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Receptores acoplados de proteína G y receptores 7-TM

Receptores acoplados de proteína G y receptores 7-TM

Los receptores acoplados a proteínas G (GPCR) y los receptores de 7 dominios transmembrana (7-TM) son una gran familia de proteínas de membrana que desempeñan un papel clave en la comunicación celular y la transducción de señales. Estos receptores están involucrados en una amplia gama de procesos fisiológicos, incluyendo la percepción sensorial, la respuesta inmunitaria y la regulación hormonal. Los GPCR son objetivos principales en el descubrimiento de fármacos, lo que los convierte en esenciales para la investigación en farmacología y medicina. En CymitQuimica, ofrecemos una amplia selección de reactivos y compuestos de alta calidad relacionados con los GPCR y los receptores 7-TM para apoyar su investigación y esfuerzos en el desarrollo de medicamentos.

Se han encontrado 5973 productos para "Receptores acoplados de proteína G y receptores 7-TM".

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productos por página.
  • MK-0249 FA


    MK-0249 FA is an H3 inverse agonist that can be used to study attention-deficit, hyperactivity disorder and cognitive disorders in adults.
    Fórmula:C24H26F3N3O4
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:477.48

    Ref: TM-T12054L

    1mg
    175,00€
    5mg
    745,00€
    10mg
    982,00€
    25mg
    1.485,00€
    50mg
    2.008,00€
  • YNT-185

    CAS:
    YNT-185 is a nonpeptide, selective agonist of the orexin type-2 receptor (OX2R), demonstrating EC50 values of 0.028 μM and 2.75 μM for OX2R and OX1R,
    Fórmula:C33H37N5O5S
    Pureza:99.67%
    Forma y color:Solid
    Peso molecular:615.74

    Ref: TM-T39229

    1mg
    63,00€
    5mg
    137,00€
    10mg
    215,00€
    25mg
    430,00€
    50mg
    695,00€
    100mg
    945,00€
  • Blonanserin

    CAS:
    Blonanserin (AD-5423), approved in Japan (2008), is an atypical antipsychotic with fewer side effects like EPS, sedation, or hypotension.
    Fórmula:C23H30FN3
    Pureza:99.85% - 99.99%
    Forma y color:Solid
    Peso molecular:367.50

    Ref: TM-T1180

    1mL*10mM (DMSO)
    33,00€
    25mg
    49,00€
    50mg
    66,00€
    100mg
    93,00€
  • Dimenhydrinate

    CAS:
    Dimenhydrinate (Vomex A) is an ethanolamine and histamine antagonist with anti-allergic activity.
    Fórmula:C24H28ClN5O3
    Pureza:99.57% - 99.77%
    Forma y color:Solid
    Peso molecular:469.96

    Ref: TM-T0298

    1mL*10mM (DMSO)
    33,00€
    100mg
    34,00€
    200mg
    49,00€
    500mg
    73,00€
    1g
    92,00€
  • Azatadine dimaleate

    CAS:
    Azatadine dimaleate (SCH10649) is an inhibitor for histamine(IC50=6.5 nM) and cholinergic(IC50=10 nM).
    Fórmula:C28H30N2O8
    Pureza:99.7% - >99.99%
    Forma y color:Solid
    Peso molecular:522.55

    Ref: TM-T0236

    50mg
    40,00€
    100mg
    62,00€
    200mg
    89,00€
  • Levosulpiride

    CAS:
    Levosulpiride (S-(-)-Sulpiride) is the (S)-enantiomer of sulpiride, which is a D2 receptor antagonist, an atypical antipsychotic drug of the benzamide class.
    Fórmula:C15H23N3O4S
    Pureza:98.20% - 99.88%
    Forma y color:White Solid
    Peso molecular:341.43

    Ref: TM-T1211

    25mg
    34,00€
    50mg
    42,00€
    100mg
    52,00€
    1mL*10mM (DMSO)
    52,00€
    500mg
    105,00€
    1g
    152,00€
  • Fluparoxan hydrochloride

    CAS:
    Fluparoxan hydrochloride is a highly selective and potent α2-adrenoceptor antagonist for the prevention, amelioration or treatment of neurodevelopmental
    Fórmula:C10H11ClFNO2
    Pureza:99.98%
    Forma y color:Solid
    Peso molecular:231.65

    Ref: TM-T77565

    1mg
    109,00€
    5mg
    233,00€
    10mg
    344,00€
    25mg
    532,00€
    50mg
    735,00€
    100mg
    982,00€
  • Indacaterol maleate

    CAS:
    Indacaterol maleate (QAB149) is an ultra-long-acting β-adrenoceptor agonist.
    Fórmula:C28H32N2O7
    Pureza:99.03% - 99.67%
    Forma y color:Solid
    Peso molecular:508.56

    Ref: TM-T1239

    10mg
    34,00€
    25mg
    50,00€
    1mL*10mM (DMSO)
    52,00€
    50mg
    71,00€
    100mg
    92,00€
    200mg
    138,00€
  • CYM 50769

    CAS:
    CYM 50769 is a neuropeptide W/B receptor 1 (NPBWR1, GPR7) antagonist(IC50 = 0.12 μM).
    Fórmula:C24H17ClN2O3
    Pureza:98% - 99.08%
    Forma y color:Solid
    Peso molecular:416.86

    Ref: TM-T22702

    1mg
    49,00€
    5mg
    92,00€
    10mg
    166,00€
    25mg
    358,00€
    50mg
    530,00€
    100mg
    758,00€
  • AH 6809

