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Receptor de cannabinoides

Receptor de cannabinoides

Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.

Se han encontrado 196 productos de "Receptor de cannabinoides"

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  • Pregnenolone

    CAS:
    <p>Pregnenolone (Arthenolone) is an endogenous steroid hormone synthesized from cholesterol, used in the treatment of Alzheimer's disease.</p>
    Fórmula:C21H32O2
    Pureza:99.5% - >99.99%
    Forma y color:Solid
    Peso molecular:316.48
  • Anandamide

    CAS:
    <p>Anandamide ((5Z,8Z,11Z,14Z)-N-(2-Hydroxyethyl)icosa-5,8,11,14-tetraenamide), an immune modulator, acts via not only cannabinoid receptors (CB1 and CB2) but also</p>
    Fórmula:C22H37NO2
    Pureza:95.037% - 99.22%
    Forma y color:Light Yellow Oil
    Peso molecular:347.53
  • EHP-101

    CAS:
    <p>EHP-101 is a PPARγ/CB2 dual agonist with anti-inflammatory properties, inhibits fat formation, and combats diet-related obesity.</p>
    Fórmula:C28H35NO3
    Pureza:98.36%
    Forma y color:Solid
    Peso molecular:433.58
  • 6-Iodopravadoline

    CAS:
    <p>6-Iodopravadoline (AM630) is an antagonist of CB2 (Ki: 31.2 nM). And it shows 165-fold selectivity more than CB1 receptors.</p>
    Fórmula:C23H25IN2O3
    Pureza:99.29%
    Forma y color:Off-White Solid
    Peso molecular:504.36
  • JHU 75528

    CAS:
    <p>JHU 75528 (JHU-75528) is a novel PET tracer with inhibitory effects on CB that can be used to study the cannabinoid system in schizophrenic patients.</p>
    Fórmula:C23H21Cl2N5O2
    Pureza:99.79%
    Forma y color:Solid
    Peso molecular:470.35
  • Rimonabant hydrochloride

    CAS:
    <p>Rimonabant hydrochloride (SR 141716A) 是中心大麻素受体 1 的高效选择性反向激动剂, Ki 值为1.8 nM。它也能够抑制分枝杆菌膜蛋白3。</p>
    Fórmula:C22H22Cl4N4O
    Pureza:98.24% - 99.5%
    Forma y color:Off-White To White Crystalline Powder
    Peso molecular:500.25
  • CB1 antagonist 2

    CAS:
    <p>CB1 antagonist 2 (AM4113) is caimabinoid 1 (CB1) antagonist which inhibits CB1 in vivo with an IC50 of 25.5 nM.</p>
    Fórmula:C17H12Cl3N3O
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:380.66
  • Rimonabant

    CAS:
    <p>Rimonabant (SR141716) is an inverse agonist for the cannabinoid receptor CB1.</p>
    Fórmula:C22H21Cl3N4O
    Pureza:98% - 99.91%
    Forma y color:White Or Almost White Crystalline Powder
    Peso molecular:463.79
  • VIP36


    <p>VIP36 is an agonist of the cannabinoid type 1 receptor (CB1) with analgesic properties. It reduces the recruitment of inhibitory proteins, thereby exerting its pain-relieving effects, and is applicable in research related to chronic pain.</p>
    Fórmula:C27H35FN6O4
    Forma y color:Solid
    Peso molecular:526.603
  • Hemopressin(rat)

    CAS:
    <p>Peptide inhibitor for ep24.15, neurolysin &amp; ACE with Ki 27.76, 3.43, 1.87 μM. Lowers blood pressure, modulates CB1 receptor, reduces pain &amp; food intake.</p>
    Fórmula:C53H77N13O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1088.27
  • CB2 PET Radioligand 1


    <p>CB2 PET Radioligand 1 (compound [18F]9) is a positron emission tomography (PET) radioligand with high affinity for the human cannabinoid receptor 2 (hCB2, Ki=7.</p>
    Fórmula:C20H19F3N4O
    Pureza:98%
    Forma y color:Solid
    Peso molecular:388.39
  • GPR55 agonist 4


