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Receptor de dopamina

Receptor de dopamina

Los receptores de dopamina son un grupo de receptores acoplados a proteínas G (GPCR) que responden al neurotransmisor dopamina, jugando un papel clave en la regulación del movimiento, la motivación, la recompensa y varias funciones cognitivas. Estos receptores se dividen en familias similares a D1 y D2, cada una con funciones y perfiles farmacológicos distintos. Los moduladores de los receptores de dopamina se estudian ampliamente por sus aplicaciones en el tratamiento de la enfermedad de Parkinson, la esquizofrenia, la adicción y otros trastornos neuropsiquiátricos. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores de dopamina de alta calidad para apoyar su investigación en neurociencia, salud mental y señalización GPCR.

Se han encontrado 407 productos de "Receptor de dopamina"

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  • Bromopride

    CAS:
    <p>Bromopride (Valopride), a metoclopramide-like dopamine antagonist and prokinetic, is an antiemetic not sold in the US or UK.</p>
    Fórmula:C14H22BrN3O2
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:344.25
  • Oxidopamine hydrobromide

    CAS:
    <p>Oxidopamine hydrobromide (6-OHDA hydrobromide) is a neurotransmitter dopamine antagonist.</p>
    Fórmula:C8H12BrNO3
    Pureza:98.22% - 99.88%
    Forma y color:Beige To Brown Fine Crystalline Powder
    Peso molecular:250.09
  • NEO 376

    CAS:
    <p>NEO 376 (SPI-376) is a selective 5-HT1 receptor, GABA receptor and dopamine receptor modulator, showing anti-psychotic actively.</p>
    Fórmula:C20H24ClN3O
    Pureza:99.56%
    Forma y color:Solid
    Peso molecular:357.88
  • GR 103691

    CAS:
    <p>GR 103691 is a potent, selective dopamine D3 receptor antagonist (Ki: 0.4 nM).</p>
    Fórmula:C30H35N3O3
    Pureza:98.94% - 99.29%
    Forma y color:Solid
    Peso molecular:485.62
  • Bromperidol

    CAS:
    <p>Bromperidol (R-11333) is a butyrophenone derivative and it is a potent and long-acting neuroleptic.</p>
    Fórmula:C21H23BrFNO2
    Pureza:99.89%
    Forma y color:Tan Solid
    Peso molecular:420.32
  • Quetiapine hemifumarate

    CAS:
    <p>Quetiapine hemifumarate (ICI-204636), an atypical antipsychotic, is used in the treatment of bipolar I mania, schizophrenia, bipolar I/II depression,.</p>
    Fórmula:C46H54N6O8S2
    Pureza:99.32% - >99.99%
    Forma y color:White Crystalline Solid
    Peso molecular:883.09
  • Prochlorperazine Maleate

    CAS:
    <p>Prochlorperazine Maleate (Capazine) is a phenothiazine antipsychotic used principally in the treatment of NAUSEA; VOMITING; and VERTIGO.</p>
    Fórmula:C28H32ClN3O8S
    Pureza:99.78%
    Forma y color:Off-White Powder
    Peso molecular:606.09
  • Tiapride hydrochloride

    CAS:
    <p>Tiapride is a selective blocker of D2/3 dopamine receptors in the brain.</p>
    Fórmula:C15H24N2O4S·HCl
    Pureza:99.4% - 99.77%
    Forma y color:Solid
    Peso molecular:364.89
  • L-DOPA

    CAS:
    <p>L-DOPA (Levodopa) is an amino acid precursor of dopamine with antiparkinsonian properties. Levodopa that is converted to dopamine by DOPA decarboxylase.</p>
    Fórmula:C9H11NO4
    Pureza:98.99% - 99.93%
    Forma y color:Colorless To White Crystals Or Crystalline Powder; Needles From Water Solid
    Peso molecular:197.19
  • Ziprasidone hydrochloride

    CAS:
    <p>Ziprasidone hydrochloride (CP-88059 hydrochloride) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic</p>
    Fórmula:C21H22CL2N4OS
    Pureza:97.97% - 99.82%
    Forma y color:Solid
    Peso molecular:449.4
  • Thioridazine hydrochloride

    CAS:
    <p>Thioridazine hydrochloride (Mellaril) , an antipsychotic drug, is used in the therapy of psychosis and schizophrenia and shows serotonin antagonism or D4</p>
    Fórmula:C21H27ClN2S2
    Pureza:99.55% - 99.957%
    Forma y color:White To Off-White Solid
    Peso molecular:407.04
  • Metoclopramide hydrochloride

    CAS:
    <p>Metoclopramide hydrochloride (Metoclopramide HCl) is a selective dopamine D2 receptor antagonist, used as an antiemetic.</p>
    Fórmula:C14H22ClN3O2·HCl
    Pureza:99.99%
    Forma y color:White To Off-White Powder
    Peso molecular:336.26
  • Quetiapine

    CAS:
    <p>Quetiapine treats schizophrenia and bipolar I, targeting serotonin, dopamine, and adrenoreceptor subtypes, plus H1 histamine receptor.</p>
    Fórmula:C21H25N3O2S
    Pureza:99.14% - 99.63%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:383.51
  • Sulpiride

    CAS:
    <p>Sulpiride (Aiglonyl) is a dopamine D2-receptor antagonist, used therapeutically as an antidepressant, antipsychotic, and as a digestive aid.</p>
    Fórmula:C15H23N3O4S
    Pureza:99.94%
    Forma y color:White Crystalline Powder
    Peso molecular:341.43
  • Amisulpride

    CAS:
    <p>Amisulpride (Solian/Deniban), a dopamine antagonist antipsychotic, treats psychosis and schizophrenia in Europe/Australia, not in the US.</p>
    Fórmula:C17H27N3O4S
    Pureza:99.97%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:369.48
  • L-741626

    CAS:
    <p>L-741626 (3-(4-(4-Chlorophenyl-4-hydroxypiperidino)methyl)indole) is a selective antagonist of D2 dopamine receptor (Ki: 2.4, 100, and 220 nM for human D2, D3</p>
    Fórmula:C20H21ClN2O
    Pureza:98.57%
    Forma y color:Solid
    Peso molecular:340.85
  • Ziprasidone

    CAS:
    <p>Ziprasidone (Geodon) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of antipsychotic activity.</p>
    Fórmula:C21H21ClN4OS
    Pureza:99.55%
    Forma y color:Tan Solid
    Peso molecular:412.94
  • Dexpramipexole dihydrochloride

    CAS:
    <p>Dexpramipexole dihydrochloride (KNS-760704 dihydrochloride) ((R)-Pramipexole dihydrochloride) is a neuroprotective agent and is a weak non-ergoline dopamine</p>
    Fórmula:C10H19Cl2N3S
    Pureza:99.75% - 99.88%
    Forma y color:Solid
    Peso molecular:284.25
  • Flunarizine dihydrochloride

    CAS:
    <p>Flunarizine dihydrochloride: a calcium blocker also targeting calmodulin and histamine H1, used for migraine, vertigo, vascular disease, and epilepsy aid.</p>
    Fórmula:C26H28Cl2F2N2
    Pureza:99.53% - 99.89%
    Forma y color:White Crystalline Powder Odorless And Tasteless
    Peso molecular:477.42
  • Tipepidine hydrochloride

    CAS:
    <p>Tipepidine hydrochloride: reversible DA D2 receptor inhibitor, IC50 7.0 μM, with antidepressant effects.</p>
    Fórmula:C15H18ClNS2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:311.89
  • Blonanserin

    CAS:
    <p>Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.</p>
    Fórmula:C23H30FN3
    Pureza:99.85%
    Forma y color:Solid
    Peso molecular:367.5
  • Levosulpiride

    CAS:
    <p>Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.</p>
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Forma y color:White Crystalline Powder
    Peso molecular:341.43
  • Mefexamide hydrochloride

