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Receptor de bradicinina

Receptor de bradicinina

Los receptores de bradicinina son GPCR que median los efectos de la bradicinina, un péptido involucrado en las respuestas inflamatorias, la sensación de dolor y la regulación de la presión arterial. Hay dos tipos principales de receptores de bradicinina, B1 y B2, cada uno con roles distintos en procesos fisiopatológicos. Los antagonistas de los receptores de bradicinina se utilizan en el tratamiento de afecciones como el angioedema hereditario, el dolor crónico y la hipertensión. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de bradicinina de alta calidad para apoyar su investigación en inflamación, manejo del dolor y biología cardiovascular.

Se han encontrado 59 productos de "Receptor de bradicinina"

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  • SSR240612

    CAS:
    <p>SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,</p>
    Fórmula:C42H53ClN4O7S
    Pureza:98.59% - 99.16%
    Forma y color:Solid
    Peso molecular:793.41
  • Bradykinin (acetate)

    CAS:
    <p>Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.</p>
    Fórmula:C52H77N15O13
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1120.26
  • Lys-[Des-Arg9]Bradykinin,TFA


    <p>Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and B2</p>
    Fórmula:C54H75F6N13O15
    Pureza:97.35%
    Forma y color:Solid
    Peso molecular:1260.24
  • [Des-Arg9]-Bradykinin TFA

    CAS:
    <p>[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.</p>
    Fórmula:C46H62F3N11O12
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1018.05
  • Bradykinin (2-9)

    CAS:
    <p>Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.</p>
    Fórmula:C44H61N11O10
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:904.02
  • R715 TFA(185052-09-9 free base)


    <p>R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).</p>
    Fórmula:C59H82F3N13O14
    Pureza:>99.99%
    Forma y color:Solid
    Peso molecular:1254.36
  • Lys-Bradykinin acetate(342-10-9 free base)

    CAS:
    <p>Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.</p>
    Fórmula:C58H89N17O14
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:1248.43
  • Lys-[Des-Arg9]Bradykinin acetate


    <p>Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and &gt; 30000 nM at human B1 and</p>
    Fórmula:C52H77N13O13
    Pureza:99.93%
    Forma y color:Solid
    Peso molecular:1092.27
  • BKM-570

    CAS:
    <p>BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.</p>
    Fórmula:C34H34Cl2F5N3O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:698.55
  • Anatibant

    CAS:
    <p>Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.</p>
    Fórmula:C34H36Cl2N6O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:711.66
  • Fulimetibant

    CAS:
    <p>Fulimetibant is a bradykinin receptor antagonist.</p>
    Fórmula:C25H21F4N3O3
    Forma y color:Solid
    Peso molecular:487.45
  • B 4148

    CAS:
    <p>B 4148 is a bradykinin inhibitor.</p>
    Fórmula:C62H95N19O14S2
    Forma y color:Solid
    Peso molecular:1394.67
  • NPC 17731

    CAS:
    <p>NPC 17731 is a bradykinin receptor antagonist.</p>
    Fórmula:C59H95N19O14
    Forma y color:Solid
    Peso molecular:1294.5
  • MK-0686

    CAS:
    <p>MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.</p>
    Fórmula:C22H19ClF4N2O4
    Pureza:99.88%
    Forma y color:Solid
    Peso molecular:486.84
  • Safotibant

    CAS:
    <p>Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edema</p>
    Fórmula:C25H34N4O5S
    Pureza:99.62% - 99.67%
    Forma y color:Solid
    Peso molecular:502.63
  • NVP-SAA164

    CAS:
    <p>NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.</p>
    Fórmula:C36H45N5O5S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:659.84
  • FK-3657

    CAS:
    <p>FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.</p>
    Fórmula:C30H27Cl2N5O4
    Forma y color:Solid
    Peso molecular:592.47
  • Fasitibant

    CAS:
    <p>Fasitibant is a potent and selective nonpeptide kinin B2 receptor antagonist.</p>
    Fórmula:C36H49Cl2N6O6S
    Forma y color:Solid
    Peso molecular:764.78
  • BI-113823

    CAS:
    <p>BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.</p>
    Fórmula:C26H44N4O5S
    Forma y color:Solid
    Peso molecular:524.716