Receptor de cannabinoides
Los receptores cannabinoides son GPCR que median los efectos de los cannabinoides endógenos (endocannabinoides) y los fitocannabinoides, como los encontrados en el cannabis. Los dos tipos principales de receptores cannabinoides, CB1 y CB2, están involucrados en la regulación de una amplia gama de procesos fisiológicos, incluida la percepción del dolor, el apetito, el estado de ánimo y la función inmunitaria. Los moduladores de los receptores cannabinoides tienen potencial terapéutico en el tratamiento de afecciones como el dolor crónico, la epilepsia y la esclerosis múltiple. En CymitQuimica, ofrecemos una amplia gama de moduladores de receptores cannabinoides de alta calidad para apoyar su investigación en neurofarmacología, manejo del dolor e inmunología.
Se han encontrado 217 productos de "Receptor de cannabinoides"
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(±)-Ibipinabant
CAS:(±)-Ibipinabant ((±)-SLV319) has been used in trials studying the treatment of Obesity and Obesity and Type 2 Diabetes.Fórmula:C23H20Cl2N4O2SPureza:99.28% - 99.83%Forma y color:SolidPeso molecular:487.4GW 405833
CAS:GW 405833 (L-768242) is an agonist of cannabinoid-2 (CB(2)) receptor-selectiveFórmula:C23H24Cl2N2O3Pureza:99.82% - 99.93%Forma y color:SolidPeso molecular:447.35Linoleoyl Ethanolamide
CAS:Linoleoyl Ethanolamide is an endocannabinoid agent.Fórmula:C20H37NO2Pureza:99.97%Forma y color:SolidPeso molecular:323.51Ref: TM-T8425
1mg35,00€5mg67,00€10mg90,00€25mg164,00€50mg239,00€100mg348,00€200mg522,00€1mL*10mM (DMSO)85,00€AM281
CAS:AM 281, a cannabinoid antagonist, reduces neurologic dysfunction and mortality rate after cecal ligation and puncture in rats.Fórmula:C21H19Cl2IN4O2Pureza:98.6% - >99.99%Forma y color:White To Off-White SolidPeso molecular:557.21Ref: TM-T2264
1mg80,00€5mg169,00€10mg259,00€25mg523,00€50mg750,00€100mg1.035,00€500mg2.062,00€1mL*10mM (DMSO)233,00€AM-2232
CAS:AM-2232 (UNII-40KCH8YIKP) is a potent and unselective agonist of the cannabinoid receptors.Fórmula:C24H20N2OPureza:99.37%Forma y color:SolidPeso molecular:352.43LY2828360
CAS:LY2828360: CB2 agonist, Ki=40.3 nM; biases CB2 over CB1 with EC50s of 20.1 nM and >100 μM.Fórmula:C22H27ClN6OPureza:98.45% - 99.51%Forma y color:SolidPeso molecular:426.94CID 16020046
CAS:CID 16020046 (C390-0219) is a selective GPR55 antagonist, inhibiting GPR55 constitutive activity with IC50 of 0.15 μM in yeast.Fórmula:C25H19N3O4Pureza:99.03%Forma y color:SolidPeso molecular:425.44Otenabant
CAS:Otenabant (CP-945598) has been investigated for the treatment of Obesity.Fórmula:C25H25Cl2N7OPureza:99.43%Forma y color:SolidPeso molecular:510.42CB1-IN-1
CAS:CB1-IN-1 (DBPR211) is a peripherally restricted CB1R antagonist, for CB1R and CB2R with Ki of 0.3 nM and 21 nM,respectively.Fórmula:C33H31Cl2F3N6O3S2Pureza:99.08% - 99.76%Forma y color:SolidPeso molecular:751.67Ref: TM-T5996
1mg82,00€2mg110,00€5mg180,00€10mg258,00€25mg423,00€50mg588,00€100mg793,00€500mg1.594,00€1mL*10mM (DMSO)215,00€Tetrahydromagnolol
CAS:Tetrahydromagnolol can activate cannabinoid (CB) receptors.Fórmula:C18H22O2Pureza:99.86% - >99.99%Forma y color:SolidPeso molecular:270.37Ref: TM-TN2268
2mg37,00€5mg52,00€10mg81,00€25mgA consultar50mg170,00€100mg243,00€1mL*10mM (DMSO)63,00€BML-190
CAS:BML-190 (Indomethacin morpholinylamide) 是一种 CB2 受体的配体，其对 CB2 受体 (Ki:435 nM) 和 CB1受体 (Ki> 2 μM)。Fórmula:C23H23ClN2O4Pureza:97.70%Forma y color:SolidPeso molecular:426.89CB1/2 agonist 3
CAS:CB1/2 agonist 3 is a competitive and potent CB1/CB2 agonist with high affinity for hCB1 and hCB2 and can be used to study neurological disorders.Fórmula:C25H41NO2Pureza:98.78%Forma y color:SolidPeso molecular:387.6S-Methoprene
CAS:S-Methoprene (ZR2458), a juvenile hormone analog, acts as an insecticide influencing redox activity and male sex differentiation.
Fórmula:C19H34O3Pureza:97.05% - 98.55%Forma y color:SolidPeso molecular:310.47Dehydroabiethylamine
CAS:Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.Fórmula:C20H31NPureza:98.79%Forma y color:Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber LiquidPeso molecular:285.47PSB-KK1445
CAS:PSB-KK1445 is a potent and selective agonist of GPR18, exhibiting EC50 values of 45.4 nM for humans and 124 nM for mice. The selectivity of PSB-KK1445 for GPR18 over the CB receptor subtypes GPR55 and GPR183 exceeds 200-fold.Fórmula:C24H23FN6O2Peso molecular:446.48GPR55 agonist 3
CAS:Compound 26, a GPR55 agonist, exhibits potent activity with EC50 values of 0.239 nM for hGPR55 and 1.76 nM for rGPR55.Fórmula:C19H16F4N4Forma y color:SolidPeso molecular:376.35PM226
CAS:CB2 agonist with Ki of 12.8 nM; EC50 of 38.67 nM. Negligible CB1 affinity, no GPR55 activity. Anti-inflammatory, neuroprotective, crosses BBB.Fórmula:C22H31NO3Forma y color:SolidPeso molecular:357.49CID1792197
CAS:CID1792197 is a selective agonist of GPR55.Fórmula:C24H23N3O4S2Pureza:98%Forma y color:SolidPeso molecular:481.59VSN-16
CAS:VSN-16, a cannabinoid receptor agonist, is used potentially for the treatment of spasticity in multiple sclerosis.Fórmula:C18H26N2O3Forma y color:SolidPeso molecular:318.41GAT229
CAS:GAT229 is a CB1 positive modulator, enhancing CB agonist activity without direct activation; influences binding, signaling, and lowers ocular pressure in mice.Fórmula:C22H18N2O2Forma y color:SolidPeso molecular:342.39