    CAS:
    <p>Mefexamide hydrochloride is a central stimulant.</p>
    Fórmula:C15H25ClN2O3
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:316.83
  • Ziprasidone hydrochloride monohydrate

    CAS:
    <p>Ziprasidone hydrochloride monohydrate (CP 88059) is a united 5-HT (serotonin) and dopamine receptor antagonist which shows potent effects of the antipsychotic</p>
    Fórmula:C21H21ClN4OS·HCl·H2O
    Pureza:98% - 99.83%
    Forma y color:Off-White Powder
    Peso molecular:467.12
  • Loxapine succinate

    CAS:
    <p>Loxapine succinate (Loxapac), a D2DR and D4DR inhibitor, is utilized in schizophrenia.</p>
    Fórmula:C22H24ClN3O5
    Pureza:99.69%
    Forma y color:White To Of-White Solid
    Peso molecular:445.9
  • Tetrahydropalmatine

    CAS:
    <p>Tetrahydropalmatine (DL-Tetrahydropalmatine) is an active component isolated from corydalis, suppressing amygdaloid release of dopamine to inhibit an epileptic</p>
    Fórmula:C21H25NO4
    Pureza:99.59% - 99.95%
    Forma y color:Solid
    Peso molecular:355.43
  • Talipexole dihydrochloride

    CAS:
    <p>Talipexole dihydrochloride (Domnin) is a dopamine D2 receptor agonist, α2-adrenoceptor agonist, and 5-HT3 receptor antagonist in both rat cortical and</p>
    Fórmula:C10H17Cl2N3S
    Pureza:99.89%
    Forma y color:Light Yellow Solid
    Peso molecular:282.23
  • Benserazide hydrochloride

    CAS:
    <p>Benserazide hydrochloride (Ro 4-4602) is a peripherally-acting L-amino acid decarboxylase (AAAD) or DOPA decarboxylase inhibitor.</p>
    Fórmula:C10H15N3O5·HCl
    Pureza:98.63% - 99.74%
    Forma y color:White Crystalline Solid
    Peso molecular:293.7
  • BP 897 hydrochloride

    CAS:
    <p>BP 897: potent D3 agonist (Ki: 0.92 nM), weak D2 antagonist (Ki: 61 nM), low affinity for D1/D4.</p>
    Fórmula:C26H32ClN3O2
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:454
  • Pipamperone

    CAS:
    <p>Pipamperone (McN-JR 3345) binds 5-HT2A closely as receptor.</p>
    Fórmula:C21H30FN3O2
    Pureza:99.85%
    Forma y color:White Powder
    Peso molecular:375.48
  • Chlorprothixene hydrochloride

    CAS:
    <p>Chlorprothixene hydrochloride, a typical antipsychotic, blocks 5-HT2, D1-D3, H1, muscarinic, and alpha1 receptors.</p>
    Fórmula:C18H18ClNS·HCl
    Pureza:99.76%
    Forma y color:White Powder
    Peso molecular:352.32
  • Promazine hydrochloride

    CAS:
    <p>Promazine hydrochloride, a phenothiazine less potent than chlorpromazine, treats disturbed behavior and nausea.</p>
    Fórmula:C17H21ClN2S
    Pureza:99.90%
    Forma y color:Solid
    Peso molecular:320.88
  • Ro 10-5824 dihydrochloride

    CAS:
    <p>Ro 10-5824 dihydrochloride is a selective agonist of dopamine D4 receptor partial, (Ki of 5.2 nM).</p>
    Fórmula:C17H22Cl2N4
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:353.29
  • Fosopamine(HCl)

    CAS:
    <p>Fosopamine(HCl) is a DRDs agonist that can be used to study hypertension.</p>
    Fórmula:C9H15ClNO5P
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:283.65
  • Domperidone

    CAS:
    <p>Domperidone (R33812)(Motilium) is a dopamine blocker and an antidopaminergic reagent.</p>
    Fórmula:C22H24ClN5O2
    Pureza:98% - 99.82%
    Forma y color:Solid
    Peso molecular:425.91
  • Talquetamab

    CAS:
    <p>Talquetamab (JNJ-64407564) is a T-cell retargeting GPRC5D bispecific antibody with antitumor activity for the treatment of multiple myeloma.</p>
    Forma y color:Liquid
    Peso molecular:144.59 kDa
  • Itopride hydrochloride

    CAS:
    <p>Itopride hydrochloride (Ganaton) is an AChE and D2DR inhibitor.</p>
    Fórmula:C20H27ClN2O4
    Pureza:99.59%
    Forma y color:White Or Pale Brownish Crystal
    Peso molecular:394.9
  • Oxidopamine hydrochloride

    CAS:
    <p>Oxidopamine hydrochloride (6-Hydroxydopamine hydrochloride) is an neurotransmitter dopamine antagonist.</p>
    Fórmula:C8H12ClNO3
    Pureza:98.34% - 99.85%
    Forma y color:Physical Description Beige Solid (Ntp 1992)
    Peso molecular:205.64
  • Benztropine mesylate

    CAS:
    <p>Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON</p>
    Fórmula:C21H25NO·CH4SO3
    Pureza:98.41% - 99.96%
    Forma y color:White Crystalline Powder; Odourless Or Almost Odourless
    Peso molecular:403.53
  • Paliperidone

    CAS:
    <p>Paliperidone (9-hydroxyrisperidone)(Invega) is used as an atypical antipsychotic.</p>
    Fórmula:C23H27FN4O3
    Pureza:95% - 99.08%
    Forma y color:Off White To Light Orange Coloured Solid
    Peso molecular:426.48
  • Bendazol

    CAS:
    <p>Bendazol (Dibazol) is always used as the drug for hypertension and cerebral Angiospasm.</p>
    Fórmula:C14H12N2
    Pureza:98.7% - 99.87%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:208.26
  • Pericyazine

    CAS:
    <p>Pericyazine (Propericiazine) is a selective D2-dopamine receptor antagonist.</p>
    Fórmula:C21H23N3OS
    Pureza:99.61%
    Forma y color:Solid
    Peso molecular:365.49
  • Tetrabenazine

    CAS:
    <p>Tetrabenazine (Ro 1-9569) is a drug formerly used as an antipsychotic and treatment of various movement disorders.</p>
    Fórmula:C19H27NO3
    Pureza:98% - 99.91%
    Forma y color:White To Off-White White To Off-White Solid
    Peso molecular:317.42
  • Perphenazine

    CAS:
    <p>Perphenazine (Trilafon) is a phenothiazine derivative and a dopamine antagonist with antiemetic and antipsychotic properties.</p>
    Fórmula:C21H26ClN3OS
    Pureza:99.3% - 99.99%
    Forma y color:Solid
    Peso molecular:403.97
  • Clozapine

    CAS:
    <p>Clozapine (HF 1854) is a tricylic dibenzodiazepine, classified as an atypical antipsychotic agent.</p>
    Fórmula:C18H19ClN4
    Pureza:99.91% - 99.93%
    Forma y color:Yellow Crystals From Acetone-Petroleum Ether Solid
    Peso molecular:326.82
  • Olanzapine

    CAS:
    <p>Olanzapine (LY170053) is an atypical antipsychotic that is used currently in the treatment of schizophrenia and bipolar illness.</p>
    Fórmula:C17H20N4S
    Pureza:99.86% - ≥95%
    Forma y color:Yellowish Crystalline Powder
    Peso molecular:312.43
  • Acetophenazine dimaleate

    CAS:
    <p>Acetophenazine dimaleate is an antipsychotic agent, effective in anxious depression. Acetophenazine dimaleate primarily targets the dopamine D2 receptor.</p>
    Fórmula:C31H37N3O10S
    Pureza:99.39% - 99.48%
    Forma y color:Solid
    Peso molecular:643.71
  • Pramipexole

