Receptor de adenosina
Los receptores de adenosina son una clase de GPCR que responden al nucleósido endógeno adenosina. Estos receptores están involucrados en la regulación de diversos procesos fisiológicos, incluidos la función cardiovascular, los ciclos sueño-vigilia y las respuestas inmunitarias. Los moduladores de los receptores de adenosina tienen un potencial terapéutico en el tratamiento de afecciones como las arritmias cardíacas, la inflamación y las enfermedades neurodegenerativas. En CymitQuimica, ofrecemos una selección de moduladores de receptores de adenosina de alta calidad para apoyar su investigación en biología cardiovascular, neurociencia e inmunología.
Se han encontrado 242 productos de "Receptor de adenosina"
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Amp579 TFA
<p>Amp579 TFA is a novel adenosine A1/A2a receptor agonist that induces acute and delayed preconditioning against myocardial shock in vivo.</p>Fórmula:C24H29ClF3N5O5SPureza:96.56%Forma y color:SoildPeso molecular:592.03Pamabrom
CAS:<p>Pamabrom is a diuretic for premenstrual and menstrual bloating, swelling, and fullness.</p>Fórmula:C11H18BrN5O3Pureza:99.84% - >99.99%Forma y color:CoaPeso molecular:348.2Adenosine 5'-monophosphate monohydrate
CAS:<p>Adenosine 5'-monophosphate monohydrate (5'-AMP) , also known as 5'-adenylic acid, is a nucleotide that is used as a monomer in RNA.</p>Fórmula:C10H14N5O7P·H2OPureza:97.68% - 98.49%Forma y color:White PowderPeso molecular:365.24Ticlopidine hydrochloride
CAS:<p>Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.</p>Fórmula:C14H15Cl2NSPureza:99.85% - >99.99%Forma y color:White PowderPeso molecular:300.25Quercetin-3'-o-phosphate TEA
<p>Quercetin-3'-o-phosphate TEA (Quercetin 3'-phosphate TEA) is an adenosine A receptor antagonist that can be used to prevent and treat metabolic disorders.</p>Fórmula:C21H26NO10PPureza:95.63%Forma y color:SoildPeso molecular:483.41AB928
CAS:<p>AB928 is an orally bioavailable, selective dual adenosine receptor (A2aR/A2bR) antagonist. It has immunomodulatory activity[1].</p>Fórmula:C23H22N8OPureza:98.09% - >99.99%Forma y color:SolidPeso molecular:426.47Pentoxifylline
CAS:<p>Pentoxifylline (PTX) stimulates cytokines, inhibits phosphodiesterase, enhances blood flow, and increases cell flexibility.</p>Fórmula:C13H18N4O3Pureza:99.26% - 99.93%Forma y color:SolidPeso molecular:278.31Diphylline
CAS:<p>Diphylline is a bronchodilator with mild vasodilator and diuretic properties, used for asthma, bronchitis, and emphysema.</p>Fórmula:C10H14N4O4Pureza:98.54%Forma y color:Crystals From Alcohol SolidPeso molecular:254.24Doxofylline
CAS:<p>Doxofylline (Doxophylline) is a methylxanthine derivative with the presence of a dioxolane group in position 7.</p>Fórmula:C11H14N4O4Pureza:99.958% - >99.99%Forma y color:SolidPeso molecular:266.25Theophylline
CAS:<p>Theophylline (1,3-Dimethylxanthine) is a methyl xanthine derivative from tea with diuretic, smooth muscle relaxant, bronchial dilation, cardiac and central</p>Fórmula:C7H8N4O2Pureza:99.65% - 99.98%Forma y color:White Solid PowderPeso molecular:180.16DPTN dihydrochloride
CAS:<p>DPTN dihydrochloride is a potent and selective A3AR antagonist with Ki values of 1.65, 9.61 and 8.53 nM in human, mouse and rat, respectively.</p>Fórmula:C22H20Cl2N4OSPureza:99.95%Forma y color:SoildPeso molecular:459.39Adenosine A1 receptor activator T62
CAS:<p>Adenosine A1 receptor activator T62 is an allosteric enhancer of adenosine A1 receptor, and it produces antinociception in animal models of acute pain and also</p>Fórmula:C15H14ClNOSPureza:97.83%Forma y color:SolidPeso molecular:291.8YT 146
CAS:<p>YT 146 is a biochemical.</p>Fórmula:C18H25N5O4Pureza:98.81% - 99.25%Forma y color:SolidPeso molecular:375.42Theophylline monohydrate
CAS:<p>Theophylline monohydrate (Quibron) appears to inhibit phosphodiesterase and prostaglandin production, regulate calcium flux and intracellular calcium</p>Fórmula:C7H8N4O2·H2OPureza:99.78%Forma y color:SolidPeso molecular:198.18Aminophylline