    <p>GPR55 agonist 4 (Compound 28), with an EC50 of 131 nM for hGPR55 and 1.41 nM for rGPR55, effectively induces β-arrestin recruitment to human GPR55 [1].</p>
    Fórmula:C19H16FN5O2
    Forma y color:Solid
    Peso molecular:365.36
  • (±)-9-Nor-9α-hydroxy Hexahydrocannabinol

    CAS:
    <p>(±)-9-Nor-9α-hydroxy Hexahydrocannabinol is a cannabinoid-structured compound that exhibits potent cannabinoid-like activity in both dogs and mice.</p>
    Fórmula:C20H30O3
    Forma y color:Solid
    Peso molecular:318.45
  • Vicasinabin

    CAS:
    <p>Vicasinabin: potent CB2 agonist; researches chronic pain, atherosclerosis, bone mass, neuroinflammation.</p>
    Fórmula:C15H22N10O
    Forma y color:Solid
    Peso molecular:358.41
  • N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide

    CAS:
    <p>N-(1-(3,4-Dihydroxyphenyl)propan-2-yl)oleamide: binds CB1 (Ki=365 nM), activates PPARα (EC50=698 nM), reduces rat food intake, no FAAH inhibition.</p>
    Fórmula:C27H45NO3
    Forma y color:Solid
    Peso molecular:431.661
  • CB2R/FAAH modulator-3

    CAS:
    <p>CB2R/FAAH modulator-3 (compound 27) is a modulator targeting at CB2R and FAAH.</p>
    Fórmula:C22H31NO2
    Pureza:99.81%
    Forma y color:Soild
    Peso molecular:341.49
  • (R)-Zevaquenabant


    <p>(R)-Zevaquenabant ((R)-MRI-1867) is the enantiomer of Zevaquenabant. Zevaquenabant ((S)-MRI-1867) is a peripherally restricted, orally bioavailable dual antagonist of the cannabinoid CB1 receptor and inducible nitric oxide synthase (iNOS). It is beneficial in improving chronic kidney disease (CKD) caused by obesity.</p>
    Forma y color:Odour Solid
  • GFB-024


    <p>GFB-024 is a humanized antibody targeting CB1, which can be used to study obesity.</p>
    Forma y color:Liquid
    Peso molecular:145.5kDa
  • Δ8-THC methyl ether

    CAS:
    <p>Δ8-THC methyl ether (compound 3) demonstrates a strong docking score of -10.167 kcal/mol for the CB2 receptor. Additionally, Δ8-THC methyl ether exhibits antinociceptive activity in mice.</p>
    Fórmula:C22H32O2
    Forma y color:Solid
    Peso molecular:328.49
  • exo-Tetrahydrocannabivarin

    CAS:
    <p>exo-Tetrahydrocannabivarin (Compound 12) is an analog of Δ9,11-THC. It weakly binds to cannabinoid receptors (CB) with an IC50 of 1.4 μM. In mice, exo-Tetrahydrocannabivarin exhibits activity related to both motor function and analgesia.</p>
    Fórmula:C19H26O2
    Forma y color:Solid
    Peso molecular:286.41
  • CB2 receptor agonist 2

    CAS:
    <p>CB2 receptor agonist 2 (ZINC72105556): potent, Ki=8.5 nM, high selectivity for CB2.</p>
    Fórmula:C30H36N2O4
    Pureza:99.75%
    Forma y color:Solid
    Peso molecular:488.62
  • CB2R agonist 2


    <p>CB2R agonist 2 (cis-17-para) is a CB2R agonist [1].</p>
    Pureza:98%
    Forma y color:Odour Solid
  • CB2R/FAAH modulator-2

    CAS:
    <p>CB2R/FAAH modulator-2 (compound 26) is a dual modulator targeting at CB2R and FAAH.</p>
    Fórmula:C24H33NO2
    Pureza:99.15%
    Forma y color:Soild
    Peso molecular:367.52
  • PSB-SB-1203

    CAS:
    <p>PSB-SB-1203 (Compound 25b) is a dual CB1/CB2 ligand that blocks the CB1 receptor and activates the CB2 receptor with a CB1 Ki of 0.244 μM, a CB2 Ki of 0.210 μM, and an EC50 of 0.054 μM. It shows potential for research in obesity and cancer.</p>
    Fórmula:C25H30O4
    Forma y color:Solid
    Peso molecular:394.5
  • Zevaquenabant