    CAS:
    <p>Pramipexole (SND 919), a dopamine agonist for Parkinson's, may cause mild, temporary enzyme spikes, not acute liver injury.</p>
    Fórmula:C10H17N3S
    Pureza:98% - 99.96%
    Forma y color:Solid
    Peso molecular:211.33
  • Iloperidone

    CAS:
    <p>Iloperidone (HP 873) is an atypical antipsychotic agent that is used for treatment of schizophrenia.</p>
    Fórmula:C24H27FN2O4
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:426.48
  • Dopamine hydrochloride

    CAS:
    <p>Dopamine hydrochloride (ASL279) is a natural catecholamine neurotransmitter, dopamine receptors (D1-5 receptors) (EC50=2.7 nM). High-Quality, Low-Cost!</p>
    Fórmula:C8H12ClNO2
    Pureza:99.47% - 99.72%
    Forma y color:Solid
    Peso molecular:189.64
  • Fluphenazine dihydrochloride

    CAS:
    <p>Fluphenazine dihydrochloride (Prolixin) is an inhibitor of phenothiazine-class D1DR and D2DR. Fluphenazine can be used to probe effects and metabolic process.</p>
    Fórmula:C22H28Cl2F3N3OS
    Pureza:99.23%
    Forma y color:Off-White Solid
    Peso molecular:510.44
  • Trifluoperazine dihydrochloride

    CAS:
    <p>Trifluoperazine dihydrochloride (SKF5019) is a potent dopamine D2 receptor inhibitor used as an antipsychotic and an antiemetic.</p>
    Fórmula:C21H26Cl2F3N3S
    Pureza:99.57% - 99.96%
    Forma y color:Cream Fine Powder
    Peso molecular:480.43
  • Molindone hydrochloride

    CAS:
    <p>Molindone hydrochloride (EN-1733A) is an indole derivative effective in schizophrenia and other psychoses by blocking the effects of dopamine in the brain.</p>
    Fórmula:C16H24N2O2·HCl
    Pureza:99% - 99.99%
    Forma y color:Solid
    Peso molecular:312.84
  • Droperidol

    CAS:
    <p>Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.</p>
    Fórmula:C22H22FN3O2
    Pureza:97.16% - 98%
    Forma y color:Solid
    Peso molecular:379.43
  • Spiperone

    CAS:
    <p>Spiperone (Spiropitan) is a spiro butyrophenone analog similar to HALOPERIDOL and other related compounds.</p>
    Fórmula:C23H26FN3O2
    Pureza:99.34% - 99.91%
    Forma y color:Solid
    Peso molecular:395.47
  • Romergoline 2HCl


    <p>Romergoline 2HCl is a D1 agonist and D2 antagonist used in the study of Parkinson's disease.</p>
    Fórmula:C20H24Cl2N4O2
    Pureza:99.01% - 99.40%
    Forma y color:Soild
    Peso molecular:423.34
  • Haloperidol

    CAS:
    <p>Haloperidol (Serenace) is a highly potent neuroleptic by relieving nervous through the depression of nerve function.</p>
    Fórmula:C21H23ClFNO2
    Pureza:98.69% - 98.97%
    Forma y color:Crystals Solid
    Peso molecular:375.86
  • Risperidone

    CAS:
    <p>Risperidone (R 64 766) is a selective blocker of dopamine D2 receptors and serotonin 5-HT2 receptors that act as an atypical antipsychotic agent.</p>
    Fórmula:C23H27FN4O2
    Pureza:99.73%
    Forma y color:Crystalline Solid
    Peso molecular:410.48
  • UCM-1306

    CAS:
    <p>UCM-1306: an oral dopamine D1 receptor PAM; boosts DA efficacy, may enhance motor and cognitive function in PD.</p>
    Fórmula:C14H14FNO2S
    Pureza:99.98%
    Forma y color:Soild
    Peso molecular:279.33
  • ONC206

    CAS:
    <p>ONC206, an analogue of the TRAIL inducer ONC201, acts as a selective antagonist of the D2-like dopamine receptors (DRD2/3/4) at nanomolar concentrations and</p>
    Fórmula:C23H22F2N4O
    Pureza:99.38% - 99.81%
    Forma y color:Solid
    Peso molecular:408.44
  • Octodrine

    CAS:
    <p>Octodrine (2-Amino-6-methylheptane) is primarily used as a pharmaceutical intermediate for Octamylamine; it also functions as a local anesthetic and vasoconstrictor.</p>
    Fórmula:C8H19N
    Pureza:99.98%
    Forma y color:Clear Colorless To Light Yellow Liquid
    Peso molecular:129.24
  • D5R agonist 1


    <p>D5R Agonist 1 (Compound 5j) is a selective, orally active partial agonist of the D5 receptor that can penetrate the blood-brain barrier (EC50: 269.7 nM). It has been demonstrated to enhance cognitive abilities in a scopolamine-induced amnesia model.</p>
    Forma y color:Odour Solid
  • Losulazine

    CAS:
    <p>Losulazine: a new antihypertensive, requires functional sympathetic nervous system; mechanism undefined.</p>
    Fórmula:C27H22F4N4O3S
    Pureza:98.83%
    Forma y color:Solid
    Peso molecular:558.55
  • Fenoldopam

    CAS:
    <p>Fenoldopam is a selective D1-like dopamine receptor partial agonist (EC50 = 57 nM).</p>
    Fórmula:C16H16ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:305.76
  • Preclamol hydrochloride

    CAS:
    <p>Preclamol hydrochloride: selective dopamine agonist with research potential in schizophrenia.</p>
    Fórmula:C14H22ClNO
    Forma y color:Solid
    Peso molecular:255.78
  • (R)-Preclamol hydrochloride

    CAS:
    <p>(R)-Preclamol HCl is a dopamine agonist stimulating both auto and postsynaptic receptors.</p>
    Fórmula:C14H22ClNO
    Forma y color:Solid
    Peso molecular:255.78
  • Neurotransmitter Receptor Compound Library


    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening;</p>
    Forma y color:Odour Solid
  • (-)-GSK598809 hydrochloride

    CAS:
    <p>(-)-GSK598809 hydrochloride, a DRD3 selective antagonist, may correct reward deficits in substance dependence.</p>
    Fórmula:C22H24ClF4N5OS
    Pureza:98.36%
    Forma y color:Soild
    Peso molecular:517.97
  • 7-Hydroxy-PIPAT maleate

    CAS:
    <p>7-Hydroxy-PIPAT maleate is a D3R agonist.</p>
    Fórmula:C16H22INO
    Forma y color:Solid
    Peso molecular:371.262
  • Quinelorane

    CAS:
    <p>Quinelorane is dextrorotary isomer.</p>
    Fórmula:C14H22N4
    Forma y color:Solid
    Peso molecular:246.35
  • Fluphenazine free base

    CAS:
    <p>Flufenazine: antipsychotic for schizophrenia, blocks dopamine D2 receptors, reduces hallucinations and delusions.</p>
    Fórmula:C22H26F3N3OS
    Forma y color:Solid
    Peso molecular:437.52
  • Moperone

    CAS:
    <p>Moperone (R 1658) is an antagonist of both the D2 dopamine receptor (D2 dopamine receptor) and the D3 dopamine receptor (D3 dopamine receptor), with IC50 values for each of 1.0 nM.</p>
    Fórmula:C22H26FNO2
    Forma y color:Solid
    Peso molecular:355.45
  • Vanicoside E

    CAS:
    <p>Vanicoside E is an antioxidant and antitumor agent. Vanicoside E inhibits L-Tyrosine and L-DOPA with IC 50 s of 45.23 μM and 189.96 μM, respectively [1] [2] .</p>
    Fórmula:C53H52O22
    Forma y color:Solid
    Peso molecular:1040.97
  • Dopamine D2 receptor agonist-2

    CAS:
    <p>Dopamine D2 receptor agonist-2 (Dopamine D2 Receptor) is a ligand targeting the dopamine D2 receptor.</p>
    Fórmula:C25H31Cl2N5OS
    Pureza:98.93%
    Forma y color:Soild
    Peso molecular:520.52
  • ADTN hydrobromide