CAS:<p>Aminophylline (Phyllocontin) is a competitive nonselective phosphodiesterase inhibitor giving a bronchodilatory effect.</p>Fórmula:C7H8O2·C2H8N2Pureza:99.31%Forma y color:White Or Slightly Yellowish Granules Or Powder SolidPeso molecular:420.43N6-Ethyladenosine
CAS:<p>N6-Ethyladenosine is an adenosine derivative, acts as an agonist of Adenosine receptor(hA1AR and hA3AR with Kis of 4.9 and 4.7 nM , respectively).</p>Fórmula:C12H17N5O4Pureza:99.96%Forma y color:SolidPeso molecular:295.29Acefylline
CAS:<p>Acefylline (Theophylline-7-acetic acid), a stimulant drug of the xanthine chemical class, acts as an adenosine receptor antagonist.</p>Fórmula:C9H10N4O4Pureza:99.57%Forma y color:White Crystalline SolidPeso molecular:238.2CGS 15943
CAS:<p>CGS 15943 is an orally bioavailable non-xanthine antagonist of Adenosine Receptor.</p>Fórmula:C13H8ClN5OPureza:97.4%Forma y color:SolidPeso molecular:285.69N6-Cyclohexyladenosine
CAS:<p>N6-Cyclohexyladenosine (CHA) is a selective agonist of A1 receptor with EC50 of 8.2 Nm.</p>Fórmula:C16H23N5O4Pureza:99.84% - 99.98%Forma y color:SolidPeso molecular:349.38A3AR agonist 2
<p>Compound 19, a selective A3 Adenosine Receptor (A3AR) agonist (K i : 22.1 nM), effectively stimulates β-arrestin2 recruitment with an EC 50 value of 4.36 nM.</p>Fórmula:C34H34N6O6Pureza:98%Forma y color:SolidPeso molecular:622.67Adenosine receptor agonist 1
<p>Compound 6m, an A3 adenosine receptor (AR) partial agonist, exhibits a K i value of 6.7 nM as an adenosine receptor agonist.</p>Fórmula:C12H14ClN5O2SeForma y color:SolidPeso molecular:374.68hA3AR agonist 2
<p>hA3AR agonist 2 is a potent activator of A3AR, with a Ki value of 3.5 nM.</p>Fórmula:C11H14ClN5O2SForma y color:SolidPeso molecular:315.78Xanthine amine congener dihydrochloride
CAS:<p>XAC dihydrochloride is an Adenosine A1 and A2 receptor antagonist with IC50s of 1.8 nM and 114 nM, also a mouse convulsant.</p>Fórmula:C21H30Cl2N6O4Forma y color:SolidPeso molecular:501.41Heterobivalent ligand-1
<p>Heterobivalent ligand-1 targets A2A-D2 receptor heteromer with affinity: Kd for A2A=2.1 nM, D2=0.13 nM.</p>Fórmula:C86H115FN16O21Forma y color:SolidPeso molecular:1727.93LUF6096
CAS:<p>LUF6096 (CF-602) is a potent allosteric enhancer of the adenosine A3 receptor, exhibiting the capability to enhance agonist binding allosterically while</p>Fórmula:C22H21Cl2N3OPureza:99.5%Forma y color:SolidPeso molecular:414.33ABT-702
CAS:<p>ABT-702 is an orally active, competitive, and reversible non-nucleoside adenosine kinase (AK) inhibitor analgesic and anti-inflammatory.</p>Fórmula:C22H19BrN6OPureza:99.57%Forma y color:SoildPeso molecular:463.33Apadenoson TFA
<p>Apadenoson TFA is a potent adenosine A2A receptor (A2AR) agonist that can be used to improve survival in patients infected with SARS.</p>Fórmula:C25H31F3N6O8Pureza:98.08%Forma y color:SoildPeso molecular:600.558-Chloro caffeine
CAS:<p>8-Chloro caffeine binds to adenosine receptors with a Ki of 30 µM. It enhances UV-induced chromosomal aberrations in the Cl-I type Chinese hamster embryo lung cells. 8-Chloro caffeine is a derivative of the methylxanthine alkaloid caffeine.</p>Fórmula:C8H9ClN4O2Forma y color:SolidPeso molecular:228.64PSB 0777 ammonium hydrate
<p>PSB 0777 ammonium hydrate is a potent and selective adenosine A2A receptor full agonist, exhibiting K i values of 44.4 nM for rat A2A receptors and 360 nM for</p>Fórmula:C18H20N5O7S2·NH4·75H2OPureza:98%Forma y color:SolidPeso molecular:532.09A3AR agonist 1
<p>A3AR Agonist 1 (Compound 12), with a Ki of 25.8 nM, is a potent A3 adenosine receptor (A3AR) agonist that promotes β-arrestin2 recruitment with an effective</p>Fórmula:C28H34N6O6Pureza:98%Forma y color:SolidPeso molecular:550.61AR ligand 40
<p>AR ligand 40 (compound 19c) is an Adenosine A1 Receptor ligand with antagonistic activity. It exhibits antiproliferative effects on SW480, SW48, HCT116, K562, MDA-MB-231, and A549 cells, with EC50 values of 7, 10, 12, 13, 15, and 39 μM, respectively.</p>Fórmula:C21H25N5Forma y color:SolidPeso molecular:347.211PSB 0777 ammonium salt
