Proteasa del VIH
Los inhibidores de la proteasa del VIH son una clase de fármacos antirretrovirales que atacan específicamente la enzima proteasa del virus de la inmunodeficiencia humana (VIH). Al inhibir esta enzima, estos compuestos evitan que el virus procese sus poliproteínas en proteínas maduras y funcionales, bloqueando así la producción de nuevos viriones infecciosos. Los inhibidores de la proteasa del VIH son una piedra angular de la terapia antirretroviral altamente activa (TARGA) utilizada para manejar el VIH/SIDA. En CymitQuimica, ofrecemos una variedad de inhibidores de la proteasa del VIH para apoyar su investigación en el tratamiento del VIH, la resistencia a los medicamentos y la virología.
Se han encontrado 451 productos de "Proteasa del VIH"
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HIV p17 Gag (77-85)
CAS:<p>Targeting HIV Gag p17 (77-85) with intracellular Ab cDNA disrupts viral replication pre/post-integration.</p>Fórmula:C44H72N10O15Pureza:98%Forma y color:SolidPeso molecular:981.1Globotriaosylceramides (porcine)
CAS:Globotriaosylceramides, cell membrane glycosphingolipids, act as Shiga toxin receptors and accumulate in Fabry disease, resisting HIV by blocking gp120.Fórmula:C60H113NO18Forma y color:SolidPeso molecular:1136.553SPD-756
CAS:<p>SPD-756, a nucleoside reverse transcriptase inhibitor, is used potentially for the treatment of HIV infection.</p>Fórmula:C12H16N6O3Pureza:98%Forma y color:SolidPeso molecular:292.29Scirpusin A
CAS:<p>Scirpusin A is a hydroxystilbene dimer from the rhizome of Scirpus fluviatilis and Xinjiang wine grape.</p>Fórmula:C28H22O7Forma y color:SolidPeso molecular:470.47HIV-1 inhibitor-58
<p>HIV-1 Inhibitor-58 (Compound 10c) is a non-nucleoside reverse transcriptase inhibitor with broad-spectrum antiviral properties, effective against both wild-type</p>Fórmula:C26H24N6O2Forma y color:SolidPeso molecular:452.51Salvianan A
CAS:<p>1,6,11-Trimethyl-1,2-dihydrofuro[2',3':1,2]phenanthro[4,3-d]oxazole (compound 1) serves as an effective anti-HIV-1 agent [1].</p>Fórmula:C20H17NO2Forma y color:SolidPeso molecular:303.35VRC01LS
<p>VRC01LS is a humanized monoclonal antibody inhibitor that targets the CD4 binding site of the HIV-1 envelope glycoprotein (Env). By blocking the interaction between HIV-1 and the host cell's CD4 receptor, VRC01LS inhibits viral entry. It holds potential for research in HIV-1 infection.</p>Forma y color:Odour LiquidDitiocarb
CAS:<p>Ditiocarb speeds up copper cementation, cuts HIV risk, and boosts high-risk breast cancer immunoresearch.</p>Fórmula:C5H11NS2Forma y color:SolidPeso molecular:149.28HIV protease-IN-1
CAS:<p>HIV protease-IN-1 (compound 1·succinate), a potent non-peptidic inhibitor of HIV protease, is utilized for AIDS research [1].</p>Fórmula:C39H40ClF7N10O7Forma y color:SolidPeso molecular:929.24Epicoccone B
CAS:<p>Epicoccone B from C. globosum has DPPH scavenging (IC50=10.8μM) and α-glucosidase inhibition (IC50=27.3μM), also anti-HIV.</p>Fórmula:C9H8O5Forma y color:SolidPeso molecular:196.16Bictegravir Sodium
CAS:<p>Bictegravir Sodium is an HIV-1 integrase inhibitor with 7.5 nM IC50, offering strong, selective anti-HIV effects and minimal toxicity.</p>Fórmula:C21H17F3N3NaO5Pureza:99.97%Forma y color:SolidPeso molecular:471.36TAT peptide
<p>TAT peptide, a CPP, delivers molecules into cells by traversing membrane barriers using aa49-57 of TAT protein.</p>Fórmula:C65H124N34O15Pureza:98%Forma y color:SolidPeso molecular:1621.91Peritassine A
CAS:<p>Peritassine A, an alkaloid derived from Tripterygium wilfordii Hook. f., exhibits anti-HIV properties.</p>Fórmula:C38H47NO18Forma y color:SolidPeso molecular:805.783Indoline
CAS:<p>Compound PDK0239, with CAS No. 496-15-1, is a fragment molecule that serves as an important scaffold for molecular linking, expansion, and modification. Compound PDK0239 provides a structural basis and research tool for the design and screening of novel drug candidates, and is commonly used in drug discovery, drug synthesis, and related research.</p>Fórmula:C8H9NForma y color:Clear To Yellow LiquidPeso molecular:119.16Lopinavir Metabolite M-1
CAS:<p>Lopinavir Metabolite M-1, derived from Lopinavir, inhibits HIV protease (Ki=0.7 pM) and shows antiviral activity in vitro.</p>Fórmula:C37H46N4O6Forma y color:SolidPeso molecular:642.78Hypoglaunine D
CAS:<p>Hypoglaunine D, an anti-HIV analogue of Triptonine B, inhibits HIV in H9 cells with an EC50 of 22 μg/ml.</p>Fórmula:C41H47NO19Forma y color:SolidPeso molecular:857.81HIV-1 protease-IN-4
HIV-1 protease-IN-4, a prodrug of atazanavir, delivers 5x AUC & 67x C24 compared to atazanavir.Fórmula:C48H69N7O11Forma y color:SolidPeso molecular:920.1(+)-Carbovir triphosphate
CAS:<p>(+)-Carbovir triphosphate, Abacavir's active metabolite, studied for HIV-1 resistance and inhibition mechanisms.</p>Fórmula:C11H16N5O11P3Forma y color:SolidPeso molecular:487.19HIV-1 protease-IN-14
<p>HIV-1protease-IN-14 (compound 5ae) is an effective inhibitor of HIV-1protease, exhibiting Ki values of 0.28 nM and 56.9 nM against WTHIV-1PR and R41THIV-1PR, respectively. This compound also demonstrates low cytotoxicity.</p>Forma y color:Odour SolidEnfuvirtide
CAS:Enfuvirtide (INN) is an HIV fusion inhibitor, the first of a class of antiretroviral drugs used in combination therapy for the treatment of HIV-1 infection.Fórmula:C204H301N51O64Pureza:98%Forma y color:White To Off-White Amorphous SolidPeso molecular:4491.945
