
Receptor de adenosina
Los receptores de adenosina son una clase de GPCR que responden al nucleósido endógeno adenosina. Estos receptores están involucrados en la regulación de diversos procesos fisiológicos, incluidos la función cardiovascular, los ciclos sueño-vigilia y las respuestas inmunitarias. Los moduladores de los receptores de adenosina tienen un potencial terapéutico en el tratamiento de afecciones como las arritmias cardíacas, la inflamación y las enfermedades neurodegenerativas. En CymitQuimica, ofrecemos una selección de moduladores de receptores de adenosina de alta calidad para apoyar su investigación en biología cardiovascular, neurociencia e inmunología.
Se han encontrado 242 productos de "Receptor de adenosina"
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Adenosine receptor inhibitor 1
CAS:<p>Potent, selective adenosine receptor blocker with strong affinity, especially A2A (Ki 68.5 nM). Promising for cancer, neurodegeneration study.</p>Fórmula:C17H19ClFN5O3Forma y color:SolidPeso molecular:395.82A1/A3 AR antagonist 2
CAS:<p>The compound is an a1/a3 adenosine receptor antagonist, which helps to treat (neurological) inflammatory diseases.</p>Fórmula:C22H16N2O3SForma y color:SolidPeso molecular:388.44AB-MECA
CAS:<p>AB-MECA is a high affinity A3 adenosine receptor agonist. It has high affinity for recombinant A1 and A3 receptors.</p>Fórmula:C18H21N7O4Pureza:98%Forma y color:SolidPeso molecular:399.4A2AAR/HDAC-IN-1
CAS:<p>A2AAR/HDAC-IN-1 (compound 14c) is an orally active, balanced A2AAR/HDAC dual inhibitor of A2AAR (Ki: 163.5 nM), HDAC1 (IC50: 145.3 nM). effect.</p>Fórmula:C24H21N7O2Forma y color:SolidPeso molecular:439.47LASSBio-1359
CAS:<p>LASSBio-1359 is an adenosine receptor agonist. It acts by inducing relaxation of the corpus cavernosum. It also acts as a novel selective phosphodiesterase.</p>Fórmula:C17H18N2O3Pureza:98%Forma y color:SolidPeso molecular:298.34PSB 11 hydrochloride
CAS:<p>PSB 11 hydrochloride is a human adenosine A3 receptor antagonist.</p>Fórmula:C16H18ClN5OPureza:98%Forma y color:SolidPeso molecular:331.8Adenosine receptor antagonist 3
CAS:<p>Adenosine receptor antagonist 3 has the potential for cancer disease research which is a potent adenosine receptor antagonist [1].</p>Fórmula:C16H14N6SForma y color:SolidPeso molecular:322.39Adentri
CAS:<p>Adentri is a novel antagonist of adenosine A1 receptor with unique diuretic activity.</p>Fórmula:C18H24N4O3Pureza:98%Forma y color:SolidPeso molecular:344.41A2A receptor antagonist 3
CAS:<p>A2A receptor antagonist 3 (Example 92) is an adenosine A2a receptor antagonist (Ki: 0.4 nM). receptor (Ki: 1467 nM).</p>Fórmula:C26H26N6O2Forma y color:SolidPeso molecular:454.52MRS1186
CAS:<p>MRS1186 is an effective and selective antagonist of the human Adenosine A3 receptor (Ki: 7.66 nM).</p>Fórmula:C16H12ClN5O2Pureza:98%Forma y color:SolidPeso molecular:341.75Adenosine receptor A1 antagonist 5
CAS:<p>1,3-Dipropyl-8-phenylxanthine is an adenosine antagonist, oxypurine, insecticide, and reduces high blood pressure.</p>Fórmula:C17H20N4O2Pureza:99.97%Forma y color:SolidPeso molecular:312.37MRS1177
CAS:<p>MRS1177 is an effective and selective antagonist of the human Adenosine A3 receptor (hA3AR) (Ki: 0.3 nM).</p>Fórmula:C20H12ClN5O2Pureza:98%Forma y color:SolidPeso molecular:389.79XU1
CAS:<p>XU1(Benzo[c][1,8]naphthyridin-6(5h)-One) is an Aurora protein kinase inhibitor used for the treatment of diseases suitable for inhibition, regulation or</p>Fórmula:C12H8N2OPureza:98.58% - 99.59%Forma y color:SolidPeso molecular:196.2HEMADO
CAS:<p>HEMADO is a potent and selective agonist of adenosine A3 receptor (Ki: 1.1 nM at the human A3 subtype).</p>Fórmula:C17H23N5O4Pureza:98%Forma y color:SolidPeso molecular:361.4A1AR antagonist 6
CAS:<p>A1AR antagonist 6 (compound 15) is a potent and selective antagonist of A1 adenosine receptor(A1AR) with a pKi of 7.13 and a pIC 50 of 6.38[1].</p>Fórmula:C17H15N3O2Forma y color:SolidPeso molecular:293.32Lu AA41063
CAS:<p>Lu AA41063 is a potent and selective antagonist of the hA2A receptor.</p>Fórmula:C16H17F2N3O2SForma y color:SolidPeso molecular:353.39Neladenoson dalanate HCl
CAS:<p>Neladenoson dalanate HCl is a potent, selective, orally active partial agonist of adenosine A1 receptor (EC50: 0.1 nM).</p>Fórmula:C35H35Cl2N7O4S2Pureza:98%Forma y color:SolidPeso molecular:752.73A3AR antagonist 1
CAS:<p>A3AR antagonist 1 is a potent and selective human A3adenosine receptor (AR) antagonist (Ki: 4.63) and has no affinity for the rat A3AR.</p>Fórmula:C32H24N4O4SForma y color:SolidPeso molecular:560.62Adenosine receptor antagonist 2
CAS:<p>Adenosine receptor antagonist 2 is an orally active A2a (IC50: 1 nM), A2b (IC50: 3 nM) adenosine receptor antagonist that exhibits antitumour effects.</p>Fórmula:C23H21FN8OForma y color:SolidPeso molecular:444.46CAY10498
CAS:<p>A3 AR antagonist CAY10498, with Ki of 37 nM, is 60-200x selective over A1/A2A receptors; no dedifferentiation effects shown.</p>Fórmula:C18H20N6Forma y color:SolidPeso molecular:320.39