    CAS:
    <p>ADTN hydrobromide (6,7-ADTN) is a dopamine receptor agonist (EC50s = 3.5 and 0.65 μM in rat striatal and nucleus accumbens homogenates, respectively).</p>
    Fórmula:C10H14BrNO2
    Forma y color:Solid
    Peso molecular:260.13
  • MOR agonist-2


    <p>Compound 46, designated as MOR agonist-2, serves as a D3R antagonist and a MOR agonist with respective K i values of 7.26 nM and 564 nM.</p>
    Fórmula:C37H47Cl2N5O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:680.71
  • Clomipramine D3

    CAS:
    <p>Clomipramine D3 is deuterium-labeled Clomipramine, blocking serotonin, norepinephrine, dopamine transporters (Ki: 0.14, 54, 3 nM).</p>
    Fórmula:C19H23ClN2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:317.87
  • A 77636 hydrochloride

    CAS:
    <p>A 77636 hydrochloride is a potent, orally active, selective and long acting dopamine D1 receptor agonist (pKi=7.40; Ki=39.8 nM).</p>
    Fórmula:C20H28ClNO3
    Pureza:99.57%
    Forma y color:Solid
    Peso molecular:365.89
  • Adrogolide HCl

    CAS:
    <p>Adrogolide Hydrochloride is a selective dopamine receptor D1 agonist.</p>
    Fórmula:C22H26ClNO4S
    Forma y color:Solid
    Peso molecular:435.96
  • Amisulpride hydrochloride

    CAS:
    <p>Amisulpride is an antagonist of 5-HT7 receptor and dopamine D2 and D3 receptors. It modulates beta 2- arresting signaling and increases neurite outgrowth.</p>
    Fórmula:C17H28ClN3O4S
    Forma y color:Solid
    Peso molecular:405.94
  • DETQ

    CAS:
    <p>DETQ enhances human D1 dopamine receptor signaling, EC50=5.8 nM, less effective in rats/mice, inactive on D5.</p>
    Fórmula:C22H25Cl2NO3
    Forma y color:Solid
    Peso molecular:422.34
  • Neuromedin N

    CAS:
    <p>Neuromedin N is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct expression and effects.</p>
    Fórmula:C38H63N7O8
    Pureza:98%
    Forma y color:Solid
    Peso molecular:745.95
  • Cabergoline

    CAS:
    <p>Cabergoline (FCE-21336), an ergot-derived dopamine D2-like agonist, targets D2/D3/5-HT2B, normalizes prolactin, controls pituitary tumors.</p>
    Fórmula:C26H37N5O2
    Pureza:97.69% - 99.86%
    Forma y color:White Crystalline Solid
    Peso molecular:451.6
  • ABT 724 trihydrochloride

    CAS:
    <p>ABT-724 trihydrochloride: selective D4 agonist; EC50=12.4nM(human),14.3nM(rat),23.2nM(ferret); for erectile dysfunction research.</p>
    Fórmula:C17H22Cl3N5
    Pureza:99.91%
    Forma y color:Solid
    Peso molecular:402.75
  • LE 300

    CAS:
    <p>LE 300 represents a structurally novel type of antagonists acting preferentially at the dopamine D(1)/D(5)receptors and the serotonin 5-HT(2A)receptor.</p>
    Fórmula:C20H22N2
    Pureza:97.91% - 98.79%
    Forma y color:Solid
    Peso molecular:290.4
  • [18F]-Labeled L-dopa precursor

    CAS:
    <p>[18F]-Labeled L-dopa precursor is a precursor for synthesis of 18F-labeled L-dopa[1].</p>
    Fórmula:C35H36N2O7
    Forma y color:Solid
    Peso molecular:596.67
  • Secretoneurin, rat

    CAS:
    <p>Secretoneurin, rat, a 33-amino acid polypeptide, is generated by proteolytic processing of secretogranin II (SgII).</p>
    Fórmula:C159H252N40O58
    Pureza:98%
    Forma y color:Solid
    Peso molecular:3651.95
  • MLS1082

    CAS:
    <p>MLS1082 is a D1-like dopamine receptor (D1R) orthosteric modulatothat stimulates G-protein signaling upon dopamine activation for neurodegenerative disorders.</p>
    Fórmula:C24H23N3O2
    Pureza:99.53%
    Forma y color:Solid
    Peso molecular:385.46
  • D3R/MOR antagonist 1


    <p>Compound 114 (D3R/MOR antagonist 1) exhibits dual antagonistic activity at dopamine D3 receptors (D3R) and mu-opioid receptors (MOR), with K i values of 46.5 nM</p>
    Fórmula:C22H27Cl2N3O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:420.38
  • PF-4363467

    CAS:
    <p>PF-4363467 is a dopamine D3/D2 receptor antagonist that reduces opioid-seeking behavior without the side effects associated with D2 receptors. It has a Ki value of 3.1 nM for D3R and 692 nM for D2R.</p>
    Fórmula:C22H30N2O3S
    Forma y color:Solid
    Peso molecular:402.55
  • ADTN

    CAS:
    <p>ADTN is an agonist of the dopamine receptor.</p>
    Fórmula:C10H13NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:179.22
  • D3R ligand 1


    <p>D3R Ligand 1 (compound 23b) is a potent, selective antagonist of the dopamine D3 receptor (Ki=66 nM), incorporating a THPB template.</p>
    Fórmula:C27H37NO5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:455.59
  • D3R/MOR antagonist 2


    <p>Compound 121, a D3R/MOR antagonist with K i values of 361 nM and 85.2 nM for D3R and MOR respectively, has the potential for analgesic effects through MOR</p>
    Fórmula:C25H31ClN2O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.98
  • Haloperidol D4

    CAS:
    <p>Haloperidol D4 is deuterium-labeled haloperidol.</p>
    Fórmula:C21H23ClFNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:379.89
  • N-0500 HCl

    CAS:
    <p>N-0500 HCl, a potent DA receptor agonist, displaces [3H]DP_x005f_x0002_5,6-ADTN with an IC50 of 3nM.</p>
    Fórmula:C15H22ClNO2
    Pureza:98.85% - 99.54%
    Forma y color:Solid
    Peso molecular:283.79
  • O-2172

    CAS:
    <p>O-2172 is a carbocyclic analogue serving as an inhibitor of dopamine transporter (DAT), exhibiting IC50 values of 47 nM for DAT and 7000 nM for the serotonin transporter (SERT).</p>
    Fórmula:C14H16Cl2O2
    Forma y color:Solid
    Peso molecular:287.18
  • Trimethobenzamide

    CAS:
    <p>Trimethobenzamide (Ro 2-9578) is a D2 antagonist used to prevent nausea and vomiting.</p>
    Fórmula:C21H28N2O5
    Forma y color:Solid
    Peso molecular:388.46
  • ST-836 hydrochloride

    CAS:
    <p>ST-836 hydrochloride is a dopamine receptor ligand; Antiparkinsonian agent .</p>
    Fórmula:C23H35ClN4OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:451.07
  • Haloperidol (D4')

    CAS:
    <p>Haloperidol D4' is deuterium-labeled haloperidol. Haloperidol is a dopamine D2 receptor antagonist.</p>
    Fórmula:C21H23ClFNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:379.89
  • Eticlopride hydrochloride

    CAS:
    <p>Eticlopride, an antipsychotic, is a Selective dopamine D2/D3 receptor antagonist (Ki: 0.5/0.16 nM).</p>
    Fórmula:C17H25ClN2O3·HCl
    Pureza:98%
    Forma y color:Solid
    Peso molecular:377.31
  • Tiapride-d3


    <p>Tiapride-d3 is a deuterated form of Tiapride, a selective dopamine D2 receptor antagonist and an antipsychotic compound.</p>
    Fórmula:C15H21D3N2O4S
    Forma y color:Solid
    Peso molecular:331.45
  • Aramisulpride