    CAS:
    <p>Zevaquenabant (S-MRI-1867): oral CB1/iNOS antagonist combatting obesity-induced CKD.</p>
    Fórmula:C25H21ClF3N5O2S
    Forma y color:Solid
    Peso molecular:547.98
  • CB2 receptor agonist 9

    CAS:
    <p>CB2 receptor agonist 9 (Compound 33) is an orally active agonist of cannabinoid receptor 2 (CB2 receptor) with an EC50 of 16.2 nM. It inhibits the expression of TNF-α, IL-1β, and IL-6, demonstrating anti-inflammatory activity in a DSS-induced acute colitis model in mice.</p>
    Fórmula:C16H23N3O2S
    Forma y color:Solid
    Peso molecular:321.44
  • CB2R probe 1

    CAS:
    <p>CB2R Probe 1, a cannabinoid 2 receptor (CB2R) fluorescent probe, exhibits both safety and environmental friendliness, boasting a dissociation constant (K i) of</p>
    Fórmula:C36H42N4O4
    Forma y color:Solid
    Peso molecular:594.74
  • Hemopressin (human, mouse)

    CAS:
    <p>Endogenous peptide, inhibits ep24.15/24.16/ACE with Ki of 27.76/3.43/1.87 μM. Lowers blood pressure, CB1 inverse agonist, reduces pain in vivo.</p>
    Fórmula:C50H79N13O12
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1054.26
  • Drinabant

    CAS:
    <p>Drinabant (AVE-1625) is an orally active CB1 receptor antagonist.</p>
    Fórmula:C23H20Cl2F2N2O2S
    Pureza:99.8%
    Forma y color:Solid
    Peso molecular:497.38
  • CB1R antagonist 2


    <p>CB1R antagonist 2 (Compound 11g) functions as an antagonist of the cannabinoid receptor 1 (CB1R), inhibiting the MAPK/NF-κB signaling pathway and exhibiting anti-inflammatory properties. In RAW264.7 cells, it suppresses LPS-induced expression of IL-6, IL-1β, and TNF-α. In murine models, it improves OVA-induced allergic rhinitis.</p>
    Fórmula:C24H26N4O
    Forma y color:Solid
    Peso molecular:386.49
  • Hemopressin(human, mouse) TFA

    CAS:
    <p>Hemopressin TFA: nonapeptide from hemoglobin, oral CB1 inverse agonist, eases inflammatory pain.</p>
    Fórmula:C52H80F3N13O14
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1168.27
  • Afubiata

    CAS:
    <p>ADB-FUBIATA is a synthetic cannabinoid studied for its metabolic profile, along with AFUBIATA, CH-FUBIATA, and CH-PIATA. This in vitro analysis by Watanabe S, et al., examines these compounds, as published in "Arch Toxicol," 2023 Dec;97(12):3085-3094.</p>
    Fórmula:C27H29FN2O
    Forma y color:Solid
    Peso molecular:416.53
  • NESS 0327

    CAS:
    <p>NESS 0327 is a high selectivity antagonist of the cannabinoid CB1 receptor. NESS 0327 is more than 60,000-fold selective for the CB1 receptor.</p>
    Fórmula:C24H23Cl3N4O
    Pureza:99.78%
    Forma y color:Solid
    Peso molecular:489.82
  • Cannabidivarinic acid

    CAS:
    <p>Cannabidivarinic acid (CBDVA), the carboxylic acid precursor to cannabidivarin (CBDV), is a non-psychoactive cannabinoid found in Cannabis and known for its anti-inflammatory properties.</p>
    Fórmula:C20H26O4
    Forma y color:Solid
    Peso molecular:330.42
  • APP-FUBINACA

    CAS:
    <p>APP-FUBINACA is a cannabinoid receptor agonist, classified as a phenylalanine amide-based indazole-3-carboxamide derivative. It exhibits neurostimulatory effects.</p>
    Fórmula:C24H21FN4O2
    Forma y color:Solid
    Peso molecular:416.45
  • Tocrifluor T1117

    CAS:
    <p>Fluorescent form of AM 251, CB1 receptor antagonist</p>
    Fórmula:C56H53Cl2N7O5
    Pureza:98%
    Forma y color:Solid
    Peso molecular:974.97
  • δ8-THC acetate