    CAS:
    AH 6809 blocks EP1, EP2, EP3, DP receptors (Ki: 1217-1597 nM human, 350 nM mouse EP2).
    Fórmula:C17H14O5
    Pureza:97.59%
    Forma y color:Solid
    Peso molecular:298.29

    Ref: TM-T14148

    1mg
    34,00€
    5mg
    63,00€
    1mL*10mM (DMSO)
    67,00€
    10mg
    92,00€
    25mg
    165,00€
    50mg
    250,00€
    100mg
    401,00€
    200mg
    580,00€
  • Salmeterol

    CAS:
    Salmeterol (GR33343X) is a long-acting agonist of beta2-adrenergic receptor (beta 2AR) used for treatment ofasthma.
    Fórmula:C25H37NO4
    Pureza:99.2% - 99.9%
    Forma y color:Solid
    Peso molecular:415.57

    Ref: TM-T12829

    5mg
    52,00€
    1mL*10mM (DMSO)
    58,00€
    10mg
    84,00€
    25mg
    145,00€
    50mg
    259,00€
  • (3aR,9aR)-Fluparoxan

    CAS:
    (3aR,9aR)-Fluparoxan is a highly selective and potent adrenergic receptor α2B antagonist for the prevention, amelioration or treatment of neurodevelopmental
    Fórmula:C10H10FNO2
    Pureza:97.82%
    Forma y color:Solid
    Peso molecular:195.19

    Ref: TM-T77566

    1mg
    175,00€
    5mg
    388,00€
    10mg
    572,00€
    25mg
    888,00€
    50mg
    1.224,00€
    100mg
    1.648,00€
    500mg
    3.312,00€
  • Antazoline hydrochloride

    CAS:
    Antazoline hydrochloride (Phenazoline hydrochloride), a first-generation antihistamine, can bind to the histamine H1 receptor and block the action of endogenous
    Fórmula:C17H19N3·HCl
    Pureza:98% - 99.53%
    Forma y color:White Solid
    Peso molecular:301.82

    Ref: TM-T0092

    1g
    33,00€
    1mL*10mM (DMSO)
    33,00€
  • Roxatidine Acetate hydrochloride

    CAS:
    Roxatidine Acetate hydrochloride (HOE 760) is a specific and competitive histamin H2-receptor antagonist. Roxatidine inhibits gastric acid secretion.
    Fórmula:C19H29ClN2O4
    Pureza:99.49%
    Forma y color:Solid
    Peso molecular:384.9

    Ref: TM-T0157

    1mL*10mM (DMSO)
    33,00€
    200mg
    33,00€
  • Serazapine

    CAS:
    Serazapine is a highly specific serotonin (5-HT2) binding inhibitor with anxiolytic activity for the treatment of anxiety disorders.
    Fórmula:C22H23N3O2
    Pureza:99.29% - 99.97%
    Forma y color:White Solid
    Peso molecular:361.44

    Ref: TM-T68142

    1mg
    92,00€
    5mg
    203,00€
    10mg
    294,00€
    25mg
    447,00€
    50mg
    612,00€
    100mg
    820,00€
    200mg
    1.108,00€
  • Cefaclor monohydrate

    CAS:
    Cefaclor monohydrate (Cefaclorum) is a beta-lactam, second-generation cephalosporin antibiotic with bactericidal activity.
    Fórmula:C15H16ClN3O5S
    Pureza:97.36% - 99.9%
    Forma y color:White Solid
    Peso molecular:385.82

    Ref: TM-T1495

    500mg
    46,00€
    1g
    58,00€
    5g
    124,00€
  • Trazodone hydrochloride

    CAS:
    Trazodone hydrochloride (Trazodone HCl) is a serotonin uptake inhibitor that is used as an antidepressive agent.
    Fórmula:C19H23Cl2N5O
    Pureza:99.5% - 99.52%
    Forma y color:Solid
    Peso molecular:408.33

    Ref: TM-T1619

    1mL*10mM (DMSO)
    33,00€
    500mg
    46,00€
    1g
    58,00€
    5g
    128,00€
    10g
    178,00€
  • Aripiprazole

    CAS:
    Aripiprazole (OPC-14597) is a piperazine/quinolone antipsychotic, partial agonist at 5-HT1A/D2, and antagonist at 5-HT2A.
    Fórmula:C23H27Cl2N3O2
    Pureza:99.43% - 99.62%
    Forma y color:White Solid
    Peso molecular:448.39

    Ref: TM-T1566

    10mg
    33,00€
    25mg
    34,00€
    50mg
    47,00€
    1mL*10mM (DMSO)
    52,00€
    100mg
    60,00€
    500mg
    96,00€
    1g
    126,00€
  • Ticlopidine hydrochloride

    CAS:
    Ticlopidine hydrochloride (Ticlodix) is an effective inhibitor of platelet aggregation commonly used in the placement of STENTS in CORONARY ARTERIES.
    Fórmula:C14H15Cl2NS
    Pureza:99.83% - 99.97%
    Forma y color:White Powder
    Peso molecular:300.25

    Ref: TM-T0362

    200mg
    33,00€
    1mL*10mM (DMSO)
    34,00€
  • Ondansetron hydrochloride dihydrate

    CAS:
    Ondansetron hydrochloride dihydrate (GR 38032) is a competitive serotonin type 3 receptor antagonist,which has reported anxiolytic and neuroleptic properties.
    Fórmula:C18H19N3O·HCl·2H2O
    Pureza:99.92%
    Forma y color:Solid
    Peso molecular:365.86

    Ref: TM-T1478

    25mg
    34,00€
    50mg
    42,00€
    100mg
    49,00€
    500mg
    90,00€