedema hereditario, el dolor crónico y la hipertensión. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de bradicinina de alta calidad para apoyar su investigación en inflamación, manejo del dolor y biología cardiovascular.
Se han encontrado 61 productos de "Receptor de bradicinina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Thrombostatin cont-1
CAS:Thrombostatin cont-1, an analogue of the bradykinin metabolite thrombostatin, has been shown to reduce platelet activation in the canine carotid arteryFórmula:C87H142N34O29S2Peso molecular:2192.4FR167344 free base
CAS:FR167344 free base: oral, nonpeptide B2 bradykinin receptor antagonist, high-affinity (IC50: 65 nM), no B1 affinity.Fórmula:C30H28BrCl2N5O4Pureza:98%Forma y color:SolidPeso molecular:673.38Bradykinin (1-3)
CAS:Bradykinin (1-3) is a fragment of Bradykinin. Bradykinin is an activates pain receptors.
Fórmula:C16H28N6O4Pureza:98%Forma y color:SolidPeso molecular:368.43FR190997
CAS:FR190997 is an agonist of bradykinin B2 receptor.Fórmula:C37H33Cl2N5O5Forma y color:SolidPeso molecular:698.59L 366811
CAS:L 366811 is a potent oxytocin antagonist.Fórmula:C43H56N8O6Forma y color:SolidPeso molecular:780.95MEN 11270
CAS:B2 bradykinin receptor peptide antagonist, pKi 10.3; improves hypotension, bronchoconstriction; B2-selective over 29 receptors/ion channels.Fórmula:C60H90N20O11SPureza:98%Forma y color:SolidPeso molecular:1299.56JMV-1645
CAS:JMV-1645 is an effective and selective B(1) bradykinin receptor antagonist.Fórmula:C49H69N13O12SPureza:98%Forma y color:SolidPeso molecular:1064.23Bradykinin (1-7)
CAS:Bradykinin (1-7), an amino-truncated peptide derived from Bradykinin, is a metabolite formed through enzymatic cleavage by endopeptidase.Fórmula:C35H52N10O9Pureza:98%Forma y color:White Lyophilized PowderPeso molecular:756.85Bradykinin (1-6)
CAS:Bradykinin (1-6) is a stable, CPY-cleaved metabolite that triggers pain, induces muscle contractions, and activates NO synthetase.Fórmula:C30H45N9O8Pureza:98%Forma y color:SolidPeso molecular:659.73Lys-[Des-Arg9]Bradykinin
CAS:Selective bradykinin B1 agonist with Ki 0.12 nM; inactive at B2 (>30,000 nM). Lowers blood pressure, more potent than Des-Arg9-Bradykinin.Fórmula:C50H73N13O11Pureza:98%Forma y color:SolidPeso molecular:1032.21Retrobradykinin
CAS:Bradykinin analog nonapeptide. Reverse sequence of Bradykinin. Exhibits no significant kinin activity. Can be used as a negative control.Fórmula:C50H73N15O11Forma y color:SolidPeso molecular:1060.228Lys-[Hyp3]-Bradykinin
CAS:Lys-[Hyp3]-Bradykinin, a human urine-derived kinin and bradykinin agonist, is used for inflammation research.Fórmula:C56H85N17O13Forma y color:SolidPeso molecular:1204.38[Des-Arg9]-Bradykinin
CAS:[Des-Arg9]-Bradykinin ([Des-Arg9]-Bradykinin(2TFA))(2TFA) is an agonist of Bradykinin (B1) receptor.Fórmula:C44H61N11O10Pureza:98%Forma y color:SolidPeso molecular:904.02B-Raf IN 14
CAS:B-Raf IN 14 is a BRAF inhibitor.Fórmula:C15H14BrN5O3SPureza:98.38%Forma y color:SolidPeso molecular:424.27[Des-Arg9]-Bradykinin acetate
CAS:[Des-Arg9]-Bradykinin acetate is a selective agonist of Bradykinin B1 receptor.Fórmula:C46H65N11O12Pureza:99.05%Forma y color:SolidPeso molecular:964.07Bradykinin (1-5)
CAS:Bradykinin (1-5), a stable metabolite of BK produced by ACE, serves as a marker for in vivo BK generation.Fórmula:C27H40N8O6Forma y color:SolidPeso molecular:572.66Sar-[D-Phe8]-des-Arg9-Bradykinin acetate
Sar-[D-Phe8]-des-Arg9-Bradykinin acetate is a potent and selective bradykinin B1 receptor agonist (EC50 = 9.02 nM in rabbit aorta) that is resistant toFórmula:C49H70N12O13Pureza:99.93%Forma y color:SolidPeso molecular:1035.15Icatibant Acetate
CAS:Icatibant Acetate, an antagonist of the bradykinin B2 receptor, is used in the treatment of hereditary angioedema.Fórmula:C61H93N19O15SPureza:99.68% - 99.90%Forma y color:SolidPeso molecular:1364.57Ref: TM-T22344
1mg66,00€2mg92,00€5mg177,00€10mg281,00€1mL*10mM (DMSO)355,00€25mg475,00€50mg677,00€100mg888,00€5-Hydroxy-1-methylhydantoin
CAS:5-Hydroxy-1-methylhydantoin (HD-003) is an antioxidant potentially for the treatment of renal failure.Fórmula:C4H6N2O3Pureza:99.99%Forma y color:SolidPeso molecular:130.1Bradykinin
CAS:Bradykinin is an inflammatory mediator.Fórmula:C50H73N15O11Pureza:99.68%Forma y color:SolidPeso molecular:1060.21