    CAS:
    <p>Delta8-THC acetate (Delta8-tetrahydrocannabinol) is a psychoactive cannabinoid that binds to the cannabinoid receptor 1 (CB1 receptor) and exhibits anti-nausea, appetite-stimulating, and anti-inflammatory effects. It may also offer neuroprotective benefits and has potential applications in research on anxiety and depression.</p>
    Fórmula:C23H32O3
    Forma y color:Solid
    Peso molecular:356.5
  • Noladin ether

    CAS:
    <p>Noladin ether (2-AG ether) is a cannabinoid CB1 receptor agonist.</p>
    Fórmula:C23H40O3
    Forma y color:Solid
    Peso molecular:364.56
  • TRPV1/CB2 agonist 1


    <p>TRPV1/CB2 agonist 1 (compound 41) is a dual agonist targeting hTRPV1 and CB2 receptors, with an EC50 value of 26.8 μM for hTRPV1. It is applicable in research related to the nervous system.</p>
    Forma y color:Odour Solid
  • 8β-Hydroxy-exo-THC

    CAS:
    <p>8β-Hydroxy-exo-THC, a cannabinoid ether analog, exhibits weak affinity for receptor sites with an IC50 of 1.2 μM.</p>
    Fórmula:C21H30O3
    Forma y color:Solid
    Peso molecular:330.46
  • Δ8-THC-C8

    CAS:
    <p>Δ8-THC-C8 is a semi-synthetic cannabinoid. It acts as an agonist for the cannabinoid receptor 1 (CB1) with an EC50 value of 13.8 nM.</p>
    Fórmula:C24H36O2
    Forma y color:Solid
    Peso molecular:356.54
  • RVD-Hpα

    CAS:
    <p>N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>
    Fórmula:C65H105N19O17
    Pureza:98%
    Forma y color:Solid
    Peso molecular:1424.66
  • CB2R/FAAH modulator-1

    CAS:
    <p>CB2R/FAAH modulator-1: agonizes CB2R, inhibits FAAH (IC50=4 μM), alters cytokine production; used in inflammation research. Ki: CB2R=14.8 nM, CB1R=241.3 nM.</p>
    Fórmula:C24H27NO2
    Pureza:99.77%
    Forma y color:Soild
    Peso molecular:361.48
  • CB2R agonist 3


    <p>CB2R agonist 3, a potent activator of cannabinoid receptor 2 (CB2R), exhibits an EC50 value of 0.37μM, indicative of its significant role in the immune system [</p>
    Pureza:98%
    Forma y color:Odour Solid
  • CB1R agonist 1


    <p>CB1R agonist 1 (Compound '1350) is a potent full agonist of the cannabinoid-1 receptor (CB1R) with a Ki value of 0.95 nM. It demonstrates significant pain-relieving effects in various pain models, including acute thermal pain, inflammatory pain, and neuropathic pain.</p>
    Fórmula:C20H18F3N3O3S
    Forma y color:Solid
    Peso molecular:437.435
  • Virodhamine

    CAS:
    <p>Virodhamine (O-arachidonoyl ethanolamine), an endocannabinoid, is an antagonist of CB1 receptor and an agonist of CB2 receptor.</p>
    Fórmula:C22H37NO2
    Pureza:98%
    Forma y color:Soild
    Peso molecular:347.53
  • Taranabant racemate

    CAS:
    <p>Taranabant racemate is an antagonist and/or inverse agonist of the Cannabinoid-1 (CB1) receptor.</p>
    Fórmula:C27H25ClF3N3O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:515.95
  • β-Caryophyllene

    CAS:
    <p>β-Caryophyllene ((-)-(E)-Caryophyllene) acts as an CB2 receptor agonist.</p>
    Fórmula:C15H24
    Pureza:95.43% - 99.11%
    Forma y color:Turpentine (Ntp 1992)
    Peso molecular:204.35
  • ML-184

    CAS:
    <p>ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.</p>
    Fórmula:C25H34N4O3S
    Pureza:99.45%
    Forma y color:Solid
    Peso molecular:470.63
  • AM281

