Receptor de bradicinina
Los receptores de bradicinina son GPCR que median los efectos de la bradicinina, un péptido involucrado en las respuestas inflamatorias, la sensación de dolor y la regulación de la presión arterial. Hay dos tipos principales de receptores de bradicinina, B1 y B2, cada uno con roles distintos en procesos fisiopatológicos. Los antagonistas de los receptores de bradicinina se utilizan en el tratamiento de afecciones como el angioedema hereditario, el dolor crónico y la hipertensión. En CymitQuimica, ofrecemos una variedad de moduladores de receptores de bradicinina de alta calidad para apoyar su investigación en inflamación, manejo del dolor y biología cardiovascular.
Se han encontrado 61 productos de "Receptor de bradicinina"
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Emorfazone
CAS:Emorfazone (PH011085) has an anti-nociceptive effect.Fórmula:C11H17N3O3Pureza:99.89%Forma y color:SolidPeso molecular:239.27Ref: TM-T9132
1mg84,00€1mL*10mM (DMSO)152,00€5mg168,00€10mg245,00€25mg404,00€50mg567,00€100mg767,00€200mg1.018,00€ELN-441958
CAS:ELN-441958 is a potent, neutral antagonist of B1 receptor, inhibits the binding of the B1 agonist ligand [3H]DAKD to IMR-90 cells with Ki of 0.26 nM.Fórmula:C29H29ClN4O2Pureza:99.88%Forma y color:SolidPeso molecular:501.02Ref: TM-T2086
1mg58,00€5mg128,00€1mL*10mM (DMSO)141,00€10mg200,00€25mg339,00€50mg485,00€100mg658,00€200mg889,00€SSR240612
CAS:SSR240612 is a potent, and orally active specific non-peptide bradykinin B1 receptor antagonist (Kis = 0.48-0.73 and 358-481 nM for B1 and B2 receptors,Fórmula:C42H53ClN4O7SPureza:98.59% - 99.16%Forma y color:SolidPeso molecular:793.41Ref: TM-T5048
1mg222,00€5mg512,00€1mL*10mM (DMSO)612,00€10mg700,00€25mg982,00€50mg1.333,00€100mg1.783,00€Bradykinin (acetate)
CAS:Bradykinin (acetate) is an active peptide that is generated by the kallikrein-kinin system.Fórmula:C52H77N15O13Pureza:>99.99%Forma y color:SolidPeso molecular:1120.26Lys-[Des-Arg9]Bradykinin,TFA
Lys-[Des-Arg9]Bradykinin,TFA is Endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 and B2Fórmula:C54H75F6N13O15Pureza:97.35%Forma y color:SolidPeso molecular:1260.24[Des-Arg9]-Bradykinin TFA
CAS:[Des-Arg9]-Bradykinin is an agonist of Bradykinin (B1) receptor that displays selectivity for B1 over B2 receptors.Fórmula:C46H62F3N11O12Pureza:>99.99%Forma y color:SolidPeso molecular:1018.05Bradykinin (2-9)
CAS:Bradykinin (2-9) (Des-Arg1-bradykinin) is an amino-truncated peptide compound that is a metabolite of Bradykinin.Fórmula:C44H61N11O10Pureza:>99.99%Forma y color:SolidPeso molecular:904.02Ref: TM-TP1181
1mg39,00€5mg88,00€10mg130,00€1mL*10mM (DMSO)144,00€25mg210,00€50mg313,00€100mg464,00€200mg660,00€R715 TFA(185052-09-9 free base)
R715 TFA(185052-09-9 free base) is a potent and selective bradykinin B1 receptor antagonist (pA2 = 8.49).Fórmula:C59H82F3N13O14Pureza:>99.99%Forma y color:SolidPeso molecular:1254.36Lys-Bradykinin acetate(342-10-9 free base)
CAS:Lys-Bradykinin acetate is an endogenous bradykinin receptor agonist.Fórmula:C58H89N17O14Pureza:99.86%Forma y color:SolidPeso molecular:1248.43Lys-[Des-Arg9]Bradykinin acetate
Lys-[Des-Arg9]Bradykinin acetate is an endogenous potent and highly selective bradykinin B1 receptor agonist (Ki values are 0.12 and > 30000 nM at human B1 andFórmula:C52H77N13O13Pureza:99.93%Forma y color:SolidPeso molecular:1092.27B 4148
CAS:B 4148 is a bradykinin inhibitor.Fórmula:C62H95N19O14S2Forma y color:SolidPeso molecular:1394.67NPC 17731
CAS:NPC 17731 is a bradykinin receptor antagonist.Fórmula:C59H95N19O14Forma y color:SolidPeso molecular:1294.5BKM-570
CAS:BKM-570, a bradykinin antagonist, causes impressive growth inhibition of lung and prostate tumors.Fórmula:C34H34Cl2F5N3O3Pureza:98%Forma y color:SolidPeso molecular:698.55Anatibant
CAS:Anatibant: a strong non-peptide, inhibits bradykinin B2; lowers brain swelling and damage post-trauma.Fórmula:C34H36Cl2N6O5SPureza:98%Forma y color:SolidPeso molecular:711.66Fulimetibant
CAS:Fulimetibant is a bradykinin receptor antagonist.Fórmula:C25H21F4N3O3Forma y color:SolidPeso molecular:487.45MK-0686
CAS:MK-0686 is an orally available bradykinin B1 receptor antagonist with potential anti-inflammatory activity.Fórmula:C22H19ClF4N2O4Pureza:99.88%Forma y color:SolidPeso molecular:486.84Safotibant
CAS:Safotibant (LF-22-0542) is a bradykinin B1 receptor antagonist with anti-inflammatory and analgesic activity for the topical treatment of diabetic macular edemaFórmula:C25H34N4O5SPureza:99.62% - 99.67%Forma y color:SolidPeso molecular:502.63NVP-SAA164
CAS:NVP-SAA164 is a nonpeptide bradykinin B1 receptor antagonist agent.Fórmula:C36H45N5O5SPureza:98%Forma y color:SolidPeso molecular:659.84FK-3657
CAS:FK-3657 is a non-peptide antagonist of bradykinin (BK)-B2 receptor.Fórmula:C30H27Cl2N5O4Forma y color:SolidPeso molecular:592.47BI-113823
CAS:BI-113823 is an orally active and selective bradykinin B1 receptor antagonist. It alleviates mechanical hyperalgesia induced by complete Freund's adjuvant in rats. BI-113823 is applicable for research on chronic inflammatory pain.Fórmula:C26H44N4O5SForma y color:SolidPeso molecular:524.716
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