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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Clozapine N-Oxide

    CAS:
    <p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>
    Fórmula:C18H19ClN4O
    Pureza:98.43% - 99.94%
    Forma y color:Solid
    Peso molecular:342.82
  • A-381393

    CAS:
    <p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>
    Fórmula:C20H24N4
    Pureza:99.00%
    Forma y color:Solid
    Peso molecular:320.43
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Forma y color:White Solid
    Peso molecular:463
  • Alizapride

    CAS:
    <p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>
    Fórmula:C16H21N5O2
    Forma y color:Solid
    Peso molecular:315.37
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Fórmula:C17H18BrNO
    Pureza:95.00% - 99.82%
    Forma y color:Solid
    Peso molecular:332.23
  • Protein deglycase DJ-1 against-1

    CAS:
    <p>Protein deglycase DJ-1 against-1 penetrate the BBB and bind to DJ-1 protein,restoring neuronal cellular death in a neurotoxin MPTP-induced model of PD.</p>
    Fórmula:C24H23N3O4
    Pureza:97.23%
    Forma y color:Solid
    Peso molecular:417.46
  • Trazpiroben

    CAS:
    <p>Trazpiroben (TAK-906) is a selective dopamine D2/D3 receptor antagonist used in the study of gastroparesis.</p>
    Fórmula:C31H39N3O4
    Pureza:99.41% - >99.99%
    Forma y color:Solid
    Peso molecular:517.66
  • Dexpramipexole

    CAS:
    <p>Dexpramipexole ((R)-Pramipexole) is a mitochondrial protective agent that maintains mitochondrial function and energy production.</p>
    Fórmula:C10H17N3S
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:211.33
  • Ropinirole

    CAS:
    <p>Ropinirole, D2-like agonist, no D1 affinity, Ki 29 nM for D2, treats Parkinson's.</p>
    Fórmula:C16H24N2O
    Pureza:99.68%
    Forma y color:Solid
    Peso molecular:260.38
  • L-745870

    CAS:
    <p>L-745870 is a D4 receptor antagonist that also inhibits D2 receptors, 5-HT2 receptors, and α-adrenergic receptors.</p>
    Fórmula:C18H19ClN4
    Pureza:98%
    Forma y color:Solid
    Peso molecular:326.82
  • Vanoxerine

    CAS:
    <p>Vanoxerine is an antagonist of dopamine transporter (Ki: 16.9nM).</p>
    Fórmula:C28H32F2N2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:450.56
  • Pardoprunox

    CAS:
    <p>Pardoprunox (SLV-308) is a partial dopamine D2 agonist and noradrenergic agonist with serotonin 5-HT1A agonist properties.</p>
    Fórmula:C12H15N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:233.27
  • A23887

    CAS:
    <p>A23887 is a potentially neuroleptic tetracyclic spiro amine that has affinity for dopamine D-2 receptors.</p>
    Fórmula:C22H24ClN
    Pureza:98%
    Forma y color:Solid
    Peso molecular:337.89
  • SCH-23390 maleate

    CAS:
    <p>SCH-23390 maleate (R-(+)-SCH-23390 maleate) is a potent and selective antagonist of dopamine D1-like receptor (1 and D5 receptor with Kis of 0.2 nM and 0.3 nM,</p>
    Fórmula:C21H22ClNO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:403.86
  • Quinpirole Hydrochloride

    CAS:
    <p>Quinpirole Hydrochloride (LY 171555), as an agonist with high affinity for dopamine receptor D2/D3, has been widely used to study the function of dopamine receptor D2/D3 in humans and mice</p>
    Fórmula:C13H22ClN3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:255.79
  • Fallypride

    CAS:
    <p>Fallypride is a potent and selective dopamine D2/D3 receptor antagonist.</p>
    Fórmula:C20H29FN2O3
    Pureza:98.97% - >99.99%
    Forma y color:Solid
    Peso molecular:364.45
  • CP-226269

    CAS:
    <p>CP-226269 is a potent dopamine D4 receptor agonist that regulates calcium flux and has an EC50 value of 32.0 nM.</p>
    Fórmula:C18H19FN4
    Pureza:99.08%
    Forma y color:Solid
    Peso molecular:310.37
  • PD 120697

    CAS:
    <p>PD 120697 is a dopamine antagonist with central dopamine agonist properties.</p>
    Fórmula:C11H15N3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:221.32
  • Talipexole

    CAS:
    <p>Talipexole (B-HT920) is an agonist of dopamine, and is an antiparkinsonian agent.</p>
    Fórmula:C10H15N3S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:209.31
  • Foscarbidopa

    CAS:
    <p>Foscarbidopa is a prodrug of Carbidopa. It acts as a dopamine receptor agonist.</p>
    Fórmula:C10H15N2O7P
    Pureza:96.17% - 97.27%
    Forma y color:Solid
    Peso molecular:306.21