CAS:<p>adenosine A2A receptor full agonist</p>Fórmula:C18H24N6O7S2Pureza:98%Forma y color:SolidPeso molecular:500.55MRS-1706
CAS:<p>MRS-1706: Ki of 1.39nM for A2B; selective inverse agonist; also affects A2A, A1, A3.</p>Fórmula:C27H29N5O5Pureza:99.00%Forma y color:SolidPeso molecular:503.55N6-Benzyl-5'-ethylcarboxamido adenosine
CAS:<p>N6-Benzyl-5'-ethylcarboxamido adenosine is a selective A3 adenosine receptor agonist.</p>Fórmula:C19H22N6O4Forma y color:SolidPeso molecular:398.42Norisoboldine hydrochloride
CAS:<p>Norisoboldine hydrochloride: an oral AhR agonist from Radix Linderae, for Rheumatoid arthritis and Ulcerative colitis research.</p>Fórmula:C18H20ClNO4Forma y color:SolidPeso molecular:349.81FSCPX
CAS:<p>FSCPX is a potent and selective irreversible antagonist of the A1 adenosine receptor (A1AR), exhibiting low nanomolar binding potency.</p>Fórmula:C23H27FN4O6SPureza:98%Forma y color:SolidPeso molecular:506.55Xanthine amine congener trihydrochloride
CAS:<p>Xanthine amine congener trihydrochloride: potent adenosine antagonist, reverses effects of N6-cyclohexyladenosine on urine, sodium excretion, heart rate.</p>Fórmula:C21H29ClN6O4Pureza:98.81%Forma y color:SolidPeso molecular:464.95Danshenol B
<p>Danshenol B is a natural product that can be used as a reference standard.</p>Fórmula:C22H26O4Forma y color:SolidPeso molecular:354.4463F6-9G5
<p>3F6-9G5 is a humanized monoclonal antibody targeting AA2AR/Adenosine A2aR, used in neurodegenerative disease research.</p>Pureza:>95%Forma y color:Odour LiquidTheophyllol
CAS:<p>Theophyllol (theophylline sodium acetate) can alter calcium levels in subcellular fractions of rat brain cortex.</p>Fórmula:C9H10N4Na2O4Forma y color:SolidPeso molecular:284.18Adenosine receptor antagonist 1
CAS:<p>A2aR-selective antagonist with IC50 of 0.29 nM; 14x more selective over A2bR.</p>Fórmula:C22H15ClFN7OForma y color:SolidPeso molecular:447.86LUF7690
CAS:<p>LUF7690 (Compound 9), a clickable and covalent affinity-based probe (AfBP) for the human A3 adenosine receptor (hA3AR), facilitates the detection and</p>Fórmula:C25H24FN5O6SForma y color:SolidPeso molecular:541.55A3AR modulator 1
<p>MRS8054 is an oral A3 adenosine receptor positive allosteric modulator, enhancing Cl-IB-MECA-induced activity.</p>Fórmula:C23H25IN4Forma y color:SolidPeso molecular:484.38A-286501
CAS:<p>A-286501: Oral adenosine kinase inhibitor, IC50=0.47 nM, reduces pain via non-opioid, non-NSAID ADO receptors.</p>Fórmula:C11H14BrN5O2Pureza:98%Forma y color:SolidPeso molecular:328.17GW-328267
CAS:<p>GW-328267 is an agonist of the adenosine A2 receptor.</p>Fórmula:C21H26N10O4Forma y color:SolidPeso molecular:482.5A2A/A3 AR antagonist-1
<p>A2A/A3 AR antagonist-1 is a dual fluorescent AR ligand with K i of 90 nM (hA2A) & 31.8 nM (hA3).</p>Fórmula:C56H71N15O12S2Forma y color:SolidPeso molecular:1210.39LAS101057
CAS:<p>LAS101057 is a novel orally available and potent and selective A2B receptor antagonist for the study of asthma.</p>Fórmula:C18H14FN5OPureza:99.03% - >99.99%Forma y color:SolidPeso molecular:335.34(Rac)-Mirabegron-d5
CAS:<p>(Rac)-Mirabegron D5 is a deuterium labeled (Rac)-Mirabegron. Mirabegron is a selective agonist of β3-adrenoceptor.</p>Fórmula:C21H24N4O2SPureza:98%Forma y color:SolidPeso molecular:401.54GR79236
CAS:<p>GR79236 is an effective and selective adenosine A1 receptor agonist (Ki: 3.1 nM) that has analgesic and anti-inflammatory actions.</p>Fórmula:C15H21N5O5Forma y color:SolidPeso molecular:351.36MRS-3777 hemioxalate
CAS:<p>MRS-3777 hemioxalate, a selective adenosine A3 receptor antagonist, reverses the anti-injury perception effects of its corresponding agonist and serves as a valuable tool for studying inflammatory pain.</p>Fórmula:C17H19N5OC2H2O4Pureza:97.10%Forma y color:SolidPeso molecular:354.39
