Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Se han encontrado 217 productos de "Receptor de cannabinoides"
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Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Fórmula:C18H22O2Pureza:99.86% - >99.99%Forma y color:SolidPeso molecular:270.37Ref: TM-TN2268
2mgA consultar5mg52,00€10mg81,00€25mgA consultar50mg170,00€100mg243,00€1mL*10mM (DMSO)63,00€PSB-SB-487
CAS:PSB-SB-487 is antagonist of GPR55.Fórmula:C26H32O4Pureza:98.53%Forma y color:SolidPeso molecular:408.53Ref: TM-T8975
1mg35,00€5mg80,00€10mg119,00€25mg231,00€50mg344,00€100mg480,00€200mg660,00€1mL*10mM (DMSO)87,00€ML-191
CAS:ML-191 is an inhibitor of LPI-induced phosphorylation of ERK1/2.Fórmula:C24H25N3O3Pureza:99.58%Forma y color:SolidPeso molecular:403.47GW842166X
CAS:GW842166X: Potent CB2 agonist, EC50=63 nM, inactive at CB1, in Phase 2 trials.Fórmula:C18H17Cl2F3N4O2Pureza:99.47%Forma y color:SolidPeso molecular:449.25ML-184
CAS:ML-184 (CID2440433) is a potent synthetic agonist of GPR55 with EC50 of 0.26 μM.Fórmula:C25H34N4O3SPureza:99.45%Forma y color:SolidPeso molecular:470.63RTICBM-189
CAS:RTICBM-189 is a potent, brain-penetrant allosteric modulator of the cannabinoid type-1 (CB1) receptor with a pIC50 of 7.54 in Ca2+ mobilization assay.Fórmula:C15H14Cl2N2OPureza:99.96%Forma y color:SolidPeso molecular:309.19Ref: TM-T9466
2mg34,00€5mg52,00€10mg84,00€25mg161,00€50mg250,00€100mg369,00€200mg522,00€1mL*10mM (DMSO)67,00€ARN272
CAS:ARN272 is a FAAH-like anandamide transporter (FLAT) inhibitor (IC50: 1.8 μM).Fórmula:C27H20N4O2Pureza:98.23%Forma y color:SolidPeso molecular:432.47JD-5037
CAS:JD-5037 is a novel, peripherally restricted CB1R antagonist with an IC50 of 1.5 nM.Fórmula:C27H27Cl2N5O3SPureza:99.54% - 99.84%Forma y color:SolidPeso molecular:572.51Ref: TM-T4453
1mg42,00€2mg55,00€5mg90,00€10mg133,00€25mg234,00€50mg350,00€100mg522,00€1mL*10mM (DMSO)101,00€AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Fórmula:C24H20N2OPureza:99.37%Forma y color:SolidPeso molecular:352.43Olivetol
CAS:Olivetol, found in lichens, is an organic antioxidant and THC synthesis precursor.Fórmula:C11H16O2Pureza:99.98%Forma y color:(Melting Point 102-106°F) (Ntp 1992)Peso molecular:180.24Hemopressin (rat) acetate(568588-77-2 free base)
Hemopressin is a nonapeptide, CB2 agonist, derived from rat hemoglobin, with antinociceptive properties.Fórmula:C5H81N13O14Pureza:99.37%Forma y color:SolidPeso molecular:1148.31AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Fórmula:C21H19Cl2IN4O2Pureza:98.6% - >99.99%Forma y color:White To Off-White SolidPeso molecular:557.21Ref: TM-T2264
1mg80,00€5mg169,00€10mg259,00€25mg523,00€50mg750,00€100mg1.035,00€500mg2.062,00€1mL*10mM (DMSO)233,00€RVD-Hpα acetate(1193362-76-3 free base)
RVD-Hpα acetate is the N-terminally extended form of human hemopressin that acts as a selective CB1 receptor agonist.Fórmula:C67H109N19O19Pureza:99.87%Forma y color:SolidPeso molecular:1484.71Bay 59-3074
CAS:Bay 59-3074 is a CB1/CB2 receptor partial agonist (Ki: 48.3/45.5 nM).
Fórmula:C18H13F6NO4SPureza:97.68% - 99.69%Forma y color:SolidPeso molecular:453.36AM1241
CAS:AM-1241 is a selective cannabinoid CB2 receptor agonist with Ki of 3.4 nM, exhibits 82-fold selectivity over CB1 receptor.Fórmula:C22H22IN3O3Pureza:98.937% - 99.1%Forma y color:SolidPeso molecular:503.33Ref: TM-T6755
2mg35,00€5mg49,00€10mg84,00€25mg168,00€50mg275,00€100mg495,00€500mg1.071,00€1mL*10mM (DMSO)87,00€Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Fórmula:C20H37NO2Pureza:99.97%Forma y color:SolidPeso molecular:323.51Ref: TM-T8425
1mg35,00€5mg67,00€10mg90,00€25mg164,00€50mg239,00€100mg348,00€200mg522,00€1mL*10mM (DMSO)85,00€CB1 antagonist 4
CAS:TM38837 is an antagonist of cannabinoid receptor type 1 (CB1), with potential for the treatment of obesity and type 2 diabetes.Fórmula:C30H25Cl2F3N4OSPureza:98.97%Forma y color:SolidPeso molecular:617.51Ref: TM-T8511
2mg46,00€5mg92,00€10mg152,00€25mg259,00€50mg405,00€100mg597,00€200mg848,00€1mL*10mM (DMSO)155,00€Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Fórmula:C25H25Cl2N7OPureza:99.43%Forma y color:SolidPeso molecular:510.42N-Oleoyl glycine
CAS:N-Oleoyl glycine, a lipoamino acid, was able to promote 3T3-L1 adipogenesis through the activation of CB1 receptor and the enhancement of insulin-mediated AktFórmula:C20H37NO3Pureza:97.43%Forma y color:SolidPeso molecular:339.51CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Fórmula:C33H31Cl2F3N6O3S2Pureza:99.08% - 99.76%Forma y color:SolidPeso molecular:751.67Ref: TM-T5996
1mg82,00€2mg110,00€5mg180,00€10mg258,00€25mg423,00€50mg588,00€100mg793,00€500mg1.594,00€1mL*10mM (DMSO)215,00€