    CAS:
    <p>Aramisulpride is a dual antagonist of the dopamine D2 receptor and serotonin receptor, primarily utilized for investigating metabolic disorders.</p>
    Fórmula:C17H27N3O4S
    Forma y color:Solid
    Peso molecular:369.48
  • SKF-82958 hydrobromide

    CAS:
    <p>SKF-82958 hydrobromide is a D1/D5 receptor full agonist.</p>
    Fórmula:C19H21BrClNO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:410.73
  • Clomipramine D3 hydrochloride

    CAS:
    <p>Clomipramine D3 hydrochloride is the deuterium-labeled Clomipramine. Clomipramine is a serotonin transporter, norepinephrine transporter dopamine transporter blocker (Ki: 0.14, 54 and 3 nM).</p>
    Fórmula:C19H24Cl2N2
    Forma y color:Solid
    Peso molecular:354.33
  • Docosahexaenoic acid ethyl ester

    CAS:
    <p>Docosahexaenoic acid ethyl ester (Ethyl docosahexaenoate) enhances 6-hydroxydopamine-induced neuronal damage by inducing lipid peroxidation in the mouse striatum, and can be used to study oxidative diseases of the retina or neurons.</p>
    Fórmula:C24H36O2
    Forma y color:Solid
    Peso molecular:356.54
  • Sumanirole maleate

    CAS:
    <p>Sumanirole maleate (PNU-95666E) is a D2 receptor full agonist with high selectivity that plays a vital role in Parkinson's disease and restless leg syndrome.</p>
    Fórmula:C15H17N3O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:319.31
  • Pramipexole dihydrochloride

    CAS:
    <p>Pramipexole dihydrochloride could be used to treat Parkinson disease.</p>
    Fórmula:C10H18ClN3S
    Pureza:98%
    Forma y color:White Crystalline Powder
    Peso molecular:247.79
  • cis-(Z)-Flupentixol dihydrochloride

    CAS:
    <p>cis-(Z)-Flupentixol dihydrochloride (Emergil) is a dopamine receptor antagonist.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.07%
    Forma y color:Solid
    Peso molecular:507.44
  • PD128907 HCl

    CAS:
    <p>PD128907 HCl is a potent and selective dopamine D3 receptor agonist, with EC50 of 0.64 nM, exhibits 53-fold selectivity over dopamine D2 receptor.</p>
    Fórmula:C14H20ClNO3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:285.77
  • UCSF924

    CAS:
    <p>UCSF924 is a potent and specific agonist of dopamine D4 receptor (DRD4) partial (EC50: 4.2 nM, Ki: 3 nM).</p>
    Fórmula:C20H22N2O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:322.4
  • (-)-Apomorphine hydrochloride hydrate

    CAS:
    <p>(-)-Apomorphine hydrochloride hydrate is a broad-spectrum dopamine agonist and ferroptosis inhibitor.</p>
    Fórmula:C17H17NO2HClXH2O
    Forma y color:Solid
    Peso molecular:303.8
  • ABT-724

    CAS:
    <p>ABT-724 is an agonist of dopamine D4 receptor(EC50: 12.4 nM)</p>
    Fórmula:C17H19N5
    Pureza:99.73%
    Forma y color:Solid
    Peso molecular:293.37
  • Clozapine N-Oxide

    CAS:
    <p>View and buy CLOZAPINE N-OXIDE from TargetMol.Clozapine N-oxide is a major metabolite of clozapine also known as DREADDs, technology to modulate synthetic receptors in vivo.Cited in 2 publications.</p>
    Fórmula:C18H19ClN4O
    Pureza:98.43% - 99.94%
    Forma y color:Solid
    Peso molecular:342.82
  • SKF-83566

    CAS:
    <p>SKF-83566: Blood-brain permeable, orally active D1 dopamine antagonist; weaker 5-HT2 antagonist, Ki=11 nM.</p>
    Fórmula:C17H18BrNO
    Pureza:95.00% - 99.82%
    Forma y color:Solid
    Peso molecular:332.23
  • Perospirone hydrochloride

    CAS:
    <p>Perospirone hydrochloride (Perospirone HCl) is an atypical antipsychotic agent for the treatment of schizophrenia.</p>
    Fórmula:C23H31ClN4O2S
    Pureza:99.37%
    Forma y color:White Solid
    Peso molecular:463
  • Alizapride hydrochloride

    CAS:
    <p>Alizapride hydrochloride (Alizapride HCl) is a dopamine receptor antagonist used for the treatment of nausea and vomiting.</p>
    Fórmula:C16H21N5O2·HCl
    Pureza:99.35% - 99.48%
    Forma y color:Coa
    Peso molecular:351.83
  • GBR 12935

    CAS:
    <p>GBR-12935: selective dopamine inhibitor, used in Parkinson's research.</p>
    Fórmula:C28H34N2O
    Forma y color:Solid
    Peso molecular:414.58
  • Raclopride tartrate

    CAS:
    <p>Raclopride is a selective antagonist on D2 dopamine receptor ( D2 Ki: 1.8 nm, D3 Ki: 3.5 nm, D4 Ki: 2400, D1 Ki: 18000 nM).</p>
    Fórmula:C19H26Cl2N2O9
    Forma y color:Solid
    Peso molecular:497.32
  • Bisacodyl

    CAS:
    <p>Bisacodyl (Fenilaxan) is a diphenylmethane stimulant laxative used for the treatment of constipation and for bowel evacuation.</p>
    Fórmula:C22H19NO4
    Pureza:99.45% - 99.78%
    Forma y color:Smaller Than 50 Microns Predominate White To Off-White Crystalline Powder
    Peso molecular:361.39
  • BisfluoroModafinil

    CAS:
    <p>CRL-40940 is a selective dopaminergic reuptake inhibitor</p>
    Fórmula:C15H13F2NO2S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:309.33
  • Nomifensine maleate

    CAS:
    <p>Nomifensine maleate (Nomifensine (maleate)) is a selective inhibitor of dopamine uptake. Nomifensine maleate is used in adult attention deficit disorder.</p>
    Fórmula:C20H22N2O4
    Pureza:98.46%
    Forma y color:Solid
    Peso molecular:354.4
  • OS-3-106

    CAS:
    <p>OS-3-106 is a novel arylamide phenylpiperazines, as partial agonists at the D3R in the adenylyl cyclase inhibition assay.</p>
    Fórmula:C25H30N4O2S
    Pureza:99.4% - 99.57%
    Forma y color:Solid
    Peso molecular:450.6
  • Glaucine

    CAS:
    <p>Glaucine: antitussive, antioxidative, antiviral, may fight arthritis, boosts IL-10, hinders breast cancer cell spread by inhibiting MMP-9 and NF-κB.</p>
    Fórmula:C21H25NO4
    Pureza:99.42% - 99.56%
    Forma y color:Solid
    Peso molecular:355.43
  • SCH-23390 hydrochloride

    CAS:
    <p>SCH-23390 hydrochloride (R-(+)-SCH23390 hydrochloride) is an effective dopamine receptor antagonist, and for the D1(Ki=0.2 nM) and D5(Ki=0.3 nM).</p>
    Fórmula:C17H19Cl2NO
    Pureza:98% - 99.83%
    Forma y color:Solid
    Peso molecular:324.24
  • Xaliproden hydrochloride

    CAS:
    <p>Xaliproden is a compound that mimics the effects of nerve growth factor and is also a serotonin 5-HT1A receptor agonist.</p>
    Fórmula:C24H23ClF3N
    Pureza:99.99%
    Forma y color:Solid
    Peso molecular:417.89
  • Butyrophenone

    CAS:
    <p>Butyrophenone (NSC-8463) is a chemical compound. Some of its derivatives are used to treat various psychiatric disorders.</p>
    Fórmula:C10H12O
    Pureza:99.84%
    Forma y color:Colourless To Yellow Liquid
    Peso molecular:148.2
  • 9-FLUORENOL

