Receptor de adenosina
Los receptores de adenosina son una clase de GPCR que responden al nucleósido endógeno adenosina. Estos receptores están involucrados en la regulación de diversos procesos fisiológicos, incluidos la función cardiovascular, los ciclos sueño-vigilia y las respuestas inmunitarias. Los moduladores de los receptores de adenosina tienen un potencial terapéutico en el tratamiento de afecciones como las arritmias cardíacas, la inflamación y las enfermedades neurodegenerativas. En CymitQuimica, ofrecemos una selección de moduladores de receptores de adenosina de alta calidad para apoyar su investigación en biología cardiovascular, neurociencia e inmunología.
Se han encontrado 249 productos de "Receptor de adenosina"
Ordenar por
Pureza (%)
0
100
|
0
|
50
|
90
|
95
|
100
Trabodenoson
CAS:<p>Trabodenoson (INO-8875) is a selective and potent adenosine A1 receptor agonist, an adenosine analog, for the study of primary open-angle glaucoma.</p>Fórmula:C15H20N6O6Pureza:99.94%Forma y color:SolidPeso molecular:380.36Theobromine
CAS:Theobromine (3,7-Dimethylxanthine), a xanthine alkaloid, is used as a bronchodilator and as a vasodilator.Fórmula:C7H8N4O2Pureza:99.69% - 99.91%Forma y color:White To Yellow Crystalline PowderPeso molecular:180.165'-Amino-5'-deoxyadenosine
CAS:<p>5'-Amino-5'-deoxyadenosine (NH2dAdo) is an adenosine kinase inhibitor targeting malignant tumors of the inert lymphatic system with antitumor and anticancer</p>Fórmula:C10H14N6O3Pureza:95.55%Forma y color:SolidPeso molecular:266.26Blontuvetmab
CAS:Blontuvetmab (AT 004), a caninized CD20 monoclonal antibody, is utilized in the study of Canine B-cell lymphoma [1].Forma y color:LiquidAdenosine receptor inhibitor 1
CAS:Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.Fórmula:C17H19ClFN5O3Forma y color:SolidPeso molecular:395.82A1AR antagonist 2
CAS:Compound 18h is a potent A1 adenosine receptor blocker with Ki of 1.49 nM for hA1, 10.2 nM for hA2A, 50.1 nM for hA2B.Fórmula:C17H12N4OForma y color:SolidPeso molecular:288.3TC-G 1004
CAS:adenosine A2A receptors antagonistFórmula:C22H27N7O2Pureza:98%Forma y color:SolidPeso molecular:421.5SCH-202676 HBr
CAS:SCH-202676 HBr is an allosteric agonist. It also an GPCR antagonist.Fórmula:C15H13N3SPureza:98%Forma y color:SolidPeso molecular:267.35A2AR-agonist-1
CAS:<p>A2AR-agonist-1 targets A2A Receptor/ENT1 for neuroprotection; potent with Ki of 4.39 (A2AR), 3.47 (ENT1).</p>Fórmula:C20H22N6O4Pureza:99.9%Forma y color:SolidPeso molecular:410.43Lu AA 47070
CAS:adenosine A2A receptor antagonistFórmula:C17H20F2N3O6PSPureza:98%Forma y color:SolidPeso molecular:463.39VUF8507
CAS:Vuf8507 is an allosteric regulator of adenosine receptor.Fórmula:C21H15N3OForma y color:SolidPeso molecular:325.36Acefylline piperazine
CAS:Acefylline piperazine, a less toxic theophylline derivative, treats asthma and bronchitis by bronchodilation, stimulating respiration and CNS.Fórmula:C9H10N4O4·xC4H10N2Forma y color:SolidPeso molecular:562.54CAY10498
CAS:A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.Fórmula:C18H20N6Forma y color:SolidPeso molecular:320.39Apadenoson
CAS:<p>Apadenoson: potent A2 agonist, A3 inhibitor (IC 45 nM), anti-inflammatory, for neurological research.</p>Fórmula:C23H30N6O6Pureza:98%Forma y color:SolidPeso molecular:486.52CVT-2759
CAS:CVT-2759, potential A(1)-ADOR partial agonist, could slow ventricular rate without severe cardiac side effects.Fórmula:C17H24N6O6Forma y color:SolidPeso molecular:408.41MRS-1191
CAS:MRS-1191 is an effective and selective A3 adenosine receptor antagonist (KB: 92 nM, a Ki: 31.4 nM for human A3 receptor and an IC50: 120 nM for CHO cells).Fórmula:C31H27NO4Forma y color:SolidPeso molecular:477.55PD 81723
CAS:Allosteric potentiator at the adenosine A1 receptorFórmula:C14H12F3NOSPureza:98%Forma y color:SolidPeso molecular:299.31Sipagladenant
CAS:Sipagladenant: oral inverse agonist for A2A adenosine receptor, may aid frontal lobe dysfunction research.Fórmula:C20H19N3O4SForma y color:SolidPeso molecular:397.45Adenosine receptor inhibitor 2
CAS:Compound 14b is a potent AR inhibitor with dual affinity, stronger for A1 (Ki = 52.2 nM) than A2A (Ki = 167 nM) ARs.Fórmula:C17H20BrN5O2Forma y color:SolidPeso molecular:406.28Inupadenant
CAS:Inupadenant is an orally active, highly selective A2A receptor antagonist. Inupadenant is not brain-penetrant. Inupadenant has potent anti-tumor activity[1].Fórmula:C25H26F2N8O4S2Forma y color:SolidPeso molecular:604.65