    CAS:
    <p>AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.</p>
    Fórmula:C21H19Cl2IN4O2
    Pureza:98.6% - >99.99%
    Forma y color:White To Off-White Solid
    Peso molecular:557.21
  • Linoleoyl Ethanolamide

    CAS:
    <p>Linoleoyl Ethanolamide is an endocannabinoid agent.</p>
    Fórmula:C20H37NO2
    Pureza:99.97%
    Forma y color:Solid
    Peso molecular:323.51
  • Otenabant

    CAS:
    <p>Otenabant (CP-945598) has been investigated for the treatment of Obesity.</p>
    Fórmula:C25H25Cl2N7O
    Pureza:99.43%
    Forma y color:Solid
    Peso molecular:510.42
  • CB1 antagonist 4

    CAS:
    <p>TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.</p>
    Fórmula:C30H25Cl2F3N4OS
    Pureza:98.97%
    Forma y color:Solid
    Peso molecular:617.51
  • LY2828360

    CAS:
    <p>LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and &gt;100 μM.</p>
    Fórmula:C22H27ClN6O
    Pureza:98.45% - 99.51%
    Forma y color:Solid
    Peso molecular:426.94
  • A-836339

    CAS:
    <p>A-836339: Potent cannabinoid, CB2-focused (Ki=0.64nM), lesser CB1 affinity (Ki=270nM); analgesic, anti-inflammatory in mice.</p>
    Fórmula:C16H26N2O2S
    Pureza:99.94%
    Forma y color:Solid
    Peso molecular:310.45
  • Tetrahydromagnolol

    CAS:
    <p>Tetrahydromagnolol can activate cannabinoid (CB) receptors.</p>
    Fórmula:C18H22O2
    Pureza:99.86% - >99.99%
    Forma y color:Solid
    Peso molecular:270.37
  • CB1-IN-1

    CAS:
    <p>CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.</p>
    Fórmula:C33H31Cl2F3N6O3S2
    Pureza:99.08% - 99.76%
    Forma y color:Solid
    Peso molecular:751.67
  • ML-193

    CAS:
    <p>ML-193: GPR55 antagonist, IC50 221nM, 27x selective over GPR35/CB1/CB2, may aid Parkinson's symptoms.</p>
    Fórmula:C28H25N5O4S
    Pureza:97.74%
    Forma y color:Solid
    Peso molecular:527.59
  • Otenabant hydrochloride

    CAS:
    <p>Otenabant hydrochloride (Otenabant) (CP-945598) is a competitive, high affinity, selective antagonist of the CB1 receptor (Ki: 0.7 nM).</p>
    Fórmula:C25H26Cl3N7O
    Pureza:99.79% - ≥95%
    Forma y color:Solid
    Peso molecular:546.88
  • Cannabigerol

    CAS:
    <p>Cannabigerol is a high affinity α±2-adrenergic receptor agonist, moderate affinity 5-HT1A receptor antagonist, and low affinity CB1 receptor antagonist ; also</p>
    Fórmula:C21H32O2
    Pureza:99.59% - 99.92%
    Forma y color:Solid
    Peso molecular:316.48
  • AM251

    CAS:
    <p>AM251: potent CB1 blocker (IC50: 8 nM), 306x CB2 selective; GPR55 activator (EC50: 39 nM).</p>
    Fórmula:C22H21Cl2IN4O
    Pureza:97.43% - 98.79%
    Forma y color:A Crystalline Solid
    Peso molecular:555.24
  • Hemopressin (human, mouse) acetate


    <p>Hemopressin: Nonapeptide, α1-hemoglobin derivative, CB1 inverse agonist, isolated from rats, oral, reduces inflammatory pain.</p>
    Fórmula:C52H83N13O14
    Pureza:99.86%
    Forma y color:Solid
    Peso molecular:1114.29
  • ARN272

    CAS:
    <p>ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).</p>
    Fórmula:C27H20N4O2
    Pureza:98.23%
    Forma y color:Solid
    Peso molecular:432.47
  • Voacamine

    CAS:
    <p>Voacamine: an indole alkaloid, CB1 antagonist, inhibits P-gp, may affect rhythm.</p>
    Fórmula:C43H52N4O5
    Pureza:98.54% - 99.82%
    Forma y color:Solid
    Peso molecular:704.9
  • AM1241