    CAS:
    <p>9-FLUORENOL is a dopamine reuptake inhibitor with IC50 of 9 μM, and a major metabolite of a compound developed as a wakefulness-promoting agent.</p>
    Fórmula:C13H10O
    Pureza:99.98%
    Forma y color:Off-White Crystalline Powder
    Peso molecular:182.22
  • NGB 2904

    CAS:
    <p>NGB 2904 is a potent and selective antagonist of dopamine D3 receptor. NGB2904 potently antagonizes mitogenesis stimulated by quinpirole (IC50 = 6.8 nM).</p>
    Fórmula:C28H29Cl2N3O
    Pureza:98.79%
    Forma y color:Solid
    Peso molecular:494.46
  • DOPEXAMINE

    CAS:
    <p>Dopexamine is a dopaminergic agonist</p>
    Fórmula:C22H32N2O2
    Pureza:99.42%
    Forma y color:Solid
    Peso molecular:356.5
  • PD-168077 maleate

    CAS:
    <p>PD-168077 maleate is a selective agonist of dopamine D4 receptor(Ki : 9 nM)</p>
    Fórmula:C24H26N4O5
    Pureza:99.13%
    Forma y color:Solid
    Peso molecular:450.49
  • ML417

    CAS:
    <p>ML417 is a selective and brain penetrant agonist of D3 Dopamine (EC50 : 38 nM).</p>
    Fórmula:C22H25N3O3
    Pureza:98.4% - 99.42%
    Forma y color:Solid
    Peso molecular:379.45
  • 3-CPMT

    CAS:
    <p>3-CPMT (FC-1) is a dopamine uptake inhibitor and a potent long-acting antihistaminic agent.</p>
    Fórmula:C21H25Cl2NO
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:378.33
  • A-381393

    CAS:
    <p>A-381393 is a selective and brain penetrate dopamine D4 receptor antagonist (Kis: 1.9/1.5/1.6 nM for human dopamine D4.2/D4.4/D4.7 receptor).</p>
    Fórmula:C20H24N4
    Pureza:99.00%
    Forma y color:Solid
    Peso molecular:320.43
  • GSK163090

    CAS:
    <p>GSK163090 is a specific and orally active 5-HT1A/B/D receptor antagonist (pKis: 9.4/8.5/9.7, and 6.3/6.7 for 5-HT1A/B/D, and dopamine D2/D3).</p>
    Fórmula:C25H29N5O
    Pureza:99.2%
    Forma y color:Solid
    Peso molecular:415.53
  • Bromocriptine mesylate

    CAS:
    <p>Bromocriptine mesylate (CB-154) is a potent dopamine receptor agonist that binds the D2 receptor with highest affinity (Ki = 2.5 nM)</p>
    Fórmula:C33H44BrN5O8S
    Pureza:99.85% - 99.96%
    Forma y color:White Solid
    Peso molecular:750.7
  • Nomifensine

    CAS:
    <p>Nomifensine ((±)-Nomifensin) is a norepinephrine-dopamine reuptake inhibitor that prevents dopamine reuptake into synaptosomes.</p>
    Fórmula:C16H18N2
    Pureza:99.83% - ≥95%
    Forma y color:Solid
    Peso molecular:238.33
  • Mesdopetam

    CAS:
    <p>Mesdopetam (IRL790), a D3 antagonist, has Ki=90 nM, IC50=9.8 μM, stabilizes psychomotors, used in Parkinson's research.</p>
    Fórmula:C12H18FNO3S
    Forma y color:Solid
    Peso molecular:275.34
  • Propionylpromazine hydrochloride

    CAS:
    <p>Propionylpromazine hydrochloride (Propiopromazine hydrochloride) is a dopamine receptor D2 (DRD2) antagonist.</p>
    Fórmula:C20H25ClN2OS
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:376.94
  • Fluoroclebopride

    CAS:
    <p>Fluoroclebopride is a dopamine (DA) D2 receptor ligand.</p>
    Fórmula:C20H23ClFN3O2
    Pureza:99.68% - 99.91%
    Forma y color:Solid
    Peso molecular:391.87
  • Ansofaxine hydrochloride

    CAS:
    <p>Ansofaxine hydrochloride (LY03005) is a serotonin-norepinephrine-dopamine reuptake inhibitor (IC50s: 723, 763 and 491 nM, respectively).</p>
    Fórmula:C24H32ClNO3
    Pureza:99.57% - 99.77%
    Forma y color:Solid
    Peso molecular:417.97
  • Cariprazine

    CAS:
    <p>Cariprazine (RGH-188) is a novel antipsychotic drug candidate that exhibits high affinity for the D3 (Ki=0.085 nM) and D2 (Ki=0.49 nM) receptors, and moderate</p>
    Fórmula:C21H32Cl2N4O
    Pureza:99.68% - 99.87%
    Forma y color:Solid
    Peso molecular:427.41
  • Chlorprothixene

    CAS:
    <p>Chlorprothixene (Truxal) is a typical antipsychotic drug of the thioxanthene class, which was the first of the series to be synthesized.</p>
    Fórmula:C18H18ClNS
    Pureza:98.77% - 99.756%
    Forma y color:Pale Yellow Crystals Solid
    Peso molecular:315.86
  • GSK 789472 hydrochloride

    CAS:
    <p>GSK 789472 hydrochloride is both a dopamine D3 receptor antagonist and a D2 partial agonist.</p>
    Fórmula:C15H22ClN3O
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:295.81
  • Veralipride

    CAS:
    <p>Veralipride ((±)-Veralipride) is an antagonist of D2 receptor.</p>
    Fórmula:C17H25N3O5S
    Pureza:99.65%
    Forma y color:Solid
    Peso molecular:383.46
  • Cariprazine hydrochloride

    CAS:
    <p>Cariprazine hydrochloride (RGH188 hydrochloride) is an antipsychotic drug, is a D3 and D2 receptor partial agonist((Ki of 0.085 nM and 0.49 nM, respectively)</p>
    Fórmula:C21H33Cl3N4O
    Pureza:99.78% - >99.99%
    Forma y color:Solid
    Peso molecular:463.87
  • Pridopidine

    CAS:
    <p>Pridopidine (FR310826), a low-affinity D2R antagonist, enhances motor skills and has neuroprotective effects in Huntington's R6/2 mice.</p>
    Fórmula:C15H23NO2S
    Pureza:95.2% - 99.89%
    Forma y color:Solid
    Peso molecular:281.41
  • D-tetrahydropalmatine

    CAS:
    <p>D-Tetrahydropalmatine inhibits OCT1, reducing MCT uptake and hepatocyte damage in MDCK-hOCT1 cells and rat livers.</p>
    Fórmula:C21H25NO4
    Pureza:99.34%
    Forma y color:Solid
    Peso molecular:355.43
  • Neuromedin N acetate(92169-45-4 free base)


    <p>Neuromedin N acetate(92169-45-4 free base) is a neuropeptide derived from the same precursor polypeptide as neurotensin, and with similar but subtly distinct</p>
    Fórmula:C40H67N7O10
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:805.9
  • Ocaperidone

    CAS:
    <p>Ocaperidona (Ocaperidone (Ocaperidona)), a very high affinity dopamine D2 antagonist.</p>
    Fórmula:C24H25FN4O2
    Pureza:99.33%
    Forma y color:Solid
    Peso molecular:420.48
  • Perospirone

    CAS:
    <p>Perospirone (Lullan) is an antagonist of serotonin 5HT2A receptors and dopamine D2 receptors.</p>
    Fórmula:C23H30N4O2S
    Pureza:99.23%
    Forma y color:White Powder
    Peso molecular:426.57
  • carfenazine

    CAS:
    <p>carfenazine targets the Dopamine receptor and is used for schizophrenia research.</p>
    Fórmula:C24H31N3O2S
    Pureza:98.06%
    Forma y color:Solid
    Peso molecular:425.59
  • Pergolide

    CAS:
    <p>Pergolide is a long-acting and orally active dopamine receptor D1/D2 agonist and ergoline derivative, used in the study of Parkinson's disease</p>
    Fórmula:C19H26N2S
    Pureza:99.95%
    Forma y color:Solid
    Peso molecular:314.49
  • Rotundine

    CAS:
    <p>Rotundine (Gindarine) (L-tetrahydropalmatine, L-THP) is a selective dopamine D1 receptor antagonist with IC50 of 166 nM.</p>
    Fórmula:C21H25NO4
    Pureza:99.8% - 99.91%
    Forma y color:Off-White Solid
    Peso molecular:355.43
  • Pergolide mesylate

    CAS:
    <p>Pergolide mesylate (LY127809), a dopamine agonist for Parkinson's and hyperprolactinemia, was withdrawn for heart valve risk.</p>
    Fórmula:C20H30N2O3S2
    Pureza:99.70%
    Forma y color:White To Off-White Solid
    Peso molecular:410.59
  • J-147

    CAS:
    <p>J-147, a curcumin derivative, is an experimental drug with reported effects against both Alzheimer's disease and ageing in mouse models of accelerated aging.</p>
    Fórmula:C18H17F3N2O2
    Pureza:99.61% - >99.99%
    Forma y color:Solid
    Peso molecular:350.33
  • Zotepine

    CAS:
    <p>Zotepine, an antipsychotic agent, is a potent antagonist of 5-HT2A, 5-HT2C, Histamine H1, α1-adrenergic, and Dopamine D2 receptors, with Kds of 2.6 nM, 3.2 nM,</p>
    Fórmula:C18H18ClNOS
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:331.86
  • Rotigotine-

    CAS:
    <p>Rotigotine (N-0923) is a non-ergot dopamine receptor agonist used in the therapy of Parkinson disease and restless leg syndrome.</p>
    Fórmula:C19H25NOS
    Pureza:98.08% - 99.59%
    Forma y color:Solid
    Peso molecular:315.47
  • Tavapadon

    CAS:
    <p>Tavapadon (CVL-751) is an orally active and highly selective dopamine D1/D5 receptor partial agonist.</p>
    Fórmula:C19H16F3N3O3
    Pureza:99.33% - 99.8%
    Forma y color:Solid
    Peso molecular:391.34
  • Ritanserin

    CAS:
    <p>Ritanserin (R 55667) is a long-acting, highly potent, relatively selective, orally bioavailable 5-HT2 receptor antagonist.Cost-effective and quality-assured.</p>
    Fórmula:C27H25F2N3OS
    Pureza:99.77% - 99.89%
    Forma y color:Solid
    Peso molecular:477.57
  • Vanoxerine dihydrochloride

    CAS:
    <p>Vanoxerine dihydrochloride (GBR-12909 dihydrochloride) is a potent inhibitor that blocks dopamine uptake (IC50 : 1-51 nM)</p>
    Fórmula:C28H34Cl2F2N2O
    Pureza:98.16% - 98.35%
    Forma y color:White Solid
    Peso molecular:523.49
  • Pramipexole dihydrochloride hydrate

    CAS:
    <p>Pramipexole dihydrochloride hydrate (Mirapex) is a selective, blood-brain barrier-crossing D2 dopamine receptor agonist, and is used in the study of PD.</p>
    Fórmula:C10H17N3S·2HCl·H2O
    Pureza:99.68%
    Forma y color:White To Off-White Crystalline Powder
    Peso molecular:302.26
  • Azaperone

    CAS:
    <p>Azaperone, a sedative and antiemetic veterinary tranquilizer, belongs to pyridinylpiperazine and butyrophenone classes.</p>
    Fórmula:C19H22FN3O
    Pureza:98.73%
    Forma y color:White Or Off-White Crystalline
    Peso molecular:327.4
  • SKF38393 hydrobromide

    CAS:
    <p>SKF38393 hydrobromide is the salt form of SKF38393.a dopamine D1 receptor agonist that increases the expression of Shati/Nat8L mRNA in the NAc of mice;</p>
    Fórmula:C16H18BrNO2
    Pureza:98.99%
    Forma y color:Solid
    Peso molecular:336.22
  • FAUC 346

    CAS:
    <p>FAUC 346 is a highly selective D3 partial agonist with EC50 of 1.5 nM.</p>
    Fórmula:C24H29N3O2S
    Pureza:99.46%
    Forma y color:Solid
    Peso molecular:423.57
  • Sultopride hydrochloride

    CAS:
    <p>Sultopride hydrochloride (LIN-1418 hydrochloride) is a selective dopamine D2 and D3 receptor antagonist.</p>
    Fórmula:C17H27ClN2O4S
    Pureza:≥95%
    Forma y color:White Or Yellowish Powder
    Peso molecular:390.93
  • Dasotraline

    CAS:
    <p>Dasotraline: a triple reuptake inhibitor targeting DA, NE, and 5-HT with IC50 values of 4, 6, 11 nM. Possible new antidepressant class.</p>
    Fórmula:C16H15Cl2N
    Forma y color:Solid
    Peso molecular:292.2
  • PD 168568

    CAS:
    <p>PD 168568: Oral DRD4 antagonist, selective over D2/D3, K_i - 8.8 nM. Used in GBM research.</p>
    Fórmula:C22H27N3O
    Forma y color:Solid
    Peso molecular:349.47
  • Alizapride

    CAS:
    <p>Alizapride is an antagonist of dopamine receptor. Alizapride can be used in human digestive disorders which is a potent antiemetic [1] [3].</p>
    Fórmula:C16H21N5O2
    Forma y color:Solid
    Peso molecular:315.37
  • BP 897

    CAS:
    <p>BP 897: potent selective dopamine D3 agonist, weak D2 antagonist. Ki: 0.92 nM (D3), 61 nM (D2), low affinity at D1/D4.</p>
    Fórmula:C26H31N3O2
    Pureza:99.44%
    Forma y color:Solid
    Peso molecular:417.54
  • Brexpiprazole

    CAS:
    <p>Brexpiprazole (OPC-34712) is a partial agonist of human 5-hydroxytryptamine (5-HT) 5-HT1A and dopamine D2 receptors.</p>
    Fórmula:C25H27N3O2S
    Pureza:99.06% - 99.96%
    Forma y color:Solid
    Peso molecular:433.57
  • JNJ-37822681

    CAS:
    <p>JNJ-37822681 is a novel, highly selective dopamine D₂ receptor antagonist characterized by a rapid dissociation rate from the dopamine D₂ receptor.</p>
    Fórmula:C17H17F5N4
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:372.34
  • Rotigotine Hydrochloride

    CAS:
    <p>Rotigotine HCl, D3-preferential dopamine agonist, is 50x stronger than quinpirole in anti-Parkinson's efficacy.</p>
    Fórmula:C19H26ClNOS
    Pureza:99.53% - 99.56%
    Forma y color:Almost White To White Crystalline Powder
    Peso molecular:351.93
  • Piribedil

    CAS:
    <p>Piribedil (Trivastan) is a dopamine D2 agonist, used in the treatment of Parkinson's disease.</p>
    Fórmula:C16H18N4O2
    Pureza:99.79% - 99.82%
    Forma y color:Solid
    Peso molecular:298.34
  • Haloperidol hydrochloride

    CAS:
    <p>Haloperidol hydrochloride is a potent dopamine D2 receptor antagonist which is a potent antipsychotic agent.</p>
    Fórmula:C21H24Cl2FNO2
    Forma y color:Solid
    Peso molecular:412.33
  • FAUC 213

    CAS:
    <p>FAUC 213 is a selective full antagonist of the dopamine D4 receptor.</p>
    Fórmula:C18H19ClN4
    Pureza:99.84%
    Forma y color:Solid
    Peso molecular:326.82
  • Metoclopramide