    CAS:
    <p>AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.</p>
    Fórmula:C22H22IN3O3
    Pureza:98.937% - 99.1%
    Forma y color:Solid
    Peso molecular:503.33
  • yangonin

    CAS:
    <p>Yangonin (Y100550) is a novel CB1 receptor ligand with affinity for human recombinant CB1 receptors.</p>
    Fórmula:C15H14O4
    Pureza:98.82% - 99.55%
    Forma y color:Pale Yellow Powder
    Peso molecular:258.27
  • Olivetol

    CAS:
    <p>Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.</p>
    Fórmula:C11H16O2
    Pureza:99.98%
    Forma y color:(Melting Point 102-106°F) (Ntp 1992)
    Peso molecular:180.24
  • ML-191

    CAS:
    <p>ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.</p>
    Fórmula:C24H25N3O3
    Pureza:99.58%
    Forma y color:Solid
    Peso molecular:403.47
  • Hemopressin (rat) acetate(568588-77-2 free base)


    <p>Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.</p>
    Fórmula:C5H81N13O14
    Pureza:99.37%
    Forma y color:Solid
    Peso molecular:1148.31
  • Org 27569

    CAS:
    <p>Org 27569, an allosteric modulator of cannabinoid CB1 receptor, can induce a CB1 receptor state that is characterized by decreased inverse agonist affinity and</p>
    Fórmula:C24H28ClN3O
    Pureza:>99.99% - ≥95%
    Forma y color:Solid
    Peso molecular:409.95
  • JD-5037

    CAS:
    <p>JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.</p>
    Fórmula:C27H27Cl2N5O3S
    Pureza:99.54% - 99.84%
    Forma y color:Solid
    Peso molecular:572.51
  • PSB-SB-487

    CAS:
    <p>PSB-SB-487 is antagonist of GPR55.</p>
    Fórmula:C26H32O4
    Pureza:98.53%
    Forma y color:Solid
    Peso molecular:408.53
  • BML-190

    CAS:
    <p>BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体,其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki&gt; 2 μM)。</p>
    Fórmula:C23H23ClN2O4
    Pureza:97.70%
    Forma y color:Solid
    Peso molecular:426.89
  • CID 16020046

    CAS:
    <p>CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.</p>
    Fórmula:C25H19N3O4
    Pureza:99.03%
    Forma y color:Solid
    Peso molecular:425.44
  • GW 405833

    CAS:
    <p>GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selective</p>
    Fórmula:C23H24Cl2N2O3
    Pureza:99.82% - 99.93%
    Forma y color:Solid
    Peso molecular:447.35
  • GW842166X

    CAS:
    <p>GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.</p>
    Fórmula:C18H17Cl2F3N4O2
    Pureza:99.47%
    Forma y color:Solid
    Peso molecular:449.25
  • RTICBM-189

    CAS:
    <p>RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.</p>
    Fórmula:C15H14Cl2N2O
    Pureza:99.96%
    Forma y color:Solid
    Peso molecular:309.19
  • Bay 59-3074

    CAS:
    <p>Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).</p>
    Fórmula:C18H13F6NO4S
    Pureza:97.68% - 99.69%
    Forma y color:Solid
    Peso molecular:453.36
  • (±)-Ibipinabant

    CAS:
    <p>(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.</p>
    Fórmula:C23H20Cl2N4O2S
    Pureza:99.28% - 99.83%
    Forma y color:Solid
    Peso molecular:487.4
  • N-Oleoyl glycine

    CAS:
    <p>N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated Akt</p>
    Fórmula:C20H37NO3
    Pureza:97.43%
    Forma y color:Solid
    Peso molecular:339.51
  • RVD-Hpα acetate(1193362-76-3 free base)


    <p>RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.</p>
    Fórmula:C67H109N19O19
    Pureza:99.87%
    Forma y color:Solid
    Peso molecular:1484.71
  • CB1/2 agonist 3

    CAS:
    <p>CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.</p>
    Fórmula:C25H41NO2
    Pureza:98.78%
    Forma y color:Solid
    Peso molecular:387.6
  • S-Methoprene

    CAS:
    <p>S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.</p>
    Fórmula:C19H34O3
    Pureza:97.05% - 98.55%
    Forma y color:Solid
    Peso molecular:310.47
  • Dehydroabiethylamine

    CAS:
    <p>Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs &amp; cholesterol transport, and has anti-tumor effects.</p>
    Fórmula:C20H31N
    Pureza:98.79%
    Forma y color:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber Liquid
    Peso molecular:285.47
  • AM404

    CAS:
    <p>AM404 is a cannabinoid reuptake inhibitor and a TRPV (1) activator with neuroprotective and anticancer activities that blocks anandamide transport.</p>
    Fórmula:C26H37NO2
    Forma y color:Solid
    Peso molecular:395.58
  • LEI-101

    CAS:
    <p>LEI-101: potent CB2 agonist, pEC50=8, bioavailable, &gt;100x selective over CB1, potential for inflammatory diseases.</p>
    Fórmula:C23H25FN4O4S
    Pureza:98%
    Forma y color:Solid
    Peso molecular:472.53
  • UCM 707

    CAS:
    <p>endocannabinoid transport inhibitor</p>
    Fórmula:C25H37NO2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:383.57
  • CB1-IN-2

    CAS:
    <p>CB1-IN-2 (4g) inhibits CB1 receptor with 0.644 μM IC50; crosses blood-brain barrier, may cause CNS side effects like Rimonabant.</p>
    Fórmula:C17H19Cl2N5O
    Forma y color:Solid
    Peso molecular:380.27
  • VSN-16

    CAS:
    <p>VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.</p>
    Fórmula:C18H26N2O3
    Forma y color:Solid
    Peso molecular:318.41
  • CB1R Allosteric modulator 4

    CAS:
    <p>Modulates CB1R positively; inhibits cAMP production; strong β-arrestin-2 recruitment.</p>
    Fórmula:C20H17N3O2S
    Forma y color:Solid
    Peso molecular:363.43
  • UCM710

    CAS:
    <p>UCM710 is a dual inhibitor of α/β hydrolase domain 6 (ABHD6) and fatty acid amide hydrolase (FAAH).</p>
    Fórmula:C19H34O3
    Pureza:98%
    Forma y color:Solid
    Peso molecular:310.47
  • CB1/2 agonist 4

    CAS:
    <p>CB1/2 agonist 4 is a potent CB1 full agonist (EC50: 15.09 nM) and CB2 partial agonist (EC50: 1.16 nM), with anti-pain and TRPV1 activation properties.</p>
    Fórmula:C27H45NO3
    Forma y color:Solid
    Peso molecular:431.65
  • Palmitoyl serinol

    CAS:
    <p>Anticancer agent 110 is an anticancer compound with cytotoxic, antitumor and antileukemic activities.</p>
    Fórmula:C19H39NO3
    Forma y color:Solid
    Peso molecular:329.52
  • (R)-SLV 319

    CAS:
    <p>(R)-SLV 319: potent CB1 antagonist, K i of 894 nM, dextrorotatory isomer.</p>
    Fórmula:C23H20Cl2N4O2S
    Forma y color:Solid
    Peso molecular:487.4
  • LH 21

    CAS:
    <p>LH-21, a strong CB1 receptor antagonist, curbs eating and lessens weight gain in obese rats.</p>
    Fórmula:C20H20Cl3N3
    Forma y color:Solid
    Peso molecular:408.75
  • NIDA 41020

    CAS:
    <p>NIDA 41020 is a CB1 receptor antagonist.</p>
    Fórmula:C23H24Cl2N4O2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:459.37
  • AM-6538

    CAS:
    <p>AM6538: long-acting, high-affinity CB antagonist similar to rimonabant, useful for studying cannabinoid agonists.</p>
    Fórmula:C26H25Cl2N5O4
    Forma y color:Solid
    Peso molecular:542.41
  • CID1792197

    CAS:
    <p>CID1792197 is a selective agonist of GPR55.</p>
    Fórmula:C24H23N3O4S2
    Pureza:98%
    Forma y color:Solid
    Peso molecular:481.59
  • PM226

    CAS:
    <p>CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.</p>
    Fórmula:C22H31NO3
    Forma y color:Solid
    Peso molecular:357.49
  • GPR55 agonist 3

    CAS:
    <p>Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.</p>
    Fórmula:C19H16F4N4
    Forma y color:Solid
    Peso molecular:376.35