    CAS:
    <p>Metoclopramide: dopamine D2 antagonist, treats nausea, vomiting, gastroparesis, GERD; safe for pregnancy.</p>
    Fórmula:C14H22ClN3O2
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:299.80
  • Trimethobenzamide hydrochloride

    CAS:
    <p>Trimethobenzamide hydrochloride (Ro 2-9578) is a blocker of the D2 receptor. Trimethobenzamide is an antiemetic used to prevent nausea and vomiting.</p>
    Fórmula:C21H29ClN2O5
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:424.92
  • L-745870 trihydrochloride

    CAS:
    <p>L-745870 trihydrochloride is a highly potent and selective D4 dopamine receptor antagonist.</p>
    Fórmula:C18H22Cl4N4
    Pureza:97.52%
    Forma y color:Solid
    Peso molecular:436.21
  • Raclopride

    CAS:
    <p>Raclopride is a selective antagonist of dopamine D2/D3 receptor.</p>
    Fórmula:C15H20Cl2N2O3
    Pureza:99.17%
    Forma y color:Solid
    Peso molecular:347.24
  • Tiapride

    CAS:
    <p>Tiapride, an atypical neuroleptic, is a selective dopamine D2-receptor antagonist with varying IC50 values for D1-D4.</p>
    Fórmula:C15H24N2O4S
    Forma y color:Solid
    Peso molecular:328.43
  • Nuciferine

    CAS:
    <p>Nuciferine ((-)-Nuciferine) is an alkaloid found within the plants Nymphaea caerulea and Nelumbo nucifera.</p>
    Fórmula:C19H21NO2
    Pureza:98.76% - 99.79%
    Forma y color:Solid
    Peso molecular:295.38
  • L-DOPA methyl ester (hydrochloride)

    CAS:
    <p>L-DOPA methyl ester (LDME) is an agonist of dopamine D1 receptor.</p>
    Fórmula:C10H14ClNO4
    Pureza:98.69% - 99.81%
    Forma y color:White Solid
    Peso molecular:247.675
  • Zuclopenthixol dihydrochloride

    CAS:
    <p>Zuclopenthixol dihydrochloride is an D1 and D2 dopamine receptors antagonist.</p>
    Fórmula:C22H27Cl3N2OS
    Pureza:98%
    Forma y color:Solid
    Peso molecular:473.89
  • AHN 1-055 hydrochloride

    CAS:
    <p>AHN 1-055 hydrochloride (3α-Bis-(4-fluorophenyl) Methoxytropane hydrochloride) is an inhibitor of dopamine transporter (DAT) and dopamine uptake(IC50 = 71 nM).</p>
    Fórmula:C21H24ClF2NO
    Pureza:99.89%
    Forma y color:Solid
    Peso molecular:379.87
  • L-745870 hydrochloride

    CAS:
    <p>L-745870 hydrochloride has excellent brain penetration. L-745870 hydrochloride is a high-affinity, selective and orally active human dopamine D4 receptor</p>
    Fórmula:C18H20Cl2N4
    Pureza:97.36%
    Forma y color:Solid
    Peso molecular:363.28
  • FAUC-365

    CAS:
    <p>FAUC-365 is a D3 dopamine receptor agonist.</p>
    Fórmula:C23H25Cl2N3OS
    Pureza:99.62%
    Forma y color:Solid
    Peso molecular:462.44
  • Lurasidone

    CAS:
    <p>Lurasidone (SM-13496) is an antagonist of both dopamine D2 and 5-HT7(IC50=1.68 and 0.495 nM, respectively).It also a partial agonist of 5-HT1A receptor(IC50 : 6</p>
    Fórmula:C28H36N4O2S
    Pureza:99.78% - 99.91%
    Forma y color:Solid
    Peso molecular:492.68
  • Metergoline

    CAS:
    <p>Metergoline (Methergoline) is a dopamine agonist and serotonin antagonist.</p>
    Fórmula:C25H29N3O2
    Pureza:99.83% - 99.97%
    Forma y color:Solid
    Peso molecular:403.52
  • (+)-PD 128907 hydrochloride

    CAS:
    <p>(+)-PD 128907 hydrochloride is an agonist of D3 dopamine receptor .</p>
    Fórmula:C14H20ClNO3
    Pureza:97.76%
    Forma y color:Solid
    Peso molecular:285.77
  • Mesdopetam hemitartrate

    CAS:
    <p>Mesdopetam hemitartrate antagonizes dopamine D3 receptor (Ki=90 nM; IC50=9.8 μM) and stabilizes psychomotor function.</p>
    Fórmula:C28H42F2N2O12S2
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:700.77
  • WAY-100635 Monomaleate

    CAS:
    <p>WAY-100635 maleate is a selective 5-hydroxytryptamine 1A receptor antagonist with an IC50 value of 0.91 nM and a Ki value of 0.39 nM.</p>
    Fórmula:C25H34N4O2·C4H4O4
    Pureza:98.44% - 99.46%
    Forma y color:Solid
    Peso molecular:538.64
  • Sertindole

    CAS:
    <p>Sertindole, atypical antipsychotic, targets D2, 5-HT1D, 5-HT2A, 5-HT2C receptors (Kds: 2.7, 20, 0.14, 6 nM).</p>
    Fórmula:C24H26ClFN4O
    Pureza:99.87% - 99.92%
    Forma y color:Off-White To Pale Yellow Solid
    Peso molecular:440.94
  • Clebopride malate

    CAS:
    <p>Clebopride malate is a dopamine antagonist drug Used to treat functional gastrointestinal disorders such as nausea or vomiting.</p>
    Fórmula:C24H30ClN3O7
    Pureza:99.52%
    Forma y color:Solid
    Peso molecular:507.96
  • Fenoldopam mesylate

    CAS:
    <p>Fenoldopam mesylate (Corlopam mesylate) is a selective dopamine-1 receptor (DA1) agonist with natriuretic/diuretic properties.</p>
    Fórmula:C16H16ClNO3·CH4O3S
    Pureza:99.19%
    Forma y color:Solid
    Peso molecular:401.86
  • Flupentixol dihydrochloride

    CAS:
    <p>Flupentixol dihydrochloride is used in therapy of schizophrenia as well as in anxiolytic and depressive disorders.</p>
    Fórmula:C23H27Cl2F3N2OS
    Pureza:98.76% - >99.99%
    Forma y color:White Or Off-White Solid
    Peso molecular:507.43
  • GBR 12935 dihydrochloride

    CAS:
    <p>GBR 12935 dihydrochloride (GBR 12935) can induce the increase of the extracellular levels of dopamine to basal levels.</p>
    Fórmula:C28H36Cl2N2O
    Pureza:99.09% - ≥95%
    Forma y color:Solid
    Peso molecular:487.5
  • Decynium 22

    CAS:
    <p>Decynium 22 is a plasma membrane monoamine transporter (PMAT) inhibitor</p>
    Fórmula:C23H23IN2
    Pureza:99.92%
    Forma y color:Dark Red Crystals
    Peso molecular:454.35
  • Domperidone monomaleate

    CAS:
    <p>Domperidone monomaleate, a selective oral dopamine-2 antagonist, aids gastric motility and has antiemetic properties.</p>
    Fórmula:C26H28ClN5O6
    Forma y color:Solid
    Peso molecular:541.98
  • Tetrahydropalmatine hydrochloride

    CAS:
    <p>Tetrahydropalmatine HCl (Gindarine) is a muscle relaxant alkaloid from Corydalis plants.</p>
    Fórmula:C21H26ClNO4
    Pureza:98% - 99.59%
    Forma y color:Solid
    Peso molecular:391.888
  • Fluphenazine decanoate

    CAS:
    <p>Fluphenazine decanoate is dopamine D2 receptor blocke,and is a long-acting phenothiazine neuroleptic that used to treat schizophrenia.</p>
    Fórmula:C32H44F3N3O2S
    Pureza:98.14%
    Forma y color:Solid
    Peso molecular:591.77